Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XFTCKLNUSFOJAU
|
8.4 | IC50 | 3 | Yes | |
YRRRHSNOXWKVDL
|
8.4 | IC50 | 5 | — | |
ZRQXCQXWTLVASO
|
8.4 | Ki | 36 | — | |
NDFXSHIIGXVOKT
|
8.4 | IC50 | 2 | — | |
HVEXJKQESNIDLM
|
8.4 | Kd | 10 | — | |
KUAAAOFBHQLFAD
|
8.4 | IC50 | 2 | — | |
HFCIUXUUWFLDQF
|
8.4 | IC50 | 2 | — | |
PQOGJESGKNBNIP
|
8.4 | IC50 | 2 | — | |
NZMAVPMPPORZNT
|
8.3 | IC50 | 2 | — | |
TVOFBUNUDWXBSZ
|
8.3 | IC50 | 2 | — | |
WQUSEPBJMLQZJS
|
8.3 | IC50 | 2 | — | |
YLVVCSCPLBFQFV
|
8.3 | IC50 | 3 | — | |
MHBKUCFDNISLNC
|
8.3 | IC50 | 2 | — | |
ODMDEVGMHNNVJK
|
8.3 | IC50 | 2 | — | |
OLKIZDOBETVOFT
|
8.3 | IC50 | 2 | — | |
FHCSBLWRGCOVPT
|
8.3 | Ki | 2 | — | |
AKYXUYKRNRLTAG
|
8.3 | IC50 | 2 | — | |
BTEDJGZRXQWYSZ
|
8.3 | IC50 | 2 | — | |
CJJKTILOCMYOOH
|
8.3 | Ki | 3 | — | |
DDLZLOKCJHBUHD
|
8.3 | IC50 | 23 | — | |
GJWWXUHHULUCNL
|
8.3 | IC50 | 3 | — | |
KPVCGFZWGAYXMV
|
8.3 | IC50 | 7 | — | |
MLJSTZOBGVWFLQ
|
8.3 | IC50 | 2 | — | |
NJFATVGYCPEPCY
|
8.3 | IC50 | 2 | — | |
NSDIHUXUFJHXRA
|
8.3 | Ki | 11 | — | |
OLOJSTRISMGUEK
|
8.3 | IC50 | 5 | — | |
PPIPFZAGLGRLCJ
|
8.3 | IC50 | 2 | — | |
SWZAXOLMRPWGRZ
|
8.3 | IC50 | 2 | — | |
UJNZJFWHEHUMNG
|
8.3 | IC50 | 2 | — | |
WZEMTZHNQZDUFC
|
8.3 | IC50 | 2 | — | |
XFRYMFRHCLWJQY
|
8.3 | Ki | 3 | — | |
YMOZGQKWFWKZJV
|
8.3 | IC50 | 2 | — | |
ZJQQJUGCEKHDGB
|
8.3 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.3 | IC50 | 408 | — | |
UVTJZQHSPPYGDG
|
8.3 | IC50 | 3 | — | |
LJUDIYPNWBIDNH
|
8.3 | IC50 | 2 | — | |
OAUZYEUYSSRWDJ
|
8.2 | IC50 | 2 | — | |
QWJULXPIBCHMDX
|
8.2 | IC50 | 2 | — | |
LYVOHPYWGZFHPE
|
8.2 | IC50 | 2 | — | |
BGVFZHIFEQILLB
|
8.2 | IC50 | 2 | — | |
BRBGAJDUHBVSLV
|
8.2 | IC50 | 2 | — | |
JTXGWTJLZDKHJQ
|
8.2 | IC50 | 8 | — | |
LOLPPWBBNUVNQZ
|
8.2 | Kd | 97 | Yes | |
WXZHKVLOSBCWDY
|
8.2 | IC50 | 2 | — | |
CYLGCMABIBXHIQ
|
8.2 | Ki | 16 | — | |
FGLPGUCHBHILNS
|
8.2 | Ki | 10 | — | |
IMHKMKWSWHFKTM
|
8.2 | Ki | 13 | — | |
KDUHTFCGEYDKBT
|
8.2 | IC50 | 3 | — | |
PVIMTNAWPMEBAK
|
8.2 | IC50 | 2 | — | |
QTTYXMRMIOCNGZ
|
8.2 | Ki | 3 | — |