Target Details
| UniProt AC | P49760 |
|---|---|
| Gene Symbol | CLK2 |
| Protein Name | Dual specificity protein kinase CLK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 806
- Clinical molecules 29
- Avg pChEMBL 6.95
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CYUDBMRFRZUOTH
|
7.2 | IC50 | 5 | — | |
IJFKKIMDRSZOOW
|
7.2 | IC50 | 8 | — | |
IINWRBNZDZJCAH
|
7.2 | IC50 | 2 | — | |
JBWDTSLHUJHODF
|
7.2 | IC50 | 9 | — | |
WREJZZXSNOJGIW
|
7.2 | IC50 | 9 | — | |
FVIUKIZPDJZQKD
|
7.2 | IC50 | 5 | — | |
PPALZSWDMRGSQV
|
7.2 | IC50 | 5 | — | |
RMQZLMLMRYHGDT
|
7.2 | IC50 | 2 | — | |
VNRCXZCFCYFZQN
|
7.2 | IC50 | 2 | — | |
HRRUGRNBEPWHFW
|
7.2 | IC50 | 2 | — | |
HRRUGRNBEPWHFW
|
7.2 | IC50 | 2 | — | |
HXESDBWWDYJEJQ
|
7.2 | Ki | 10 | — | |
RVSKJUNTDGBSSS
|
7.2 | Ki | 25 | — | |
ZGZVRPRSFXRGCF
|
7.2 | Ki | 76 | — | |
PDQWWZCYXKWWON
|
7.2 | IC50 | 2 | — | |
RJTQBPCQZQSZFF
|
7.2 | Kd | 9 | — | |
ABDPBSXQLBJPTL
|
7.2 | IC50 | 6 | — | |
GRHRWVRWLAIBGN
|
7.2 | IC50 | 5 | — | |
IXRCZLGBPPMVSP
|
7.2 | Kd | 9 | — | |
KHTCIOWVELAJLF
|
7.2 | IC50 | 2 | — | |
MXRBAJVBWGVZJI
|
7.2 | IC50 | 4 | — | |
OGXQCQYWBIOFNU
|
7.2 | IC50 | 3 | — | |
CRZIGHVWJFDSFR
|
7.2 | IC50 | 5 | — | |
HLJDNMVEJYCKAW
|
7.2 | IC50 | 2 | — | |
IEDDDZFQZKDRBJ
|
7.2 | IC50 | 9 | — | |
JLUCPOPZBUWANE
|
7.2 | IC50 | 2 | — | |
YJVHRHNVCYWWCM
|
7.1 | IC50 | 5 | — | |
YSBCFQVEEKUZSU
|
7.1 | IC50 | 7 | — | |
AGSOXCIDVSMLSA
|
7.1 | IC50 | 2 | — | |
DXVSNYWBRDTHFF
|
7.1 | IC50 | 9 | — | |
DPYBFMFLTZVAGA
|
7.1 | IC50 | 2 | — | |
BWORFRWIDWQHPL
|
7.1 | IC50 | 7 | — | |
CGBKQGQXEFGPDM
|
7.1 | IC50 | 6 | — | |
CLRFYTGANQZOBS
|
7.1 | Ki | 41 | — | |
DYSRECIVMDGUQU
|
7.1 | Ki | 29 | — | |
JRNJNYBQQYBCLE
|
7.1 | Kd | 40 | Yes | |
KAZJIBCOYQRDGG
|
7.1 | Ki | 16 | — | |
RGNHKJWHFIPHIM
|
7.1 | Ki | 66 | — | |
RPGBQFNDFPEOON
|
7.1 | Ki | 22 | — | |
RWKDVIAVTRRJIR
|
7.1 | Ki | 23 | — | |
SVUIYNKSDCANAY
|
7.1 | Ki | 16 | — | |
UVJQEKJPAVSBTA
|
7.1 | IC50 | 8 | — | |
CYVGSDYVNUNREA
|
7.1 | IC50 | 5 | — | |
JPMMONIVZGUBLU
|
7.1 | IC50 | 2 | — | |
LFAHWMOZPVCJAY
|
7.1 | Kd | 8 | — | |
QQWUGDVOUVUTOY
|
7.1 | Kd | 231 | Yes | |
BULHRWBHKAVJMT
|
7.1 | IC50 | 8 | — | |
LXALJHQHXMDTSD
|
7.1 | IC50 | 2 | — | |
QVLJVHWQAKYGQI
|
7.1 | IC50 | 8 | — | |
TVUWQDLBEOZVOU
|
7.1 | IC50 | 41 | — |