Target Details
| UniProt AC | P49761 |
|---|---|
| Gene Symbol | CLK3 |
| Protein Name | Dual specificity protein kinase CLK3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 167
- Clinical molecules 7
- Avg pChEMBL 6.54
Active Molecules (167)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QQWUGDVOUVUTOY
|
6.7 | Kd | 231 | Yes | |
RYWACTNAXCMTTN
|
6.7 | IC50 | 9 | — | |
DPDVVGCNUWGGRS
|
6.7 | IC50 | 10 | — | |
LZTDWHFXSWDVAG
|
6.7 | IC50 | 7 | — | |
PPZINUUIYSVIGC
|
6.7 | IC50 | 6 | — | |
YDTHCIZMSQZYMR
|
6.7 | IC50 | 9 | — | |
COYCDCAUDJBGOV
|
6.6 | IC50 | 6 | — | |
FRPGBGWSLAGPND
|
6.6 | IC50 | 7 | — | |
NSDQDNNJFIKBKR
|
6.6 | IC50 | 6 | — | |
LMXLOYKFDZEHCS
|
6.6 | IC50 | 7 | — | |
KQCIEIGKPXQRLM
|
6.5 | IC50 | 6 | — | |
RJYLSCSDDDQEPD
|
6.5 | IC50 | 10 | — | |
UMWJBFSPIYCGRG
|
6.5 | IC50 | 7 | — | |
YGXHQYJKJUFSJI
|
6.5 | IC50 | 14 | — | |
RAQBQAXSLHDSKW
|
6.5 | IC50 | 8 | — | |
BWKADHBOXYDZFU
|
6.5 | IC50 | 10 | — | |
HAFFBDGNUZMNIJ
|
6.5 | IC50 | 7 | — | |
AOGIFFVMTGMFBP
|
6.5 | IC50 | 8 | — | |
CWJLAVRXVFHDSJ
|
6.5 | IC50 | 13 | — | |
IWKDQQIVXBSVBE
|
6.5 | IC50 | 3 | — | |
UBPYILGKFZZVDX
|
6.5 | Kd | 130 | Yes | |
KDKUVYLMPJIGKA
|
6.5 | Kd | 91 | Yes | |
RPGZQOOZHIEPJW
|
6.5 | Kd | 18 | — | |
RPGZQOOZHIEPJW
|
6.5 | Kd | 18 | — | |
WHPORTUXBLFUPA
|
6.5 | IC50 | 8 | — | |
WAJNOEPHTZIWTO
|
6.5 | IC50 | 6 | — | |
ROPFCXUWNMYMSW
|
6.5 | IC50 | 10 | — | |
MXRBAJVBWGVZJI
|
6.5 | IC50 | 4 | — | |
OGXQCQYWBIOFNU
|
6.5 | IC50 | 3 | — | |
DJHMDVUOYUYLOJ
|
6.5 | IC50 | 9 | — | |
GJYVLTPTDBQQCY
|
6.4 | IC50 | 7 | — | |
OVPNQJVDAFNBDN
|
6.4 | Kd | 44 | Yes | |
SJWUVVGOTOMGOH
|
6.4 | IC50 | 9 | — | |
PPQSZAVBAJMLRF
|
6.4 | IC50 | 5 | — | |
XTJRKTBELWGSDN
|
6.4 | IC50 | 8 | — | |
YYSXUOHHBBMQMJ
|
6.4 | IC50 | 7 | — | |
WFOMWAYINPJPDX
|
6.4 | IC50 | 9 | — | |
YMIDGKZVYFXIBW
|
6.4 | IC50 | 8 | — | |
YHZQZEGQCKWCLP
|
6.4 | IC50 | 9 | — | |
ACOQCSBMVFAWQV
|
6.4 | IC50 | 8 | — | |
FIVWKNZKXNNFCW
|
6.4 | IC50 | 9 | — | |
BDMXFIMYKGLQAL
|
6.4 | IC50 | 9 | — | |
OQSBQXVIMQMCES
|
6.4 | IC50 | 9 | — | |
OSWHZHVVVZAPRN
|
6.4 | IC50 | 6 | — | |
YORVMWUGDVGXOQ
|
6.3 | IC50 | 8 | — | |
MCNDTHVVURYHKT
|
6.3 | IC50 | 8 | — | |
NNPWUWSWEGWPMQ
|
6.3 | IC50 | 8 | — | |
QFBOPHGXTBOQRN
|
6.3 | Kd | 7 | — | |
VCCCOYOXNKTQFO
|
6.3 | IC50 | 9 | — | |
YSBCFQVEEKUZSU
|
6.3 | IC50 | 9 | — |