Target Details
| UniProt AC | P49760 |
|---|---|
| Gene Symbol | CLK2 |
| Protein Name | Dual specificity protein kinase CLK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 806
- Clinical molecules 29
- Avg pChEMBL 6.95
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WREJZZXSNOJGIW
|
7.4 | IC50 | 8 | — | |
MXEZQEFCKXVMFN
|
7.4 | IC50 | 5 | — | |
NVTNPVQFMSQPJQ
|
7.4 | IC50 | 7 | — | |
YSODDCRKIDDXKM
|
7.4 | IC50 | 9 | — | |
BBCSUMURJUYILA
|
7.4 | IC50 | 9 | — | |
BLMDVYRPCVHXPK
|
7.4 | IC50 | 6 | — | |
DQYDZCRLDYVZKY
|
7.4 | IC50 | 5 | — | |
INAVVYMHODCJNF
|
7.4 | IC50 | 5 | — | |
SJYQOVMGZOATNK
|
7.4 | IC50 | 9 | — | |
SWPXADMCNLNAGW
|
7.4 | IC50 | 10 | — | |
YHZQZEGQCKWCLP
|
7.4 | IC50 | 9 | — | |
BEJCLDKQCNVTQR
|
7.4 | Ki | 16 | — | |
CBTNARFZVOPLBO
|
7.4 | IC50 | 8 | — | |
KTWBYGUSEYSRND
|
7.4 | Ki | 28 | — | |
PCQMERRARZKTPW
|
7.4 | Ki | 68 | — | |
RFBPWKMQWSIPEO
|
7.4 | Ki | 28 | — | |
RQJIDUOCLNMUHR
|
7.4 | Ki | 15 | — | |
UQRGNUXIYRRBER
|
7.4 | IC50 | 6 | — | |
VJSOYRZFTRFBFM
|
7.4 | IC50 | 5 | — | |
XPHWIERLJBFPFV
|
7.4 | Ki | 69 | — | |
XUFLBSMTYMFOQH
|
7.4 | Ki | 43 | — | |
YDGTUAFFLKCKEE
|
7.4 | IC50 | 3 | — | |
FKRHOHUJMCOWDZ
|
7.4 | IC50 | 5 | — | |
QDNBLKZVYODRLC
|
7.4 | IC50 | 5 | — | |
RILDWXOQLWEXDG
|
7.4 | IC50 | 6 | — | |
PEICIAVUWSXRGP
|
7.4 | IC50 | 7 | — | |
UJIAQDJKSXQLIT
|
7.4 | Kd | 38 | — | |
UHOPJKMQVDXYAV
|
7.4 | IC50 | 8 | — | |
UIARLYUEJFELEN
|
7.4 | Kd | 289 | Yes | |
FRPGBGWSLAGPND
|
7.3 | IC50 | 7 | — | |
RLTCEYSNDOXWKS
|
7.3 | IC50 | 9 | — | |
AOGIFFVMTGMFBP
|
7.3 | IC50 | 8 | — | |
DSSNAGYVGTYAGH
|
7.3 | IC50 | 10 | — | |
XXNWOAPHJYPEGP
|
7.3 | IC50 | 2 | — | |
FFZALTJLOHVCOT
|
7.3 | IC50 | 2 | — | |
AAYFHKFUAWLHMY
|
7.3 | IC50 | 5 | — | |
CXJCGSPAPOTTSF
|
7.3 | IC50 | 6 | — | |
GCYXEGSPUDSZJY
|
7.3 | Ki | 82 | — | |
HOYRWTWZUFFACV
|
7.3 | Ki | 28 | — | |
MZQCXULGGNKLHX
|
7.3 | IC50 | 2 | — | |
PSCJSWRVCKUMSL
|
7.3 | Ki | 35 | — | |
SKKRZILJUKYLJS
|
7.3 | Ki | 25 | — | |
TWCARTFPHQNBPF
|
7.3 | Ki | 16 | — | |
YEHCNYAQEBQCCS
|
7.3 | Ki | 74 | — | |
YRFAWSIUIFNVQA
|
7.3 | IC50 | 9 | — | |
OQSBQXVIMQMCES
|
7.3 | IC50 | 9 | — | |
CEWIXDGUKGVYDQ
|
7.3 | IC50 | 7 | — | |
KNLSVEADBVICIJ
|
7.3 | IC50 | 5 | — | |
LXQXBEIFOYAXOP
|
7.2 | IC50 | 9 | — | |
CIICGXXZCWRFQE
|
7.2 | IC50 | 7 | — |