Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZJXSGFKUKZTHTC
|
6.3 | IC50 | 2 | — | |
ZPUWOMDAGPEJAX
|
6.3 | IC50 | 2 | — | |
ZQWMZNLGINPQKE
|
6.3 | IC50 | 2 | — | |
ZWBGOXLJLHWSLZ
|
6.3 | IC50 | 2 | — | |
ZYUPXRAUFYTHFM
|
6.3 | IC50 | 2 | — | |
QIYPQJHMRBXGMO
|
6.2 | IC50 | 3 | Yes | |
AMUSCCPWKQVJSJ
|
6.2 | IC50 | 4 | — | |
JMJNNWUSBNQXNX
|
6.2 | IC50 | 2 | — | |
VXBAJLGYBMTJCY
|
6.2 | Kd | 34 | Yes | |
XMKRZXOTGFXMPH
|
6.2 | Kd | 5 | — | |
KFJCYTXMHLMPLW
|
6.2 | IC50 | 3 | — | |
AELWDCDMPFGKBB
|
6.2 | IC50 | 2 | — | |
BHPWHRPVZOWBAN
|
6.2 | IC50 | 2 | — | |
CUQPTMGVVQNXDH
|
6.2 | IC50 | 3 | — | |
KPFROWLXOVRLMN
|
6.2 | IC50 | 2 | — | |
MDWYQYJBHPWFDF
|
6.2 | IC50 | 2 | — | |
RYNPAHUWYURCCW
|
6.2 | IC50 | 6 | — | |
YHWHYCTUDCULTF
|
6.2 | IC50 | 4 | — | |
ZZUSFIPRLCGKQL
|
6.2 | IC50 | 4 | — | |
FKMYIGXYIAVMND
|
6.2 | IC50 | 3 | — | |
AIQDZMUPVYDVLB
|
6.2 | Ki | 48 | — | |
ASNQMAVHHGGQRB
|
6.2 | Ki | 14 | — | |
DFMCXVONDDGQIY
|
6.2 | Ki | 66 | — | |
DPEXRCOBPACFOO
|
6.2 | Ki | 36 | — | |
GWXPHWSUMLUDPO
|
6.2 | Ki | 11 | — | |
HHSVICUMCOBRPT
|
6.2 | Ki | 33 | — | |
JJGSOVIZOMZMCS
|
6.2 | Ki | 35 | — | |
JRVSFZKYQCETAH
|
6.2 | Ki | 19 | — | |
LRESELHEXSUQGE
|
6.2 | Ki | 10 | — | |
MBRVCJRFWYHVHE
|
6.2 | Ki | 9 | — | |
MDMCYZGIXLRATE
|
6.2 | IC50 | 4 | — | |
NERQMDXDVAZVNX
|
6.2 | Ki | 13 | — | |
NQLZEAYJHRFSCQ
|
6.2 | IC50 | 2 | — | |
ORUUEFDGYYTXAF
|
6.2 | Ki | 26 | — | |
RJZDECGDCKOHBV
|
6.2 | Ki | 70 | — | |
RTDSHUGNRVXRHN
|
6.2 | Ki | 51 | — | |
SDBOIBYRBWPIEL
|
6.2 | Ki | 31 | — | |
SODGZPDNROVASD
|
6.2 | Ki | 7 | — | |
SOVYWBOZOBVFLP
|
6.2 | Ki | 10 | — | |
TUJUZVJICDSNLY
|
6.2 | Ki | 19 | — | |
UMULGPSQNQMYNC
|
6.2 | Ki | 6 | — | |
VARGUUBRJVQGHK
|
6.2 | IC50 | 2 | — | |
WICLISNBDMGFST
|
6.2 | Ki | 10 | — | |
WYLVFMBGPRCDQF
|
6.2 | Ki | 14 | — | |
XGOUHJLISKQBDN
|
6.2 | IC50 | 4 | — | |
XTVULKIROSNNTG
|
6.2 | Ki | 29 | — | |
YYPKOMNJRZRWIC
|
6.2 | Ki | 26 | — | |
CHGLHVVJPSESHY
|
6.2 | IC50 | 4 | — | |
ICUDJSJDWWDBHD
|
6.2 | IC50 | 4 | — | |
PRIGRJPRGZCFAS
|
6.2 | IC50 | 13 | Yes |