Target Details
| UniProt AC | P49760 |
|---|---|
| Gene Symbol | CLK2 |
| Protein Name | Dual specificity protein kinase CLK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 806
- Clinical molecules 29
- Avg pChEMBL 6.95
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QHTJZFWEQYRYQE
|
7.6 | IC50 | 9 | — | |
AGTMKVKIEQKSLY
|
7.6 | IC50 | 5 | — | |
KLYOYEDXPDCWAL
|
7.6 | IC50 | 5 | — | |
RJZDECGDCKOHBV
|
7.6 | Ki | 70 | — | |
SGHXFHRRWFLILP
|
7.6 | Ki | 29 | — | |
XXSPHNFKLDJDAK
|
7.6 | Ki | 26 | — | |
XZONYYFHQICDAM
|
7.6 | Ki | 19 | — | |
DLDXMINZRQNSDI
|
7.6 | IC50 | 3 | — | |
JPJBCKSRGYPABG
|
7.6 | IC50 | 3 | — | |
SLKJEEPATPIULR
|
7.6 | IC50 | 2 | — | |
ZYDSDRZMIWGATN
|
7.6 | IC50 | 3 | — | |
FIVWKNZKXNNFCW
|
7.6 | IC50 | 9 | — | |
JEPGNFQKCRZPHJ
|
7.6 | IC50 | 3 | — | |
XYFHSCKRPLMJIO
|
7.6 | IC50 | 3 | — | |
DCJOTKUJWJFCSP
|
7.5 | IC50 | 9 | — | |
FEZCHKAGMYXVNX
|
7.5 | IC50 | 6 | — | |
GPXCDUCDIFDAGL
|
7.5 | IC50 | 3 | — | |
JBWDTSLHUJHODF
|
7.5 | IC50 | 9 | — | |
KCTCLVINURCCIL
|
7.5 | IC50 | 7 | — | |
YGXHQYJKJUFSJI
|
7.5 | IC50 | 14 | — | |
GFUQINLLDUOCSK
|
7.5 | IC50 | 3 | — | |
XLHTXXNIKXXVAS
|
7.5 | IC50 | 2 | — | |
FGBSSPMQGRUJPS
|
7.5 | IC50 | 10 | — | |
OKBNCPDNYVDCTG
|
7.5 | IC50 | 5 | — | |
ONZFJXAFBPQUIU
|
7.5 | IC50 | 2 | — | |
BHKVSOQUPYXVRZ
|
7.5 | IC50 | 6 | — | |
RVYFLJXKEYHVBR
|
7.5 | IC50 | 5 | — | |
CNQGNADBGYCKKV
|
7.5 | Ki | 25 | — | |
CYLGCMABIBXHIQ
|
7.5 | Ki | 16 | — | |
FLEAYYMORDPWAJ
|
7.5 | Ki | 90 | — | |
HSMUWLLZAZCLHF
|
7.5 | Ki | 25 | — | |
JJTYLBBKGQOISV
|
7.5 | Ki | 15 | — | |
UYGYYOIUVFMGKQ
|
7.5 | Ki | 30 | — | |
WHPORTUXBLFUPA
|
7.5 | IC50 | 9 | — | |
WHVFDYQCAMPLMS
|
7.5 | Ki | 20 | Yes | |
RYBNARZBIXTFJS
|
7.5 | IC50 | 9 | — | |
CGRDYMCBGXJNLR
|
7.5 | IC50 | 9 | — | |
CHQYAWLKOUOTQO
|
7.5 | IC50 | 20 | — | |
FIVWKNZKXNNFCW
|
7.5 | IC50 | 8 | — | |
FPWXVWZFQXQWTH
|
7.5 | IC50 | 6 | — | |
IJFKKIMDRSZOOW
|
7.5 | IC50 | 9 | — | |
IWKDQQIVXBSVBE
|
7.5 | IC50 | 3 | — | |
RYBNARZBIXTFJS
|
7.5 | IC50 | 9 | — | |
YYSXUOHHBBMQMJ
|
7.5 | IC50 | 7 | — | |
DLDXMINZRQNSDI
|
7.5 | IC50 | 3 | — | |
CQVPRKIEJBHBLO
|
7.5 | IC50 | 2 | — | |
YAXGFAAKCUOWNM
|
7.5 | IC50 | 9 | — | |
GJYVLTPTDBQQCY
|
7.4 | IC50 | 7 | — | |
NMUDZNRXZXDYEQ
|
7.4 | IC50 | 9 | — | |
VWCSZVWZRTZNCH
|
7.4 | Kd | 8 | — |