Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DOKPTPBHIRPUBR
|
6.6 | IC50 | 2 | — | |
ROUPUTCHGWRJJN
|
6.6 | IC50 | 2 | — | |
COLRVGXKZJZTAW
|
6.6 | IC50 | 2 | — | |
IXRCZLGBPPMVSP
|
6.6 | Kd | 9 | — | |
JWRGIVHRSKLDID
|
6.6 | IC50 | 2 | — | |
OTKVWQZLCANFNT
|
6.6 | IC50 | 2 | — | |
PCGFFBLPRCUXPW
|
6.6 | IC50 | 2 | — | |
SGTDUJKKGWWCEY
|
6.6 | IC50 | 2 | — | |
AXRCEOKUDYDWLF
|
6.6 | Kd | 31 | — | |
GBQLBCIOXAJQAP
|
6.6 | IC50 | 2 | — | |
OGQDHXGPFCDXGA
|
6.6 | IC50 | 4 | — | |
PJFOGIDCQLDLHH
|
6.6 | IC50 | 2 | — | |
VIFMVQBVAVNATG
|
6.6 | IC50 | 4 | — | |
GDYZFFBMSBDTAA
|
6.6 | Ki | 60 | — | |
HIYNYRWOAKCPBZ
|
6.6 | Ki | 2 | — | |
HZPACYSNLOCDLW
|
6.6 | Ki | 48 | — | |
KFTMUWPUQBCIED
|
6.6 | IC50 | 2 | — | |
LHQWPYOYDRVMFI
|
6.6 | Ki | 21 | — | |
LJHWVFJTDNXUTQ
|
6.6 | IC50 | 2 | — | |
NFMGZVPRGVERNN
|
6.6 | Ki | 44 | — | |
NMHMCXTYPRADBA
|
6.6 | Ki | 20 | — | |
NPHKXSDZIKFIRU
|
6.6 | IC50 | 5 | — | |
NRFIAFHOBIQDRE
|
6.6 | IC50 | 2 | — | |
OLVBAUVSICCWEJ
|
6.6 | Ki | 39 | — | |
ZCXXFPLQFFRMPN
|
6.6 | Ki | 12 | — | |
HFIYFKUCCHWYDX
|
6.6 | IC50 | 4 | — | |
IKLOROWNYFUEKV
|
6.6 | IC50 | 4 | — | |
TXDQGBBBTIUCBD
|
6.6 | IC50 | 2 | — | |
MZDKLVOWGIOKTN
|
6.6 | Kd | 80 | — | |
RZFJBSIAXYEPBX
|
6.6 | IC50 | 6 | — | |
XPTBENXBQDKVHB
|
6.6 | IC50 | 2 | — | |
AQKVJQFKLCIABA
|
6.6 | IC50 | 2 | — | |
CURXWONZHCZVOV
|
6.6 | IC50 | 5 | — | |
WMSHTIRWIOFMAY
|
6.6 | IC50 | 3 | — | |
KGPGFQWBCSZGEL
|
6.6 | Kd | 59 | Yes | |
YBFJEMNJNCMXOO
|
6.6 | IC50 | 3 | — | |
DTYGFXKVLYKJLW
|
6.5 | IC50 | 3 | — | |
JCSZOMMQIMMAMS
|
6.5 | IC50 | 4 | — | |
JRNJNYBQQYBCLE
|
6.5 | Kd | 40 | Yes | |
JUDQUEPWMOKMGQ
|
6.5 | IC50 | 2 | — | |
YWBUMBUFDDSLCR
|
6.5 | IC50 | 4 | — | |
YYWGDJIEQNZXDR
|
6.5 | IC50 | 3 | Yes | |
BOKIQWSDLBGRGI
|
6.5 | IC50 | 2 | — | |
OGLXQFQATMRTEA
|
6.5 | IC50 | 2 | — | |
QKZKUCIKRGDWHQ
|
6.5 | IC50 | 3 | — | |
RASCHEQRJMEENP
|
6.5 | IC50 | 4 | — | |
HZKOUKPIDXDOOI
|
6.5 | IC50 | 4 | — | |
STYBOAPFAFDXGS
|
6.5 | IC50 | 3 | — | |
DAGAGBZRNRKMGJ
|
6.5 | IC50 | 2 | — | |
FLDSZPYCDPPFIH
|
6.5 | IC50 | 2 | — |