Target Details
| UniProt AC | P49760 |
|---|---|
| Gene Symbol | CLK2 |
| Protein Name | Dual specificity protein kinase CLK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 806
- Clinical molecules 29
- Avg pChEMBL 6.95
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UTBSBSOBZHXMHI
|
7.0 | IC50 | 15 | Yes | |
MQRHLOPPMRFMKM
|
7.0 | IC50 | 9 | — | |
ZHMXXVNQAFCXKK
|
7.0 | IC50 | 15 | — | |
DKVWFXPMJDEBDJ
|
6.9 | IC50 | 2 | — | |
FBURYRMHEHTVED
|
6.9 | IC50 | 9 | — | |
ZZVAFDDAQGHPFE
|
6.9 | IC50 | 2 | — | |
RYWACTNAXCMTTN
|
6.9 | IC50 | 9 | — | |
WBQNJPBYOGNEQC
|
6.9 | IC50 | 5 | — | |
ACDBIJKZXKGOFW
|
6.9 | IC50 | 2 | — | |
BXNJHAXVSOCGBA
|
6.9 | IC50 | 14 | — | |
IVSYLIPATGYBCZ
|
6.9 | IC50 | 7 | — | |
JPJBCKSRGYPABG
|
6.9 | IC50 | 3 | — | |
OAVGBZOFDPFGPJ
|
6.9 | Kd | 42 | Yes | |
OXUHZNGGQZYPHE
|
6.9 | IC50 | 2 | — | |
UBUJLBVNZCRWPX
|
6.9 | IC50 | 7 | — | |
UKWWUFBDIVBOBD
|
6.9 | IC50 | 5 | — | |
CAFIVVHIKSBSPE
|
6.9 | IC50 | 2 | — | |
MDHMXWJWNZSMEC
|
6.9 | IC50 | 2 | — | |
OITUSVUYZAXFTD
|
6.9 | IC50 | 5 | — | |
ZETRLMBMIJORIT
|
6.9 | IC50 | 2 | — | |
AOFJRBMLTUGMMP
|
6.9 | Ki | 12 | — | |
ATGVCJYHNOSZEV
|
6.9 | Ki | 23 | — | |
CPGKMMMSMJKHDL
|
6.9 | Ki | 16 | — | |
FLWYCOJREJRWLJ
|
6.9 | IC50 | 3 | — | |
HFYNRAVQEUKOFF
|
6.9 | IC50 | 3 | — | |
HJYHJYGXRBYDIG
|
6.9 | Ki | 23 | — | |
HKRUFMXPSVYVMY
|
6.9 | Ki | 4 | — | |
JWQOJVOKBAAAAR
|
6.9 | Ki | 29 | — | |
KNVOICXEDILAGT
|
6.9 | Ki | 17 | — | |
KQZBWTMAFLOSPA
|
6.9 | IC50 | 8 | — | |
LVSVYVPFNYRNOF
|
6.9 | IC50 | 8 | — | |
MZDKLVOWGIOKTN
|
6.9 | Ki | 80 | — | |
WHKVBWGIZNCFIH
|
6.9 | IC50 | 2 | — | |
YVSLJAICTSVCDB
|
6.9 | IC50 | 6 | — | |
ZRQXCQXWTLVASO
|
6.9 | Ki | 36 | — | |
PRJNNPMIUGYOST
|
6.9 | IC50 | 14 | — | |
ZXBOCEMSOANKPH
|
6.9 | IC50 | 2 | — | |
IRBWROIEALHOPH
|
6.9 | IC50 | 7 | — | |
JBWDTSLHUJHODF
|
6.9 | IC50 | 8 | — | |
GHQYHWMWJLSKRP
|
6.9 | IC50 | 9 | — | |
RLTCEYSNDOXWKS
|
6.9 | IC50 | 7 | — | |
WFOMWAYINPJPDX
|
6.9 | IC50 | 9 | — | |
KHQBJGWNPXLJQL
|
6.8 | IC50 | 2 | — | |
OWDVXJJCVWTPPW
|
6.8 | IC50 | 8 | — | |
RPECODXSMBBMSO
|
6.8 | IC50 | 2 | — | |
ZDJFIKFQLKJRBA
|
6.8 | IC50 | 4 | — | |
AOLMNCAPVYTEHC
|
6.8 | IC50 | 6 | — | |
LMXLOYKFDZEHCS
|
6.8 | IC50 | 7 | — | |
MWGBCUIRQLARSR
|
6.8 | IC50 | 2 | — | |
CTNPALGJUAXMMC
|
6.8 | Kd | 151 | — |