Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RKUKAACYUCUJEE
|
8.2 | Ki | 58 | — | |
WLLUQXGGNFUQGM
|
8.2 | Ki | 4 | — | |
ZFIMJZNGNMRTHA
|
8.2 | IC50 | 2 | — | |
LFAHWMOZPVCJAY
|
8.2 | Kd | 8 | — | |
NUQDMQZYZIYAFS
|
8.2 | IC50 | 2 | — | |
MDJOZDXRTJEZTG
|
8.2 | IC50 | 2 | — | |
PHEGERKTBZOREL
|
8.2 | IC50 | 2 | — | |
DFHRUTWHYJCTMH
|
8.2 | IC50 | 4 | — | |
DTTIISYOYISNJH
|
8.2 | IC50 | 3 | — | |
FMBUJPKXYCHTCB
|
8.2 | IC50 | 2 | — | |
FQQWTITYZMFQRJ
|
8.2 | IC50 | 2 | — | |
GUASZRAHLZIIEE
|
8.2 | IC50 | 2 | — | |
GVYKLTFFLMMUEN
|
8.2 | IC50 | 3 | — | |
LCFKIGOGPZGTMF
|
8.2 | IC50 | 2 | — | |
MDZCSIDIPDZWKL
|
8.2 | IC50 | 2 | — | |
WYZXNPCPQURARS
|
8.2 | IC50 | 2 | — | |
XLSYZSRXVVCHLS
|
8.2 | Kd | 48 | — | |
ZANIFKRQUQTFLO
|
8.2 | IC50 | 2 | — | |
QSGKPYRFWJINEH
|
8.1 | IC50 | 12 | — | |
VRHHAMWTRSVIEX
|
8.1 | Kd | 5 | — | |
FSDWOHNRBITTOF
|
8.1 | IC50 | 2 | — | |
AQGNHMOJWBZFQQ
|
8.1 | IC50 | 2 | — | |
BCTHVHCUWYGJKE
|
8.1 | IC50 | 4 | — | |
HATZMBUGJIBSIP
|
8.1 | IC50 | 2 | — | |
IHKGTVZWLMITRF
|
8.1 | IC50 | 3 | — | |
LYNBNVBMAGDJRW
|
8.1 | Ki | 81 | — | |
QIEFQCNWXLTEAU
|
8.1 | IC50 | 4 | — | |
RAOQCDVBADRLDK
|
8.1 | IC50 | 2 | — | |
ZKLJKKASNXVQBZ
|
8.1 | Ki | 27 | — | |
QJGILMHLEDGHMD
|
8.1 | IC50 | 2 | — | |
PKEPHTDOSDZCGK
|
8.1 | IC50 | 2 | — | |
VREUVWWSISDHAV
|
8.1 | IC50 | 2 | — | |
DNCXPYGCTRGWJY
|
8.1 | IC50 | 3 | — | |
DSHMUQCEERJXOA
|
8.1 | IC50 | 2 | — | |
QMPGEDNNYDQBID
|
8.1 | IC50 | 2 | — | |
RQFYFNAGNBUGFC
|
8.1 | IC50 | 3 | — | |
WCCYEJYTLNWYCC
|
8.1 | IC50 | 9 | — | |
ZSSPKMADGVCZPK
|
8.1 | IC50 | 2 | — | |
RYBNARZBIXTFJS
|
8.0 | IC50 | 9 | — | |
RYBNARZBIXTFJS
|
8.0 | IC50 | 9 | — | |
KCKXYZOBGBJZEG
|
8.0 | Ki | 36 | — | |
MENDIXKFTXYTHJ
|
8.0 | IC50 | 2 | — | |
MJCKUHBSAUHVJE
|
8.0 | Ki | 4 | — | |
MVUKVIIMDNACQW
|
8.0 | IC50 | 2 | — | |
SAZAEFLODZISSG
|
8.0 | IC50 | 4 | — | |
VEZQCXWMPWTPJL
|
8.0 | Ki | 5 | — | |
FVWBAHQOQFMWPU
|
8.0 | IC50 | 2 | — | |
SVEYNURJTZJXIG
|
8.0 | IC50 | 2 | — | |
YDELNSXADYPQGS
|
8.0 | IC50 | 15 | Yes | |
WUTXOFQDICTONV
|
7.9 | IC50 | 3 | — |