Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WSUSQFQQODISNM
|
6.8 | IC50 | 3 | Yes | |
LCBPOSVOPCDBGG
|
6.8 | IC50 | 2 | — | |
RMLWKXHTADHNDS
|
6.8 | IC50 | 2 | — | |
OJQQCSPYLMDJQP
|
6.7 | IC50 | 3 | — | |
AVIWDYSJSPOOAR
|
6.7 | IC50 | 11 | — | |
BRAUILVAENFWMQ
|
6.7 | IC50 | 2 | — | |
DGICZXPTVAKIDT
|
6.7 | IC50 | 2 | — | |
VMFBKDNUNVTPGE
|
6.7 | IC50 | 3 | — | |
YBCIRCIUSJGTSE
|
6.7 | IC50 | 2 | — | |
BDRSCIWOUKYOAH
|
6.7 | IC50 | 2 | — | |
GNUSRHBKQSQSGA
|
6.7 | IC50 | 2 | — | |
OBJPHIOAHHIJPG
|
6.7 | IC50 | 4 | — | |
OCGMYHIDTHTZSV
|
6.7 | IC50 | 4 | — | |
QGAMKOCDVQJIEP
|
6.7 | IC50 | 5 | — | |
AJOLXGKMRXNPKQ
|
6.7 | IC50 | 4 | — | |
HDOIATBUQVHXDJ
|
6.7 | IC50 | 4 | — | |
IUEBPIPDFMCSTP
|
6.7 | Ki | 29 | — | |
JCFJQIHDZHHMQT
|
6.7 | Ki | 42 | — | |
NEWAULHLLUCDPD
|
6.7 | Ki | 27 | — | |
OILINXINODUEIB
|
6.7 | IC50 | 8 | — | |
OKHSIZNHMYBPJZ
|
6.7 | IC50 | 2 | — | |
QBKUOOQFSVMDPB
|
6.7 | Ki | 31 | — | |
TZSJMSZEKQGCBI
|
6.7 | Ki | 15 | — | |
WKWARMGSTJGPIX
|
6.7 | Ki | 3 | — | |
WYEVMOFRKALLJA
|
6.7 | IC50 | 4 | — | |
XSRHBCYNCKAFKS
|
6.7 | Ki | 45 | — | |
YMSZHISTTIUBDG
|
6.7 | Ki | 7 | — | |
CGXCGLMVTWFROO
|
6.7 | IC50 | 4 | — | |
CLESVRTZYWZTST
|
6.7 | IC50 | 2 | — | |
FTQIAAZOFQGUCE
|
6.7 | IC50 | 2 | — | |
JWKVIXXNQQUNBC
|
6.7 | IC50 | 3 | — | |
HOBGSWDBYMRRJR
|
6.7 | IC50 | 4 | — | |
RAXZSEGXMBWYQK
|
6.7 | IC50 | 21 | — | |
VMLGIOLTESMMRK
|
6.7 | IC50 | 2 | — | |
YTFORVXPFIUVAF
|
6.7 | IC50 | 4 | — | |
GWTAEVKZCDFFEX
|
6.7 | IC50 | 3 | — | |
OSVUGUHRKMMBSE
|
6.7 | Kd | 170 | — | |
PFDTUGRHCXXOIZ
|
6.7 | IC50 | 2 | — | |
XCYIIVRZXLZJER
|
6.7 | IC50 | 2 | — | |
YCZJWFJXVYDVJB
|
6.7 | IC50 | 4 | — | |
DNTVXDZWVOVLOD
|
6.7 | IC50 | 5 | — | |
FCKZDUKVAZTJNK
|
6.7 | IC50 | 2 | — | |
KYCKVFRIBMZEAX
|
6.7 | IC50 | 2 | — | |
VXMFHVFTECVHPF
|
6.7 | IC50 | 4 | — | |
AOHZJKSTSDMBIZ
|
6.7 | IC50 | 3 | — | |
POPAKMWQVKOZMW
|
6.7 | IC50 | 4 | — | |
SEATWUHTGZDTAX
|
6.7 | IC50 | 2 | — | |
FQAOJJZIGINGIO
|
6.6 | Ki | 2 | — | |
VMHDKSJEGBWITL
|
6.6 | IC50 | 2 | — | |
WYYSOGMUPDEQEM
|
6.6 | IC50 | 2 | — |