Target Details
| UniProt AC | P49761 |
|---|---|
| Gene Symbol | CLK3 |
| Protein Name | Dual specificity protein kinase CLK3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 167
- Clinical molecules 7
- Avg pChEMBL 6.54
Active Molecules (167)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PAEKWZJLZMSTLB
|
6.3 | IC50 | 6 | — | |
GHQYHWMWJLSKRP
|
6.3 | IC50 | 9 | — | |
YKFHBMIPXGSMRS
|
6.3 | IC50 | 7 | — | |
RUQXGVGYNKIGJD
|
6.3 | IC50 | 9 | — | |
RILDWXOQLWEXDG
|
6.3 | IC50 | 6 | — | |
YSBCFQVEEKUZSU
|
6.3 | IC50 | 7 | — | |
CXJCGSPAPOTTSF
|
6.3 | IC50 | 3 | — | |
LXQXBEIFOYAXOP
|
6.3 | IC50 | 9 | — | |
YDTHCIZMSQZYMR
|
6.3 | IC50 | 7 | — | |
IJFKKIMDRSZOOW
|
6.2 | IC50 | 9 | — | |
KQZBWTMAFLOSPA
|
6.2 | IC50 | 8 | — | |
JXQZHHAAJMQJKU
|
6.2 | IC50 | 6 | — | |
QMUKOEKTUBVPFU
|
6.2 | IC50 | 12 | — | |
JFDRONLMXPRQPP
|
6.2 | IC50 | 9 | — | |
SKKBUBMBPCJYKW
|
6.2 | IC50 | 9 | — | |
XQVVPGYIWAGRNI
|
6.2 | Kd | 34 | — | |
XTJRKTBELWGSDN
|
6.2 | IC50 | 8 | — | |
CGRDYMCBGXJNLR
|
6.2 | IC50 | 9 | — | |
WHPORTUXBLFUPA
|
6.2 | IC50 | 9 | — | |
BWNQBFHVFFZHMR
|
6.2 | IC50 | 10 | — | |
URXJBXVGNBGIJA
|
6.2 | IC50 | 9 | — | |
GXCOUFPTCZUTEE
|
6.2 | IC50 | 10 | — | |
HHSNDNONCUTNQR
|
6.2 | IC50 | 7 | — | |
JBWDTSLHUJHODF
|
6.2 | IC50 | 9 | — | |
LDYVHYUGOBDUMZ
|
6.2 | IC50 | 6 | — | |
MQRHLOPPMRFMKM
|
6.2 | IC50 | 9 | — | |
PEICIAVUWSXRGP
|
6.2 | IC50 | 7 | — | |
BULHRWBHKAVJMT
|
6.2 | IC50 | 8 | — | |
IRBWROIEALHOPH
|
6.2 | IC50 | 7 | — | |
PAHHKMMVQJCPJI
|
6.2 | IC50 | 8 | — | |
YAXGFAAKCUOWNM
|
6.2 | IC50 | 9 | — | |
CEWIXDGUKGVYDQ
|
6.1 | IC50 | 7 | — | |
CXJCGSPAPOTTSF
|
6.1 | IC50 | 6 | — | |
FEZCHKAGMYXVNX
|
6.1 | IC50 | 6 | — | |
YVSLJAICTSVCDB
|
6.1 | IC50 | 6 | — | |
ACOQCSBMVFAWQV
|
6.1 | IC50 | 6 | — | |
AOLMNCAPVYTEHC
|
6.1 | IC50 | 6 | — | |
SBYPANVVFZBWDF
|
6.1 | IC50 | 9 | — | |
RLTCEYSNDOXWKS
|
6.1 | IC50 | 7 | — | |
DCHAEDURAZJASA
|
6.1 | IC50 | 9 | — | |
QCHDHJOEPUQALZ
|
6.1 | IC50 | 9 | — | |
XCTYEZWILVGTGO
|
6.1 | IC50 | 9 | — | |
ZJVGZWWTWGRGFK
|
6.1 | IC50 | 4 | — | |
HBBPDNLIBIZZFL
|
6.1 | IC50 | 7 | — | |
HEVBCYZPXGZFGS
|
6.1 | IC50 | 11 | — | |
IDOKKOQIQLHASZ
|
6.1 | IC50 | 8 | — | |
YHZQZEGQCKWCLP
|
6.1 | IC50 | 9 | — | |
ANKYADWZYKSCAJ
|
6.1 | IC50 | 7 | — | |
OEVQTWCGWDOIFZ
|
6.1 | IC50 | 6 | — | |
YRFAWSIUIFNVQA
|
6.1 | IC50 | 9 | — |