Target Details
| UniProt AC | P49760 |
|---|---|
| Gene Symbol | CLK2 |
| Protein Name | Dual specificity protein kinase CLK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 806
- Clinical molecules 29
- Avg pChEMBL 6.95
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AEYBYRSGXQFSBA
|
7.1 | IC50 | 2 | — | |
KQCIEIGKPXQRLM
|
7.1 | IC50 | 6 | — | |
NSGBWKVTGDJMAI
|
7.1 | IC50 | 2 | — | |
UMWJBFSPIYCGRG
|
7.1 | IC50 | 7 | — | |
WFOMWAYINPJPDX
|
7.1 | IC50 | 9 | — | |
XHRUYQISWOKHBR
|
7.1 | IC50 | 2 | — | |
GXCOUFPTCZUTEE
|
7.0 | IC50 | 10 | — | |
HAFFBDGNUZMNIJ
|
7.0 | IC50 | 7 | — | |
HJEKFRDOAYXXRU
|
7.0 | IC50 | 8 | — | |
MCNDTHVVURYHKT
|
7.0 | IC50 | 8 | — | |
QSGKPYRFWJINEH
|
7.0 | IC50 | 12 | — | |
YEFYCSKFDBXSSK
|
7.0 | IC50 | 7 | — | |
GPXCDUCDIFDAGL
|
7.0 | IC50 | 3 | — | |
MFHHFNYSUNIIMQ
|
7.0 | IC50 | 2 | — | |
NSDQDNNJFIKBKR
|
7.0 | IC50 | 6 | — | |
RUQXGVGYNKIGJD
|
7.0 | IC50 | 9 | — | |
HHSNDNONCUTNQR
|
7.0 | IC50 | 7 | — | |
YMEQWPWIQHLWLZ
|
7.0 | IC50 | 2 | — | |
YYLKKYCXAOBSRM
|
7.0 | Kd | 191 | — | |
BGVLELSCIHASRV
|
7.0 | Kd | 12 | — | |
DCHAEDURAZJASA
|
7.0 | IC50 | 9 | — | |
KBMQGIPVJGXLOU
|
7.0 | IC50 | 7 | — | |
PAEKWZJLZMSTLB
|
7.0 | IC50 | 6 | — | |
DNAKAECMKPNHBW
|
7.0 | IC50 | 2 | — | |
NNPWUWSWEGWPMQ
|
7.0 | IC50 | 8 | — | |
YMIDGKZVYFXIBW
|
7.0 | IC50 | 8 | — | |
GHAZVJQMLWOQLP
|
7.0 | Ki | 17 | — | |
IDOKKOQIQLHASZ
|
7.0 | IC50 | 8 | — | |
KKIQOEOELHJGQJ
|
7.0 | IC50 | 2 | — | |
NBIWQDNWQHQXFS
|
7.0 | IC50 | 5 | — | |
ODNOTLMFNVWFTJ
|
7.0 | Ki | 11 | — | |
UPPYTUNUGKDPSA
|
7.0 | Ki | 7 | — | |
UTFXYGYVDDLJER
|
7.0 | Ki | 36 | — | |
UZFPGFONVYFSRR
|
7.0 | Ki | 16 | — | |
VQPBIJGXSXEOCU
|
7.0 | Ki | 24 | — | |
VVEGARMQKNYDID
|
7.0 | Ki | 24 | — | |
XSDJOIOVIMPMHD
|
7.0 | Ki | 44 | — | |
XTJRKTBELWGSDN
|
7.0 | IC50 | 8 | — | |
YWITWZUKNXWOSD
|
7.0 | Ki | 10 | — | |
DJHMDVUOYUYLOJ
|
7.0 | IC50 | 9 | — | |
HBBPDNLIBIZZFL
|
7.0 | IC50 | 7 | — | |
KWDHKMSSYPOWFY
|
7.0 | IC50 | 2 | — | |
HDAJDNHIBCDLQF
|
7.0 | IC50 | 14 | — | |
PMDAVRLCSZSLRH
|
7.0 | IC50 | 13 | — | |
DXVSNYWBRDTHFF
|
7.0 | IC50 | 7 | — | |
BDMXFIMYKGLQAL
|
7.0 | IC50 | 9 | — | |
MVRRAWJPZXNFMK
|
7.0 | IC50 | 6 | — | |
NGFGTMFVWSDFPS
|
7.0 | IC50 | 32 | — | |
PAHHKMMVQJCPJI
|
7.0 | IC50 | 8 | — | |
QNWARURWFRZNNO
|
7.0 | IC50 | 7 | — |