Target Details
| UniProt AC | P49760 |
|---|---|
| Gene Symbol | CLK2 |
| Protein Name | Dual specificity protein kinase CLK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 806
- Clinical molecules 29
- Avg pChEMBL 6.95
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ADMFLILDQJSEIK
|
8.3 | Ki | 72 | — | |
CGPYAXSYKQBYKJ
|
8.3 | IC50 | 12 | — | |
DJVYXMINSBMUHH
|
8.3 | IC50 | 8 | — | |
DJVYXMINSBMUHH
|
8.3 | IC50 | 8 | — | |
HZPACYSNLOCDLW
|
8.3 | Ki | 48 | — | |
KAKGFGCTONHQJW
|
8.3 | Ki | 25 | — | |
NBTJWRPKGNQBJS
|
8.3 | IC50 | 8 | — | |
NLUPJKQOKWBWFC
|
8.3 | Ki | 69 | — | |
ORUUEFDGYYTXAF
|
8.3 | Ki | 26 | — | |
ASLGQVPNOSGBQR
|
8.3 | IC50 | 10 | — | |
HKSZLNNOFSGOKW
|
8.2 | IC50 | 408 | — | |
KXMLNXWIFJZEJN
|
8.2 | IC50 | 3 | — | |
UZIATSFXNVOVFE
|
8.2 | IC50 | 9 | — | |
XCTYEZWILVGTGO
|
8.2 | IC50 | 9 | — | |
ZYDSDRZMIWGATN
|
8.2 | IC50 | 5 | — | |
ZYDSDRZMIWGATN
|
8.2 | IC50 | 4 | — | |
DFMCXVONDDGQIY
|
8.2 | Ki | 66 | — | |
HUXYBQXJVXOMKX
|
8.2 | Kd | 28 | — | |
SJWUVVGOTOMGOH
|
8.2 | IC50 | 10 | — | |
SJWUVVGOTOMGOH
|
8.2 | IC50 | 12 | — | |
ZYFRJAWGLQYBTJ
|
8.2 | IC50 | 5 | — | |
AQDWDWAYVBQMAM
|
8.1 | IC50 | 7 | — | |
FUMCKNCUEAQHCV
|
8.1 | Ki | 103 | — | |
VTYLNQMEAHCYTE
|
8.1 | IC50 | 2 | — | |
WDARYLSSWBWVCU
|
8.1 | Ki | 49 | — | |
CWJLAVRXVFHDSJ
|
8.1 | IC50 | 13 | — | |
HKSZLNNOFSGOKW
|
8.1 | Kd | 213 | — | |
MLMUOABLNWGSQB
|
8.0 | IC50 | 3 | — | |
JXJKUINEFTUSOV
|
8.0 | IC50 | 2 | — | |
TXCAPEKRDSTPOS
|
8.0 | IC50 | 5 | — | |
CFDCGXXHXUZSNP
|
8.0 | Kd | 4 | — | |
QTRZNDLLYHSJSH
|
8.0 | IC50 | 9 | — | |
RPGZQOOZHIEPJW
|
8.0 | Kd | 18 | — | |
RPGZQOOZHIEPJW
|
8.0 | Kd | 18 | — | |
SLKCVFPEQGHNSI
|
8.0 | Ki | 29 | — | |
UDFDIIVNIYWXDM
|
8.0 | Ki | 74 | — | |
ZKLJKKASNXVQBZ
|
8.0 | Ki | 27 | — | |
ZYTFPHRVOZXPGZ
|
8.0 | Ki | 30 | — | |
FVXILEFBMIKZCO
|
8.0 | IC50 | 3 | — | |
JFDRONLMXPRQPP
|
8.0 | IC50 | 9 | — | |
JPJBCKSRGYPABG
|
8.0 | IC50 | 7 | — | |
YUKWHAZRUFATPE
|
7.9 | IC50 | 2 | — | |
CEDLXWRFEZCVEU
|
7.9 | IC50 | 2 | — | |
CALAEFSQWBJMDU
|
7.9 | Ki | 21 | — | |
GDYZFFBMSBDTAA
|
7.9 | Ki | 60 | — | |
NHAUZBMUXRGRCV
|
7.9 | IC50 | 3 | — | |
BWKADHBOXYDZFU
|
7.9 | IC50 | 10 | — | |
LYADGAGFYYXXIO
|
7.8 | IC50 | 82 | — | |
UGYUFJPHSWYELP
|
7.8 | IC50 | 8 | — | |
YJKPCYDSZXIODK
|
7.8 | IC50 | 8 | — |