Target Details
| UniProt AC | P49761 |
|---|---|
| Gene Symbol | CLK3 |
| Protein Name | Dual specificity protein kinase CLK3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 167
- Clinical molecules 7
- Avg pChEMBL 6.54
Active Molecules (167)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CIEDQRFRRJHOSA
|
6.1 | IC50 | 6 | — | |
JBWDTSLHUJHODF
|
6.1 | IC50 | 9 | — | |
FBURYRMHEHTVED
|
6.0 | IC50 | 9 | — | |
HKSZLNNOFSGOKW
|
6.0 | IC50 | 408 | — | |
HKSZLNNOFSGOKW
|
6.0 | Kd | 213 | — | |
USYASDQVUTWEQM
|
6.0 | IC50 | 9 | — | |
KCTCLVINURCCIL
|
6.0 | IC50 | 6 | — | |
CHQYAWLKOUOTQO
|
6.0 | IC50 | 7 | — | |
ANKYADWZYKSCAJ
|
6.0 | IC50 | 7 | — | |
AQLWSCZCZJWUMZ
|
6.0 | IC50 | 6 | — | |
BGVLELSCIHASRV
|
6.0 | Kd | 11 | — | |
BIIVYFLTOXDAOV
|
6.0 | Kd | 82 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
QTRZNDLLYHSJSH
|
6.0 | IC50 | 7 | — | |
ZYDSDRZMIWGATN
|
6.0 | IC50 | 4 | — |