Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YYGKSMKAYKZSBC
|
7.0 | IC50 | 3 | — | |
FNIJSKUUKJCDGW
|
7.0 | IC50 | 2 | — | |
IEBPZCOLCOJVHI
|
7.0 | IC50 | 2 | — | |
AEZICWXXUCODMN
|
7.0 | Ki | 8 | — | |
BEKSOHVYNHFKGU
|
7.0 | IC50 | 2 | — | |
BYTNUXIIMYFFMP
|
7.0 | IC50 | 2 | — | |
CHTMRWQLNNRRFJ
|
7.0 | Ki | 70 | — | |
CPGKMMMSMJKHDL
|
7.0 | Ki | 16 | — | |
FIQAVSYFYGVUJT
|
7.0 | IC50 | 2 | — | |
FUMJKSZLZJFCAQ
|
7.0 | IC50 | 4 | — | |
GVMDVMPNOAVKJR
|
7.0 | Ki | 26 | Yes | |
JGBCLJZMLUMHOO
|
7.0 | Ki | 6 | — | |
MVJMMLFMPWITEJ
|
7.0 | Ki | 110 | — | |
NBQJSDZRPFLUGK
|
7.0 | IC50 | 2 | — | |
OKCNACDPDSQZSE
|
7.0 | Ki | 7 | — | |
OYEBWUJVTCQTJD
|
7.0 | IC50 | 2 | — | |
PFCUZXCHLYIMTJ
|
7.0 | Ki | 18 | — | |
QNUKRWAIZMBVCU
|
7.0 | Ki | 46 | — | |
SDPIVLIBDDEFHL
|
7.0 | Ki | 4 | — | |
SPOBBSBKXJKGBG
|
7.0 | Ki | 16 | — | |
ZOVCAZRXVNBAFS
|
7.0 | IC50 | 2 | — | |
ZZRDSHKJUCIYQL
|
7.0 | IC50 | 2 | — | |
ACBZAFIQJQQSBY
|
7.0 | IC50 | 2 | — | |
IDSINMBICXAPEL
|
7.0 | IC50 | 4 | — | |
NGFGTMFVWSDFPS
|
7.0 | IC50 | 32 | — | |
OZVPIRAQIFUWJE
|
7.0 | IC50 | 2 | — | |
PDFAYXCJHTYGHT
|
7.0 | IC50 | 2 | — | |
PYFNOGGEKLQDLR
|
7.0 | IC50 | 2 | — | |
VRQZQKQMJJRPDA
|
7.0 | Ki | 2 | — | |
QFXFIEVXAUEHEV
|
6.9 | IC50 | 6 | — | |
HVRUFPHUFGFCRX
|
6.9 | IC50 | 2 | — | |
HYTACIVXVQILEM
|
6.9 | IC50 | 4 | — | |
HZDBLSKHQHIDBE
|
6.9 | IC50 | 2 | — | |
QJGBZTRYFRVOPY
|
6.9 | IC50 | 2 | — | |
VWCSZVWZRTZNCH
|
6.9 | Kd | 8 | — | |
YQXSREGMIKNZEU
|
6.9 | Ki | 8 | — | |
BUVDAZCGAKIEOI
|
6.9 | IC50 | 2 | — | |
HZRMFYAOISJZBB
|
6.9 | IC50 | 2 | — | |
LHYKFLNJIXCRLM
|
6.9 | IC50 | 4 | — | |
WGHUJKZNOQWPTN
|
6.9 | IC50 | 2 | — | |
CLRFYTGANQZOBS
|
6.9 | Ki | 41 | — | |
FDBPGAHVEGEARY
|
6.9 | Ki | 19 | — | |
GJOXRIYWDHESDF
|
6.9 | Ki | 27 | — | |
LRZYYIZFBXFSJB
|
6.9 | Ki | 69 | — | |
RKLRBLPEQCNXFE
|
6.9 | IC50 | 5 | — | |
UQFRSHRWRKYNDE
|
6.9 | Ki | 17 | Yes | |
VBNPWXWJZJNXEY
|
6.9 | Ki | 18 | Yes | |
YWTBGJGMTBHQTM
|
6.9 | Ki | 65 | — | |
ZFMMEJFOLCBUGE
|
6.9 | IC50 | 2 | — | |
HBOIGMCCSYRJJS
|
6.9 | IC50 | 2 | — |