Target Details
| UniProt AC | P49760 |
|---|---|
| Gene Symbol | CLK2 |
| Protein Name | Dual specificity protein kinase CLK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 806
- Clinical molecules 29
- Avg pChEMBL 6.95
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JOQWRLVZVPMTGG
|
6.8 | IC50 | 2 | — | |
WAJNOEPHTZIWTO
|
6.8 | IC50 | 6 | — | |
CJWBPPWAPHJBEQ
|
6.8 | IC50 | 6 | — | |
GCUNCFYJKLSBKK
|
6.8 | IC50 | 5 | — | |
FQEODTMNWMDUMD
|
6.8 | Ki | 25 | — | |
GCBJDOWIQHMCMR
|
6.8 | Ki | 84 | — | |
GCZJQTRRJPRFIP
|
6.8 | Ki | 10 | — | |
RGOPHVZLEMGMBZ
|
6.8 | Ki | 20 | — | |
ZCBUQCWBWNUWSU
|
6.8 | Ki | 11 | — | |
JXQZHHAAJMQJKU
|
6.8 | IC50 | 9 | — | |
XZMVOPBXTNARPU
|
6.8 | IC50 | 2 | — | |
YDTHCIZMSQZYMR
|
6.8 | IC50 | 9 | — | |
ZYDSDRZMIWGATN
|
6.8 | IC50 | 3 | — | |
WTHVHUDPRPCKCA
|
6.8 | IC50 | 2 | — | |
FQBRQRVXPUQKLG
|
6.8 | IC50 | 10 | — | |
LFSFZGXABLTIEJ
|
6.8 | IC50 | 3 | — | |
LXDHFJUOCGKVAV
|
6.8 | IC50 | 5 | — | |
RAQBQAXSLHDSKW
|
6.8 | IC50 | 8 | — | |
SSMQRWPVVYHQOU
|
6.8 | IC50 | 2 | — | |
UBPOBEKAVPQZHZ
|
6.8 | IC50 | 5 | — | |
ZTXIJZHBTZODLI
|
6.8 | IC50 | 2 | — | |
KVFJYXRZONDRPG
|
6.8 | IC50 | 2 | — | |
SDHAXXDYIZVWAZ
|
6.8 | IC50 | 4 | — | |
LZTDWHFXSWDVAG
|
6.7 | IC50 | 7 | — | |
PYLWPZITQSVFKG
|
6.7 | IC50 | 2 | — | |
SSLQYXLLEVVVAB
|
6.7 | IC50 | 2 | — | |
UZWDCWONPYILKI
|
6.7 | IC50 | 47 | — | |
CRHJUMKCZAOJLP
|
6.7 | IC50 | 2 | — | |
MQJVDVMWBFSFHI
|
6.7 | IC50 | 5 | — | |
UTBSBSOBZHXMHI
|
6.7 | IC50 | 3 | — | |
BYMPGMQLSBLSIU
|
6.7 | IC50 | 5 | — | |
LFXYFFIMEFNDHC
|
6.7 | IC50 | 3 | — | |
VCCCOYOXNKTQFO
|
6.7 | IC50 | 9 | — | |
AIQDZMUPVYDVLB
|
6.7 | Ki | 48 | — | |
CRKQBJZCCHKEGI
|
6.7 | Ki | 20 | — | |
DTMZXHDQZQLTHA
|
6.7 | Ki | 21 | — | |
IUEBPIPDFMCSTP
|
6.7 | Ki | 29 | — | |
KXPWWMPXNUOYOH
|
6.7 | Ki | 24 | — | |
SQXSMLLCDWJNAC
|
6.7 | Ki | 20 | — | |
SRONQUHCRFZABC
|
6.7 | Ki | 28 | — | |
XQYWZGQSHLDADK
|
6.7 | IC50 | 2 | — | |
YUOWJICKAJQZLS
|
6.7 | Ki | 35 | — | |
ZGDYBJXDIXVTLV
|
6.7 | Ki | 54 | — | |
DITIJPXRAGWNLI
|
6.7 | IC50 | 2 | — | |
ANKYADWZYKSCAJ
|
6.7 | IC50 | 7 | — | |
BFZIDBAEKWSVSX
|
6.7 | IC50 | 5 | — | |
UJBJWYNPUOLFIZ
|
6.7 | IC50 | 49 | — | |
GHOJVOKLPQVRCC
|
6.7 | IC50 | 2 | — | |
JQHTYMOOIFVIJV
|
6.7 | IC50 | 5 | — | |
MFLKPCAUPXBTPC
|
6.7 | IC50 | 5 | — |