Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FUMCKNCUEAQHCV
|
7.2 | Ki | 103 | — | |
GUMBHNMWKMFKRT
|
7.2 | Ki | 23 | — | |
HMKKDSBJGMESJD
|
7.2 | Ki | 10 | — | |
VVQQRUZZQQSDEI
|
7.2 | Ki | 6 | — | |
VWVYILCFSYNJHF
|
7.2 | Ki | 49 | — | |
HHSQVERDWJTZMP
|
7.2 | IC50 | 2 | — | |
NCKLQXXBRWCYMA
|
7.2 | IC50 | 2 | — | |
PPRYPAUDEQCBJS
|
7.2 | IC50 | 2 | — | |
UVHNIMCYDWMRAE
|
7.2 | Ki | 9 | — | |
JCJGSZCPPTXTGO
|
7.2 | IC50 | 2 | — | |
BTDCUFCJAWQJCI
|
7.2 | IC50 | 4 | — | |
OLFNGLQBEZYICE
|
7.2 | IC50 | 2 | — | |
UMGIDNPHGAJLAN
|
7.2 | IC50 | 2 | — | |
UUVNQDVUHVXJFU
|
7.2 | IC50 | 2 | — | |
MBHMKMFMXOAEHV
|
7.2 | IC50 | 2 | — | |
PHTGPVWIQSKHKK
|
7.2 | IC50 | 2 | — | |
YTOGUEKUZBZZGH
|
7.2 | IC50 | 2 | — | |
LCIMOJQEZXDWTA
|
7.1 | IC50 | 3 | — | |
NXCIXCPIWIDEJO
|
7.1 | IC50 | 2 | — | |
RJTQBPCQZQSZFF
|
7.1 | Kd | 9 | — | |
ONVZFCHLOZUXRP
|
7.1 | IC50 | 2 | — | |
RPSIDICSSBFGPU
|
7.1 | IC50 | 2 | — | |
FYLWBNLJDXFSNQ
|
7.1 | IC50 | 2 | — | |
IETGSXFTNQYZQA
|
7.1 | IC50 | 4 | — | |
PMGPBZHUTBKGCZ
|
7.1 | Ki | 4 | — | |
PQCXVIPXISBFPN
|
7.1 | IC50 | 9 | Yes | |
UNXKPCQXZUAGGJ
|
7.1 | IC50 | 2 | — | |
VAPOMSIOLKMAIW
|
7.1 | Ki | 7 | — | |
AVDPZTAJYKVDBQ
|
7.1 | IC50 | 2 | — | |
CKDGJQLBXUOVSI
|
7.1 | Ki | 2 | — | |
HZOKUCWZAVEKGI
|
7.1 | IC50 | 3 | — | |
IFQICUARAXVEIQ
|
7.1 | Ki | 18 | — | |
JJUNZYVUGWVURX
|
7.1 | IC50 | 2 | — | |
JUWGHVCIMRIFQO
|
7.1 | IC50 | 2 | — | |
KTRGYJLQTZDGPX
|
7.1 | Ki | 9 | — | |
PCQMERRARZKTPW
|
7.1 | Ki | 68 | — | |
XZWVOUQIYLZUCJ
|
7.1 | Ki | 23 | — | |
YEHCNYAQEBQCCS
|
7.1 | Ki | 74 | — | |
PYBQDPOCAWUSJF
|
7.1 | IC50 | 4 | — | |
PLKSEXHMPNQHEY
|
7.1 | IC50 | 2 | — | |
ZVSDEXYXGKLASP
|
7.1 | IC50 | 2 | — | |
BZIKSZZVJAQWMC
|
7.1 | Ki | 6 | — | |
CKNBSSMNQGLXEA
|
7.1 | IC50 | 3 | — | |
DKZYXHCYPUVGAF
|
7.1 | Kd | 112 | — | |
PZKKJJYMVWVYOZ
|
7.1 | IC50 | 2 | — | |
IJYCUHJDYAFEOT
|
7.0 | IC50 | 2 | — | |
FGYLHONNVFJRIG
|
7.0 | IC50 | 2 | — | |
HNEHMLOMNXWVTI
|
7.0 | IC50 | 2 | — | |
UABQVGRYOFOCJO
|
7.0 | IC50 | 2 | — | |
LLELAEGDEATZFN
|
7.0 | IC50 | 3 | — |