Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BSHCILRNXWKQAL
|
9.0 | IC50 | 2 | — | |
IBMFJBCXKFJOPZ
|
9.0 | IC50 | 2 | — | |
JQWXFCIJCDFZKC
|
9.0 | IC50 | 2 | — | |
NRVJSTPJGPGYAF
|
9.0 | IC50 | 3 | — | |
QCOOCCREMZWFAR
|
9.0 | IC50 | 3 | — | |
SHJYLIJHYBXPEO
|
9.0 | IC50 | 3 | — | |
VVOFXGOUMCCSEE
|
9.0 | IC50 | 2 | — | |
ZLWLGUFTYZQJRI
|
9.0 | IC50 | 3 | — | |
ZYERPFJFBXNWOJ
|
9.0 | IC50 | 2 | — | |
QORWUQJNIZUKNZ
|
9.0 | IC50 | 2 | — | |
RKWKPORPODXCMU
|
9.0 | IC50 | 2 | — | |
UGFWJLOCVRHXSF
|
9.0 | IC50 | 3 | — | |
YUFANAGBOIXUIR
|
9.0 | IC50 | 2 | — | |
JCTOCSMGNIHFPY
|
8.9 | IC50 | 2 | — | |
IOLLWTLQKNSFOR
|
8.9 | IC50 | 2 | — | |
PEJAKFMXABEULA
|
8.9 | IC50 | 2 | — | |
VMOSNFMFQKNJPH
|
8.9 | IC50 | 3 | — | |
NWMPVMMGSHXANZ
|
8.9 | Ki | 58 | — | |
HPDNAGAYFYNQBT
|
8.9 | IC50 | 2 | — | |
INJUVNWOFHYUIN
|
8.9 | IC50 | 9 | Yes | |
CHZARGSIIZBMPM
|
8.9 | IC50 | 3 | — | |
ZBLGVBFQWBVFAW
|
8.9 | IC50 | 2 | — | |
NYNFHQSIJDCJQN
|
8.9 | IC50 | 2 | — | |
BXQCCJUQGHRPJT
|
8.8 | IC50 | 2 | — | |
HVZPHINNUZGJAZ
|
8.8 | IC50 | 3 | — | |
PTABJNPXSUGRKA
|
8.8 | IC50 | 2 | — | |
FQGBFYNAGSGZFG
|
8.8 | IC50 | 2 | — | |
HRJWTAWVFDCTGO
|
8.8 | IC50 | 13 | Yes | |
QGFZDGFJYXGLAW
|
8.8 | IC50 | 3 | — | |
RPGZQOOZHIEPJW
|
8.8 | Kd | 18 | — | |
RPGZQOOZHIEPJW
|
8.8 | Kd | 18 | — | |
BMXGRFBSHSEZOP
|
8.8 | IC50 | 5 | Yes | |
PQUQTSPOFKEROK
|
8.8 | IC50 | 3 | — | |
QNUBZASKWDMCAQ
|
8.8 | IC50 | 2 | — | |
QSEIHYMIZCHHFE
|
8.8 | IC50 | 2 | — | |
AMINIFOLNFYOOD
|
8.8 | IC50 | 2 | — | |
KVVPUEYLAZZLFF
|
8.8 | IC50 | 3 | — | |
UGOONUOQGNIMGO
|
8.8 | IC50 | 2 | — | |
UNNVCPOJKXBSGS
|
8.8 | IC50 | 2 | — | |
YCVNCXIPRCVVBB
|
8.8 | IC50 | 2 | — | |
KRULSUCANQUTLR
|
8.8 | IC50 | 2 | — | |
FYBXDJNRVFIQTH
|
8.7 | IC50 | 2 | — | |
GTWJSUYVWGBQFX
|
8.7 | IC50 | 2 | — | |
ULEVDWUWWFYCCD
|
8.7 | IC50 | 2 | — | |
ZCCPLJOKGAACRT
|
8.7 | Kd | 599 | — | |
AWNNDHTUHGTAEJ
|
8.7 | IC50 | 2 | — | |
IOSOHDPFAYTRIG
|
8.7 | IC50 | 2 | — | |
ULXFFBWWZLAHEB
|
8.7 | IC50 | 2 | — | |
AYPKOBSJMAUBFQ
|
8.7 | IC50 | 2 | — | |
BJOKWHXHNKPJQG
|
8.7 | IC50 | 2 | — |