Target Details
| UniProt AC | P49760 |
|---|---|
| Gene Symbol | CLK2 |
| Protein Name | Dual specificity protein kinase CLK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 806
- Clinical molecules 29
- Avg pChEMBL 6.95
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZYDSDRZMIWGATN
|
7.8 | IC50 | 3 | — | |
YRFOQHHFWYWAST
|
7.8 | IC50 | 22 | — | |
DXVSNYWBRDTHFF
|
7.8 | IC50 | 10 | — | |
IEFFSHLHNYVSEF
|
7.8 | IC50 | 8 | — | |
OYDWEMSWMQKSLK
|
7.8 | IC50 | 8 | — | |
YORVMWUGDVGXOQ
|
7.8 | IC50 | 8 | — | |
CHADTINFLWZSKR
|
7.8 | Ki | 26 | — | |
HZTYDQRUAWIZRE
|
7.8 | Kd | 40 | Yes | |
JPJBCKSRGYPABG
|
7.8 | IC50 | 3 | — | |
LCHCSKHPVCDXAU
|
7.8 | Ki | 30 | — | |
LPILBMJJRGTKOQ
|
7.8 | Ki | 27 | — | |
LSLPDHNUWRDOGC
|
7.8 | Ki | 25 | — | |
MEZZCEDCBNWCRR
|
7.8 | IC50 | 7 | — | |
MVJMMLFMPWITEJ
|
7.8 | Ki | 110 | — | |
PLHUMPJXRHMFFR
|
7.8 | Ki | 28 | — | |
SBFPHSVZEXSHTL
|
7.8 | Ki | 62 | — | |
SJWUVVGOTOMGOH
|
7.8 | IC50 | 9 | — | |
URNZTLZSAVLTIZ
|
7.8 | Ki | 26 | — | |
XQQYRDDJENLAME
|
7.8 | IC50 | 8 | — | |
ZGGIYFOLDBTZIL
|
7.8 | Ki | 27 | — | |
QTRZNDLLYHSJSH
|
7.8 | IC50 | 9 | — | |
SBYPANVVFZBWDF
|
7.8 | IC50 | 9 | — | |
UMYSGMXAOXMMGG
|
7.8 | IC50 | 7 | — | |
ZYFRJAWGLQYBTJ
|
7.8 | IC50 | 3 | — | |
YSMNHYFBBOMUFX
|
7.8 | Kd | 3 | — | |
XLSYZSRXVVCHLS
|
7.8 | Kd | 48 | — | |
YSBCFQVEEKUZSU
|
7.7 | IC50 | 9 | — | |
BGVLELSCIHASRV
|
7.7 | Kd | 12 | — | |
GEJSQZULGDKBQV
|
7.7 | IC50 | 8 | — | |
HHUOQHKKRABAQB
|
7.7 | IC50 | 5 | — | |
HEAGNKNMQVIVMM
|
7.7 | IC50 | 8 | — | |
HKSZLNNOFSGOKW
|
7.7 | Ki | 118 | — | |
IZTPYWCVQLUFKA
|
7.7 | IC50 | 5 | — | |
JTYIDARLAQQHPP
|
7.7 | IC50 | 4 | — | |
NKDOPEFRNJXAOV
|
7.7 | IC50 | 6 | — | |
RMQRHTAARSAOHF
|
7.7 | IC50 | 5 | — | |
USYASDQVUTWEQM
|
7.7 | IC50 | 9 | — | |
WINHZLLDWRZWRT
|
7.7 | Kd | 201 | Yes | |
XNWKXXIGSPPPBH
|
7.7 | Ki | 31 | — | |
XYZNKCSDQRKAFR
|
7.7 | Ki | 53 | — | |
ACPZEELFGRNYMY
|
7.7 | IC50 | 2 | — | |
FSBMCTDYWXIBLM
|
7.7 | IC50 | 22 | — | |
JBWGGMGKNIIQGU
|
7.7 | IC50 | 5 | — | |
FFJGYBJUQCZAAY
|
7.6 | IC50 | 5 | — | |
JKIDUHXOZVXHEI
|
7.6 | IC50 | 2 | — | |
WYVDFOFDVCFARJ
|
7.6 | IC50 | 6 | — | |
DGDLNCAQWKWKOH
|
7.6 | IC50 | 2 | — | |
OVVHFDIQCYTOAS
|
7.6 | IC50 | 9 | — | |
WHPORTUXBLFUPA
|
7.6 | IC50 | 8 | — | |
YHZQZEGQCKWCLP
|
7.6 | IC50 | 9 | — |