Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AXWDQRXGOKDXJT
|
7.9 | IC50 | 6 | — | |
KQMHAQZHLWKKPG
|
7.9 | IC50 | 2 | — | |
LQLBWZJHRARWDB
|
7.9 | IC50 | 6 | — | |
NKUNFNVAHJNALA
|
7.9 | IC50 | 2 | — | |
UEZWIGHGLPNICR
|
7.9 | IC50 | 2 | — | |
ZCMFNKZSIWNHEU
|
7.9 | IC50 | 2 | — | |
JJTYLBBKGQOISV
|
7.9 | Ki | 15 | — | |
KHGPYYFCIAISBU
|
7.9 | Ki | 31 | — | |
ZAEAGGGBPKOFMY
|
7.9 | Ki | 3 | — | |
ILMHDRGZABQLEW
|
7.9 | Ki | 5 | — | |
LGYPOTRKBGDLHM
|
7.9 | IC50 | 2 | — | |
QEQDTPMQMKDYJW
|
7.9 | IC50 | 3 | — | |
UIZJZUMESFGZFJ
|
7.9 | IC50 | 2 | — | |
UJFAOQFICNRWOP
|
7.9 | IC50 | 4 | — | |
UZWDCWONPYILKI
|
7.9 | Kd | 47 | — | |
YWMJEKUKEKXNSA
|
7.9 | IC50 | 2 | — | |
QQUXFYAWXPMDOE
|
7.9 | IC50 | 31 | — | |
MLBFCSJJRVBMRM
|
7.9 | IC50 | 2 | — | |
DQYDZCRLDYVZKY
|
7.8 | IC50 | 5 | — | |
GPDQWQAEPILOQK
|
7.8 | IC50 | 2 | — | |
HDONVKMMRZKRCC
|
7.8 | IC50 | 2 | — | |
BDRSCIWOUKYOAH
|
7.8 | IC50 | 2 | — | |
CBQODTLCGVMLQR
|
7.8 | IC50 | 2 | — | |
ILMCPEAFWSFNIE
|
7.8 | IC50 | 2 | — | |
RMCVVJFCJYYDDO
|
7.8 | IC50 | 2 | — | |
RXQXACYMRVINQU
|
7.8 | IC50 | 5 | — | |
WMOHFUHNWBHUKZ
|
7.8 | IC50 | 2 | — | |
ZAGLHDIYLNNWJL
|
7.8 | IC50 | 2 | — | |
FPLAQCFCGCSDRB
|
7.8 | Ki | 4 | — | |
HKSZLNNOFSGOKW
|
7.8 | Ki | 118 | — | |
JUTMUSMWCYHBGU
|
7.8 | Ki | 3 | — | |
JXMYIDZREHNPDO
|
7.8 | Ki | 19 | — | |
MHWHPWMWKYXCRJ
|
7.8 | Ki | 32 | — | |
NHEQNFWGPSKRMJ
|
7.8 | Ki | 7 | — | |
PGJTVDLNKJZVEU
|
7.8 | IC50 | 2 | — | |
SNFNRLLKLGNUTL
|
7.8 | IC50 | 2 | — | |
TYNCGTPANDPODX
|
7.8 | IC50 | 4 | — | |
XSDJOIOVIMPMHD
|
7.8 | Ki | 44 | — | |
VQLWTLFHWAMQQX
|
7.8 | IC50 | 2 | — | |
WYBRFXSHAXWYIZ
|
7.8 | IC50 | 3 | — | |
XOXJFSRAOYMCPS
|
7.8 | IC50 | 2 | — | |
JCSGFHVFHSKIJH
|
7.8 | IC50 | 2 | — | |
QBWPHVZDFQYVMW
|
7.8 | IC50 | 2 | — | |
ZXOPGTSQJRRYHF
|
7.8 | IC50 | 4 | — | |
UJSQNTWNRHAOBC
|
7.7 | IC50 | 2 | — | |
AXMWKXSPCWMKHN
|
7.7 | IC50 | 2 | — | |
CRZIGHVWJFDSFR
|
7.7 | IC50 | 5 | — | |
MBDKLKUFQIFGCR
|
7.7 | IC50 | 2 | — | |
VCAIGCKZZLIJFZ
|
7.7 | IC50 | 2 | — | |
VCJCBOHBQULJNM
|
7.7 | IC50 | 2 | — |