Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KMPXHOHRWCFMTC
|
6.9 | IC50 | 4 | — | |
SDDXLJVXFBEYGV
|
6.9 | IC50 | 8 | — | |
UEFCSGDOOJJXTN
|
6.9 | IC50 | 46 | — | |
CPNVJHSWNCPSIP
|
6.9 | IC50 | 2 | — | |
FAYCRVHZDSFSBE
|
6.9 | IC50 | 2 | — | |
JETNNLCMZCYIJE
|
6.9 | IC50 | 2 | — | |
VUGVTCFJRKTFSE
|
6.9 | IC50 | 2 | — | |
IDPHPRPMCOPJNX
|
6.9 | IC50 | 4 | — | |
ARIOBGGRZJITQX
|
6.8 | IC50 | 24 | — | |
FJINJXZTEKDFRA
|
6.8 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
6.8 | Kd | 213 | — | |
HPXRZQICQXFGFT
|
6.8 | IC50 | 2 | — | |
IZJDKDDRAYOTGH
|
6.8 | IC50 | 4 | — | |
JZNQVKNWCJMHKJ
|
6.8 | IC50 | 2 | — | |
PURZKCWZRZSACX
|
6.8 | IC50 | 2 | — | |
SDCHARFPZYFAKJ
|
6.8 | IC50 | 2 | — | |
RLMJMTPRBLGCRP
|
6.8 | IC50 | 2 | — | |
RZMARTVDMQPCDI
|
6.8 | IC50 | 2 | — | |
BVEVXRDDVGYLHG
|
6.8 | IC50 | 2 | — | |
FJMPCGCOGLTHPC
|
6.8 | IC50 | 2 | — | |
HJVDQPRJANOXIX
|
6.8 | IC50 | 10 | — | |
HKPNVAASTVCDIR
|
6.8 | IC50 | 2 | — | |
HKXSAMUAKQJHLQ
|
6.8 | IC50 | 2 | — | |
IMKJGRXMBFNOGA
|
6.8 | IC50 | 2 | — | |
RVXAVLKJEPIRIR
|
6.8 | Ki | 2 | — | |
TVXWKAUMIVTQTA
|
6.8 | IC50 | 4 | — | |
ANHNZYQVWLXJET
|
6.8 | IC50 | 2 | — | |
PHLOAJCAGOSYSY
|
6.8 | IC50 | 2 | — | |
ADMFLILDQJSEIK
|
6.8 | Ki | 72 | — | |
BQWBZBFRJHWSEA
|
6.8 | IC50 | 5 | — | |
CXPZMHPFUWJLIA
|
6.8 | IC50 | 4 | — | |
DWHOVKRIZFMOSJ
|
6.8 | Ki | 4 | — | |
DZIPQNPWTUXXSJ
|
6.8 | Ki | 18 | — | |
FAIHBCXQSBIRIL
|
6.8 | Ki | 22 | — | |
FSWFKKQQSQHIRZ
|
6.8 | Ki | 10 | — | |
IMMZLRQJNZSTTE
|
6.8 | Ki | 15 | — | |
KDKUVYLMPJIGKA
|
6.8 | Kd | 91 | Yes | |
OAVGBZOFDPFGPJ
|
6.8 | Ki | 42 | Yes | |
OWDRQHVEJIYVOI
|
6.8 | Ki | 47 | — | |
OWRXHGAFWZFFCW
|
6.8 | Ki | 113 | — | |
QNWXRLPZIFMTBK
|
6.8 | IC50 | 12 | — | |
ROQWMUVYMUOSQS
|
6.8 | IC50 | 2 | — | |
UTFXYGYVDDLJER
|
6.8 | Ki | 36 | — | |
XPHWIERLJBFPFV
|
6.8 | Ki | 69 | — | |
YDOPLCNFRXOHCC
|
6.8 | Ki | 28 | — | |
ZBELDPMWYXDLNY
|
6.8 | IC50 | 4 | — | |
AMQWJXRKJIUZAW
|
6.8 | IC50 | 2 | — | |
BDNALELXSRUQLO
|
6.8 | IC50 | 2 | — | |
ABQLVQSYGVOLAD
|
6.8 | IC50 | 2 | — | |
JPOSFPUHBHRUAX
|
6.8 | IC50 | 40 | Yes |