Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RMKWXWRSMUTBAX
|
6.1 | IC50 | 2 | — | |
WMVCBNJJXIOYAO
|
6.1 | IC50 | 4 | — | |
ALNFKLJYTICTCF
|
6.1 | IC50 | 4 | — | |
BZMBEQLYEPQGMX
|
6.1 | IC50 | 2 | — | |
CGELEDQBCPRRSA
|
6.1 | IC50 | 3 | — | |
DHVBTKDVRAXVKY
|
6.1 | IC50 | 3 | — | |
DMZBGGYSGOPZET
|
6.1 | IC50 | 4 | — | |
DATNVJMWIKFHGB
|
6.1 | IC50 | 4 | — | |
NVOVYOYDVUPVOA
|
6.1 | IC50 | 3 | — | |
QSXQMPVZQTYTNO
|
6.1 | IC50 | 2 | — | |
TZZQSURAGPGEIF
|
6.1 | IC50 | 2 | — | |
UPVVKGJGCKBECE
|
6.1 | IC50 | 2 | — | |
VTQGLZJCCQHUJG
|
6.1 | IC50 | 4 | — | |
ZSUZNPQSAQRXJP
|
6.1 | IC50 | 4 | — | |
FGSXBNALMJRFIO
|
6.1 | IC50 | 2 | — | |
GGARDPUFELXEBN
|
6.1 | IC50 | 4 | — | |
HPQZTEVMVAVGJO
|
6.1 | Kd | 5 | — | |
NWBMEZSCKMLUTH
|
6.0 | IC50 | 3 | — | |
USBKPWRTJAXTBS
|
6.0 | IC50 | 16 | Yes | |
YGAUGCRQWVWVJK
|
6.0 | IC50 | 4 | — | |
ZDNTZQGZVGAPGQ
|
6.0 | IC50 | 4 | — | |
AZTMYWWWILJAKW
|
6.0 | Ki | 16 | Yes | |
MGVWPOMQHQAMAV
|
6.0 | IC50 | 3 | — | |
UPDASDRUBVHIJS
|
6.0 | IC50 | 4 | — | |
WRUIJSVPESNZTL
|
6.0 | IC50 | 3 | — | |
WVMANZPBOBRWCB
|
6.0 | IC50 | 9 | — | |
WCVCWAQJIQBEBG
|
6.0 | IC50 | 2 | — | |
ZYTXWIJBWLPWCM
|
6.0 | IC50 | 2 | — | |
IYFIEJRWVMLGOG
|
6.0 | Ki | 3 | — | |
OUROWULXWNIHIF
|
6.0 | IC50 | 4 | — | |
PAZVWIGCRYUCKP
|
6.0 | IC50 | 4 | — | |
ARAFZLNEXXVYMQ
|
6.0 | IC50 | 2 | — | |
BLQYVHBZHAISJM
|
6.0 | Ki | 54 | — | |
CBALVKLWBKZXIX
|
6.0 | IC50 | 3 | Yes | |
CRDNMYFJWFXOCH
|
6.0 | IC50 | 3 | Yes | |
DJUSDFVEBBYFFL
|
6.0 | Ki | 27 | — | |
FGWOKLCRQJXPPQ
|
6.0 | Ki | 14 | — | |
GHPFQRTVUDXWCC
|
6.0 | Ki | 35 | — | |
HDRKTFQABULLHE
|
6.0 | IC50 | 2 | — | |
HGILUFKJFSZULZ
|
6.0 | IC50 | 2 | — | |
HSMUWLLZAZCLHF
|
6.0 | Ki | 25 | — | |
IAEAEWGHRXXLML
|
6.0 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JCTPJYZESAMIGH
|
6.0 | Ki | 2 | — | |
JXFASNVVYCKOKY
|
6.0 | IC50 | 2 | — | |
LWBSSNRDDDFHSH
|
6.0 | Ki | 9 | — | |
MIJMZVTYIXYSDK
|
6.0 | Ki | 4 | — | |
MJLKHAZEWYICMC
|
6.0 | Ki | 4 | — | |
MKRBAPNEJMFMHU
|
6.0 | IC50 | 2 | — | |
NRZYTPAJGVTKIM
|
6.0 | Ki | 38 | — |