Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QNUKRWAIZMBVCU
|
6.5 | IC50 | 17 | Yes | |
AALWZYBTBKNLKF
|
6.5 | IC50 | 4 | — | |
DDKIKSYBXRUQAD
|
6.5 | IC50 | 2 | — | |
OUCWASUSWASVRS
|
6.5 | IC50 | 2 | — | |
ZXYVYYGVHZWKGW
|
6.5 | IC50 | 2 | — | |
MFFCVWBLWOKMQK
|
6.4 | IC50 | 2 | — | |
QNABDSWBQJKBHK
|
6.4 | IC50 | 45 | — | |
FYXULBBAJZXNDR
|
6.4 | IC50 | 2 | — | |
RPAZLTQZYXMTQP
|
6.4 | IC50 | 2 | — | |
RSOMSYHDLLNJGQ
|
6.4 | IC50 | 4 | — | |
GUBJNPWVIUFSTR
|
6.4 | Kd | 103 | — | |
MCGWMMNJZVZFCG
|
6.4 | IC50 | 2 | — | |
PQILTUGKKMWZPN
|
6.4 | IC50 | 3 | — | |
CLDZMWNXQSYUGP
|
6.4 | IC50 | 2 | — | |
HNGSMPZLGYDZOV
|
6.4 | IC50 | 4 | — | |
WPVGMQYGOHYFNN
|
6.4 | IC50 | 2 | — | |
XZCLCFIAUCVNJF
|
6.4 | IC50 | 4 | — | |
ZRHRPGSSSVYBRG
|
6.4 | IC50 | 2 | — | |
BSFNGHCTZDCQBF
|
6.4 | Ki | 93 | — | |
CFBADDSSFSYJPF
|
6.4 | Ki | 23 | — | |
GAJUUQYPFUJQCH
|
6.4 | IC50 | 2 | — | |
HATNHAMXMKJCEI
|
6.4 | Ki | 9 | — | |
HCJQIBXTZXVZLX
|
6.4 | IC50 | 2 | — | |
IPTSYCYNQJITNJ
|
6.4 | Ki | 12 | — | |
LVXRFLDTIWZWSH
|
6.4 | IC50 | 2 | — | |
MDJCUXFFMNEBHG
|
6.4 | Ki | 13 | — | |
PHWHNHYZZNJPLB
|
6.4 | Ki | 16 | — | |
PSCJSWRVCKUMSL
|
6.4 | Ki | 35 | — | |
RGNHKJWHFIPHIM
|
6.4 | Ki | 66 | — | |
RHCMQQAUBJPPPW
|
6.4 | IC50 | 4 | — | |
RYYNGWLOYLRZLK
|
6.4 | Ki | 104 | — | |
SGHXFHRRWFLILP
|
6.4 | Ki | 29 | — | |
SRUYMJRFVGLQDV
|
6.4 | Ki | 37 | — | |
WDARYLSSWBWVCU
|
6.4 | Ki | 49 | — | |
WIOFZLMIWUBUJO
|
6.4 | IC50 | 2 | — | |
WMFVCLKZYKMDNK
|
6.4 | IC50 | 8 | — | |
WUTVMXLIGHTZJC
|
6.4 | Ki | 5 | Yes | |
YGEACCLUBSGMMJ
|
6.4 | Ki | 16 | — | |
ZCAOFAAOUBUUBJ
|
6.4 | Ki | 9 | — | |
DFOQUEDJAQZZIV
|
6.4 | IC50 | 2 | — | |
FWXVGKSWZJEPQI
|
6.4 | IC50 | 5 | — | |
KRAOZXBAPOLPAO
|
6.4 | IC50 | 4 | — | |
PGPHHJBZEGSUNE
|
6.4 | IC50 | 3 | — | |
UOPHVMRUNRZBPW
|
6.4 | IC50 | 2 | — | |
ZFJLHOJPSZZLSS
|
6.4 | IC50 | 2 | — | |
BSTCRUFJLBKYMG
|
6.4 | IC50 | 4 | — | |
DTECYEKXRKVIQZ
|
6.4 | IC50 | 2 | — | |
PIMQWRZWLQKKBJ
|
6.4 | IC50 | 36 | — | |
UAILDZHGMNDSLW
|
6.4 | IC50 | 2 | — | |
AFBWGXIHPVUWLP
|
6.4 | IC50 | 2 | — |