Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YKPIWOGXCSQLFH
|
7.7 | IC50 | 2 | — | |
ZYDQWWRARYHYHC
|
7.7 | IC50 | 2 | — | |
BEYDVFUQKWNRPT
|
7.7 | IC50 | 3 | — | |
DTMZXHDQZQLTHA
|
7.7 | Ki | 21 | — | |
DYSRECIVMDGUQU
|
7.7 | Ki | 29 | — | |
FBWWNLBZZFVRQY
|
7.7 | Ki | 4 | — | |
HKECWLZKPZHUND
|
7.7 | IC50 | 8 | — | |
KGCRKAITGGKXHI
|
7.7 | Ki | 5 | — | |
OROAFGSTGRDOFR
|
7.7 | Ki | 6 | — | |
OTVFVCDVXUJJLL
|
7.7 | IC50 | 2 | — | |
OYNBEDDKSIPEQC
|
7.7 | IC50 | 3 | — | |
PFSOTOJNKFKFFB
|
7.7 | IC50 | 2 | — | |
PNKAKGKYAQLZIY
|
7.7 | IC50 | 4 | — | |
POXGYBNJJBFCDU
|
7.7 | IC50 | 2 | — | |
QOJSERWVVHZZPL
|
7.7 | IC50 | 3 | — | |
QTSSRGDJHWGQHI
|
7.7 | IC50 | 2 | — | |
UAQJVFADAYIBGC
|
7.7 | Ki | 23 | — | |
UXUQVXDYXKMCGA
|
7.7 | Ki | 21 | — | |
WZBMMJKAHHOXRG
|
7.7 | Ki | 16 | — | |
XVHXYPREJYNIQE
|
7.7 | IC50 | 2 | — | |
NDIUYMHNCUTVGE
|
7.7 | Ki | 25 | — | |
OVTRGRMOTBJXKF
|
7.7 | IC50 | 2 | — | |
OYPIIVNTYVSCNV
|
7.7 | IC50 | 4 | — | |
FQCPPVRJPILDIK
|
7.7 | IC50 | 12 | — | |
LDHIZDYQCCLGRS
|
7.7 | IC50 | 2 | — | |
BSGQUBKLPKMFRV
|
7.6 | IC50 | 2 | — | |
DMGXNXJIKAWOHP
|
7.6 | Ki | 6 | — | |
OVPNQJVDAFNBDN
|
7.6 | Kd | 44 | Yes | |
IBRKDXNYRBZUGZ
|
7.6 | IC50 | 2 | — | |
JYCUVOXSZBECAY
|
7.6 | Ki | 6 | Yes | |
KGIDFBNHNUZTPT
|
7.6 | IC50 | 3 | — | |
AWJPVXSHMIELNJ
|
7.6 | Ki | 23 | — | |
GWJHMRBQEUHFOC
|
7.6 | Ki | 42 | — | |
JJJSCYSPSKBQAX
|
7.6 | Ki | 34 | — | |
KTNYZVYVXUQVCW
|
7.6 | IC50 | 2 | — | |
KYACBMRLQMEIAI
|
7.6 | Ki | 30 | — | |
LDTNZBKHOOMMNR
|
7.6 | IC50 | 2 | — | |
RXVOXSGTUROJOL
|
7.6 | Ki | 11 | — | |
UWQBVYXTLXNIOO
|
7.6 | Ki | 10 | — | |
KQWTXAWKBUUOMU
|
7.6 | IC50 | 20 | Yes | |
QWDGTUJNIPWNGT
|
7.6 | IC50 | 2 | — | |
MFXBFPQUOABRHL
|
7.6 | IC50 | 2 | — | |
PSLRGVBAUBPLDY
|
7.6 | IC50 | 2 | — | |
SSAQMAUQLFVZJJ
|
7.6 | IC50 | 2 | — | |
UDIUKSLSDVCBFN
|
7.6 | IC50 | 2 | — | |
GPJWYYLEVMBAKU
|
7.6 | IC50 | 2 | — | |
FSCLZTCYWFNGON
|
7.5 | IC50 | 4 | — | |
IGCCKDSIYZVXOF
|
7.5 | IC50 | 2 | — | |
KYFJPYWXCUCRPE
|
7.5 | IC50 | 2 | — | |
OUSFTKFNBAZUKL
|
7.5 | Kd | 58 | Yes |