Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HHSIUHRARDLCPM
|
8.7 | IC50 | 5 | Yes | |
NEXAGSGRVBOFPO
|
8.7 | IC50 | 2 | — | |
QAFFAZAVQKPMKM
|
8.7 | IC50 | 2 | — | |
USLKSBWEDVVGFB
|
8.7 | IC50 | 2 | — | |
VJTITFHQYIFDAU
|
8.7 | IC50 | 2 | — | |
WJCNROIVPXENEU
|
8.7 | IC50 | 2 | — | |
HVIKGCPTKADTTQ
|
8.7 | IC50 | 2 | — | |
SSTMOSQZONYWBG
|
8.7 | IC50 | 2 | — | |
XEFFULWZVBHILM
|
8.7 | IC50 | 2 | — | |
IQZQCERNFAXKFQ
|
8.7 | IC50 | 3 | — | |
XAPPKVUCFSPXNL
|
8.7 | IC50 | 2 | — | |
DZUXTQCYZWQAFQ
|
8.6 | IC50 | 2 | — | |
WKJFLAJZSWRICW
|
8.6 | IC50 | 2 | — | |
FFZJQKHNKKPZAH
|
8.6 | IC50 | 2 | — | |
UXFHOMCAQUWAHI
|
8.6 | IC50 | 3 | — | |
XVPJMVOASKOHIR
|
8.6 | IC50 | 2 | — | |
ZFHYCZOXNRBREO
|
8.6 | IC50 | 2 | — | |
GBGNHUZQFPYZRM
|
8.5 | IC50 | 2 | — | |
QKSJQYPOAQOCOW
|
8.5 | IC50 | 2 | — | |
QOWGEVKZOPOWLW
|
8.5 | IC50 | 2 | — | |
RQQZTHUGRVIEQX
|
8.5 | IC50 | 2 | — | |
WYQFGFSCDJKYOY
|
8.5 | IC50 | 2 | — | |
YWMJEKUKEKXNSA
|
8.5 | IC50 | 2 | — | |
DKVBUSZSQFOSNU
|
8.5 | IC50 | 2 | — | |
FLEAYYMORDPWAJ
|
8.5 | Ki | 90 | — | |
KMXBENJAVFIELJ
|
8.5 | IC50 | 3 | — | |
KSMGIZGHYKGTPR
|
8.5 | IC50 | 2 | — | |
NOZZORCJVZKEHP
|
8.5 | IC50 | 2 | — | |
OWNFHHCNBOIRTE
|
8.5 | IC50 | 2 | — | |
WCCWJPDOCPHFPS
|
8.5 | IC50 | 2 | — | |
KLFHGYKHZZHOKY
|
8.5 | IC50 | 2 | — | |
NCJPNQVCPACJMH
|
8.5 | IC50 | 2 | — | |
JKVBLFAUDIBMEH
|
8.5 | IC50 | 3 | — | |
KQPIZIMTVIHVTG
|
8.5 | IC50 | 2 | — | |
PSPRVPOUXLRHOH
|
8.5 | IC50 | 2 | — | |
FAJGIEVMPKNFTN
|
8.4 | IC50 | 2 | — | |
QNUACCMSCPINIY
|
8.4 | IC50 | 2 | — | |
UWQKULXATKCNBV
|
8.4 | IC50 | 4 | — | |
AYSFEKIVJXIJTM
|
8.4 | IC50 | 8 | — | |
BAMRUHLBPZRRIX
|
8.4 | IC50 | 2 | — | |
CJOZQFXWSCXETF
|
8.4 | IC50 | 2 | — | |
DMFMPEWLXMKYKK
|
8.4 | IC50 | 4 | — | |
GCBJDOWIQHMCMR
|
8.4 | Ki | 84 | — | |
GCYXEGSPUDSZJY
|
8.4 | Ki | 82 | — | |
HJYHJYGXRBYDIG
|
8.4 | Ki | 23 | — | |
JIQRMBNAYWCUEG
|
8.4 | IC50 | 3 | — | |
KLSRELDSEJWOAS
|
8.4 | IC50 | 2 | — | |
LXVBELDBJGYFEM
|
8.4 | Ki | 20 | — | |
OLUKILHGKRVDCT
|
8.4 | IC50 | 44 | Yes | |
SOTUJQRAYBWHFK
|
8.4 | IC50 | 2 | — |