Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AGSPQSKJPUNTNL
|
10.1 | Ki | 2 | — | |
CJBGZDIMVHUOFK
|
10.0 | IC50 | 3 | — | |
GIIJLYUXUBPINQ
|
10.0 | IC50 | 3 | — | |
MENVSADYTLLXLP
|
10.0 | IC50 | 2 | — | |
NLDJCOJHSPZIKJ
|
10.0 | IC50 | 2 | — | |
PBPNRBLKSDOCOP
|
10.0 | Ki | 2 | — | |
COJODIOMIPYEGM
|
9.8 | IC50 | 2 | — | |
OGFGCRFMUGVFGM
|
9.7 | Ki | 2 | — | |
PYDXUBHPYGQXBU
|
9.7 | IC50 | 3 | — | |
GOMNONYNAWUWRB
|
9.7 | IC50 | 3 | — | |
NXMNKSKXYYCWRN
|
9.7 | IC50 | 3 | — | |
KZAWBYUYDLDFQY
|
9.7 | IC50 | 3 | — | |
FHAJBKJRGWQUEK
|
9.7 | IC50 | 3 | — | |
PICRXLQEOXMWHZ
|
9.7 | IC50 | 3 | — | |
GHFQRLZWDHJYKZ
|
9.7 | IC50 | 2 | — | |
QLWFPXXGZGCHFQ
|
9.6 | IC50 | 5 | — | |
CCLYDGMRCYZTFK
|
9.6 | IC50 | 2 | — | |
MENVSADYTLLXLP
|
9.5 | IC50 | 6 | — | |
NDAFUJBJGDJBNC
|
9.5 | IC50 | 3 | — | |
CJHNTUKGOQCWKH
|
9.5 | IC50 | 2 | — | |
QCOOCCREMZWFAR
|
9.5 | IC50 | 3 | — | |
MENVSADYTLLXLP
|
9.5 | IC50 | 2 | — | |
XZCZVUKTNGBHOF
|
9.5 | IC50 | 2 | — | |
KOZNFQBNKITETG
|
9.5 | IC50 | 3 | — | |
SPTOLQPXVZHQQD
|
9.4 | IC50 | 3 | — | |
DHZZLYIYWJJLRB
|
9.4 | IC50 | 3 | — | |
GSXIRUIKNXNLAP
|
9.4 | IC50 | 3 | — | |
HSFYCTPGOPYGHQ
|
9.4 | IC50 | 2 | — | |
OQKSXFCBEUFFIJ
|
9.4 | IC50 | 2 | — | |
VPGLALPDHBCDQS
|
9.4 | IC50 | 3 | — | |
CSJHKAPXYLZAOS
|
9.3 | IC50 | 2 | — | |
GQZOLEYJVGWCGW
|
9.3 | IC50 | 2 | — | |
WWEHEGICBBJKLI
|
9.2 | IC50 | 3 | — | |
NBSJZWFDNFWQDN
|
9.2 | IC50 | 29 | — | |
NPBXBJGEHIIUSM
|
9.2 | IC50 | 3 | — | |
RAUNAZYXRMQIJT
|
9.2 | IC50 | 2 | — | |
SQNUUZACFPKMEP
|
9.2 | Ki | 2 | — | |
DFTCADIVUJRTNH
|
9.2 | IC50 | 2 | — | |
NRFNSOIBXUBPGR
|
9.2 | IC50 | 2 | — | |
RTRFGHCJJJKLNN
|
9.1 | IC50 | 2 | — | |
FAACVFRHPMNIQT
|
9.1 | IC50 | 2 | — | |
LXLVKFBRQINQCN
|
9.1 | IC50 | 3 | — | |
MNIRHKZCFQNAGM
|
9.1 | IC50 | 3 | — | |
VBTNLJJWTKVDJI
|
9.1 | IC50 | 2 | — | |
VNVKSDCWJDOWNE
|
9.1 | IC50 | 3 | — | |
DRDJBBZKDSVNTH
|
9.1 | IC50 | 2 | — | |
FIUNUJMCHFAOKT
|
9.1 | IC50 | 2 | — | |
RUUPXYQCYGGBFU
|
9.1 | IC50 | 2 | — | |
RTMFABSOYYXMSU
|
9.0 | IC50 | 2 | — | |
XMLJBPQUTWBABY
|
9.0 | Ki | 2 | — |