Target Details
| UniProt AC | P49761 |
|---|---|
| Gene Symbol | CLK3 |
| Protein Name | Dual specificity protein kinase CLK3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 167
- Clinical molecules 7
- Avg pChEMBL 6.54
Active Molecules (167)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PRJNNPMIUGYOST
|
8.5 | IC50 | 14 | — | |
PMWVYONICYRLNY
|
8.2 | Kd | 4 | — | |
BHKVSOQUPYXVRZ
|
8.1 | IC50 | 6 | — | |
SJWUVVGOTOMGOH
|
8.0 | IC50 | 10 | — | |
QTHCAAFKVUWAFI
|
7.9 | IC50 | 23 | — | |
JRNJNYBQQYBCLE
|
7.9 | Kd | 40 | Yes | |
MNWOBOAJPYEQBE
|
7.8 | IC50 | 2 | — | |
BQWWOBKMDWACGC
|
7.7 | IC50 | 8 | — | |
SJWUVVGOTOMGOH
|
7.6 | IC50 | 12 | — | |
XZCWNSGWBUAUOO
|
7.5 | IC50 | 3 | — | |
ARIOBGGRZJITQX
|
7.5 | IC50 | 24 | — | |
FGBSSPMQGRUJPS
|
7.5 | IC50 | 10 | — | |
WREJZZXSNOJGIW
|
7.4 | IC50 | 8 | — | |
MNVPCONHWCXDES
|
7.4 | IC50 | 9 | — | |
OWBFCJROIKNMGD
|
7.4 | Kd | 3 | — | |
MUOKSQABCJCOPU
|
7.4 | IC50 | 36 | — | |
QTRZNDLLYHSJSH
|
7.3 | IC50 | 9 | — | |
QTRZNDLLYHSJSH
|
7.3 | IC50 | 9 | — | |
AQDWDWAYVBQMAM
|
7.2 | IC50 | 7 | — | |
IJFKKIMDRSZOOW
|
7.1 | IC50 | 8 | — | |
VCTLOEWZYIGVBO
|
7.0 | IC50 | 12 | — | |
CGPYAXSYKQBYKJ
|
7.0 | IC50 | 12 | — | |
YSODDCRKIDDXKM
|
7.0 | IC50 | 9 | — | |
IEFFSHLHNYVSEF
|
7.0 | IC50 | 8 | — | |
GRHRWVRWLAIBGN
|
6.9 | IC50 | 5 | — | |
KHVQTEBOVFILCQ
|
6.9 | IC50 | 10 | — | |
JXQZHHAAJMQJKU
|
6.9 | IC50 | 9 | — | |
DCJOTKUJWJFCSP
|
6.9 | IC50 | 9 | — | |
YORVMWUGDVGXOQ
|
6.9 | IC50 | 8 | — | |
WFOMWAYINPJPDX
|
6.9 | IC50 | 9 | — | |
OYDWEMSWMQKSLK
|
6.9 | IC50 | 8 | — | |
DXVSNYWBRDTHFF
|
6.9 | IC50 | 9 | — | |
LVSVYVPFNYRNOF
|
6.8 | IC50 | 8 | — | |
BPNUQXPIQBZCMR
|
6.8 | Kd | 83 | Yes | |
YGVLUDLFNRZMNT
|
6.8 | IC50 | 8 | — | |
OVVHFDIQCYTOAS
|
6.8 | IC50 | 9 | — | |
RUQXGVGYNKIGJD
|
6.8 | IC50 | 6 | — | |
SJYQOVMGZOATNK
|
6.8 | IC50 | 9 | — | |
BBCSUMURJUYILA
|
6.8 | IC50 | 9 | — | |
BBCSUMURJUYILA
|
6.8 | IC50 | 10 | — | |
UHOPJKMQVDXYAV
|
6.8 | IC50 | 8 | — | |
UVJQEKJPAVSBTA
|
6.7 | IC50 | 8 | — | |
DXVSNYWBRDTHFF
|
6.7 | IC50 | 10 | — | |
QIYXLIZWXGGKOO
|
6.7 | IC50 | 10 | — | |
WREJZZXSNOJGIW
|
6.7 | IC50 | 9 | — | |
QNWARURWFRZNNO
|
6.7 | IC50 | 7 | — | |
QVLJVHWQAKYGQI
|
6.7 | IC50 | 8 | — | |
RLTCEYSNDOXWKS
|
6.7 | IC50 | 9 | — | |
CHQYAWLKOUOTQO
|
6.7 | IC50 | 20 | — | |
IVSYLIPATGYBCZ
|
6.7 | IC50 | 7 | — |