Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QJIKOODYNZFJFF
|
6.2 | IC50 | 3 | Yes | |
ZGEQEMOJHVPNTB
|
6.2 | IC50 | 2 | — | |
CUDLEXBIVZPJBU
|
6.2 | IC50 | 2 | — | |
CYKJKKJPMBDBAT
|
6.2 | IC50 | 4 | — | |
NCFYJNPNQNEPRW
|
6.2 | IC50 | 2 | — | |
OTKQTETZDVGXBV
|
6.2 | IC50 | 4 | — | |
VFQNGIVBLUWECA
|
6.2 | IC50 | 4 | — | |
HXAODWZKEDXMRG
|
6.2 | IC50 | 2 | — | |
IHCLBOWQUVPHBB
|
6.2 | IC50 | 3 | — | |
OBYOBQZFZXGFMP
|
6.2 | IC50 | 3 | — | |
PUDBISUVQGIKBD
|
6.2 | IC50 | 4 | — | |
RIQXNLIRMOIENV
|
6.2 | IC50 | 4 | — | |
AMKRSTDSNXNZMY
|
6.2 | IC50 | 4 | — | |
AWINCECFBWDQTG
|
6.2 | IC50 | 2 | — | |
LUNIPUNUORVVSN
|
6.2 | IC50 | 4 | — | |
ODRITQGYYWHQGM
|
6.2 | IC50 | 4 | — | |
OXYHNOHLBLUYKQ
|
6.2 | IC50 | 2 | — | |
RPWRQYOHVXHGBO
|
6.2 | IC50 | 4 | — | |
NZWOOXILJLNOHZ
|
6.2 | IC50 | 2 | — | |
QCPXWEFKAZRXTO
|
6.2 | IC50 | 3 | — | |
HMMIVTXSLFBBHC
|
6.1 | IC50 | 4 | — | |
IEUYALOEFWZLQN
|
6.1 | IC50 | 4 | — | |
KADSTJJZALTROR
|
6.1 | IC50 | 4 | — | |
WWCYPMCZKZTTME
|
6.1 | IC50 | 3 | — | |
FBCBXRZGCIFZMS
|
6.1 | IC50 | 2 | — | |
GFJIABMYYUGNEC
|
6.1 | IC50 | 6 | — | |
SKXNXCUQPDAUDR
|
6.1 | IC50 | 4 | — | |
XUIJEFBUBZVZFL
|
6.1 | IC50 | 4 | — | |
BIIVYFLTOXDAOV
|
6.1 | IC50 | 82 | Yes | |
DTGGTIWRYHDYPL
|
6.1 | IC50 | 4 | — | |
HAVMBPZPTGEWPJ
|
6.1 | IC50 | 4 | — | |
MFVIYYFPUOHHSN
|
6.1 | IC50 | 2 | — | |
ADGQZIUZHRRUQA
|
6.1 | IC50 | 2 | — | |
BIIVYFLTOXDAOV
|
6.1 | Ki | 31 | — | |
CLEGDJQQHUTCOW
|
6.1 | Ki | 43 | — | |
DJLORVJVWIBDME
|
6.1 | Ki | 24 | — | |
GCULKEKNSKDWPK
|
6.1 | IC50 | 2 | — | |
HWGZXYUOXGVACR
|
6.1 | Ki | 6 | — | |
HXDDWVMJYDULAZ
|
6.1 | Ki | 13 | — | |
KYUYCTKUEHJRCI
|
6.1 | Ki | 3 | — | |
MCBPNFWHHNJTGN
|
6.1 | Ki | 3 | — | |
OBHMNLIBIPFXCY
|
6.1 | Ki | 15 | — | |
PEXKNSGOEOREKM
|
6.1 | Ki | 13 | — | |
QEWSTOOMTBAUAG
|
6.1 | Ki | 17 | — | |
QMBBFTGBRHKNPS
|
6.1 | IC50 | 2 | — | |
VLRRDESRPRRNAD
|
6.1 | IC50 | 4 | — | |
WKWGFJFNCXAUEX
|
6.1 | Ki | 14 | Yes | |
XUFLBSMTYMFOQH
|
6.1 | Ki | 43 | — | |
YXUQWISLOFXNGN
|
6.1 | Ki | 16 | — | |
ZWVZORIKUNOTCS
|
6.1 | Ki | 69 | — |