Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OPJUVNCYLAQSEB
|
6.0 | IC50 | 3 | — | |
PJUSCKOQLSMBPU
|
6.0 | IC50 | 2 | — | |
QGRUEQPBBBTRPN
|
6.0 | IC50 | 4 | — | |
QVNZKVACBBTKSL
|
6.0 | Ki | 38 | — | |
QZPFUALVXZAFDD
|
6.0 | Ki | 10 | — | |
SJLQDZDKTVBBLP
|
6.0 | Ki | 9 | — | |
UNVKXVCDLOLPJE
|
6.0 | Ki | 8 | — | |
UUWNXFJBBYAMDT
|
6.0 | Ki | 46 | — | |
XVVANFOECICSLK
|
6.0 | IC50 | 4 | — | |
ZGDYBJXDIXVTLV
|
6.0 | Ki | 54 | — | |
ZMNICSIMJSXCPI
|
6.0 | IC50 | 2 | — | |
ZVWRFVCNQOECJS
|
6.0 | Ki | 71 | — |