Target Details
| UniProt AC | P49760 |
|---|---|
| Gene Symbol | CLK2 |
| Protein Name | Dual specificity protein kinase CLK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 806
- Clinical molecules 29
- Avg pChEMBL 6.95
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BMGQWWVMWDBQGC
|
6.1 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.1 | Kd | 91 | Yes | |
LRCUOTROWBXXMI
|
6.1 | IC50 | 2 | — | |
VDJFUWZMISVQGO
|
6.1 | IC50 | 4 | — | |
HGMCNIGKEVZHFM
|
6.1 | IC50 | 8 | — | |
KRPDWHZTPZNLAZ
|
6.1 | IC50 | 5 | — | |
TZIIUQQIFMFTRP
|
6.1 | IC50 | 2 | — | |
HWDFAHKJNADKKP
|
6.0 | IC50 | 5 | — | |
NWQZSQAVEPZDBP
|
6.0 | IC50 | 5 | — | |
VNAJSIZEQWWMNK
|
6.0 | IC50 | 2 | — | |
AYTIPFHOSNFHGV
|
6.0 | IC50 | 5 | — | |
PKEDBIGNILOTHW
|
6.0 | IC50 | 3 | — | |
PRJZUMDFBBOMPR
|
6.0 | IC50 | 2 | — | |
TWKWEBMGDALHPN
|
6.0 | IC50 | 9 | — | |
GUBJNPWVIUFSTR
|
6.0 | Kd | 103 | — | |
JXVHFVDLYKIXHT
|
6.0 | IC50 | 2 | — | |
KFSMADUCMQUOPB
|
6.0 | IC50 | 2 | — | |
RAXZSEGXMBWYQK
|
6.0 | IC50 | 21 | — | |
HHGDGVNOHBAHKJ
|
6.0 | IC50 | 2 | — | |
LRPOHOOPSDHHPW
|
6.0 | IC50 | 5 | — | |
MNTINTDTQABOKE
|
6.0 | IC50 | 4 | — | |
YDTHCIZMSQZYMR
|
6.0 | IC50 | 7 | — | |
DBXGGXLBTWZXBB
|
6.0 | Ki | 39 | — | |
DJUSDFVEBBYFFL
|
6.0 | Ki | 27 | — | |
FISNDZKRNXBCLC
|
6.0 | Ki | 6 | — | |
FPQHXFMYXQZPSV
|
6.0 | Ki | 23 | — | |
FTVFEILOOGBUKN
|
6.0 | IC50 | 2 | — | |
HAYYBYPASCDWEQ
|
6.0 | Ki | 47 | — | |
HMDPCTZKMDHQTP
|
6.0 | IC50 | 5 | — | |
HRJWTAWVFDCTGO
|
6.0 | Ki | 13 | Yes | |
HXILKBXYIZKOHV
|
6.0 | Ki | 2 | — | |
IJNGXROUMFEKDB
|
6.0 | Ki | 39 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JZTOUVBEZONDKA
|
6.0 | Ki | 80 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
LYNBNVBMAGDJRW
|
6.0 | Ki | 81 | — | |
MADCXGNPDBWPLM
|
6.0 | Ki | 25 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MFAQYJIYDMLAIM
|
6.0 | Kd | 130 | Yes | |
MHWHPWMWKYXCRJ
|
6.0 | Ki | 32 | — | |
NHFDRBXTEDBWCZ
|
6.0 | Ki | 41 | — | |
NVRXTLZYXZNATH
|
6.0 | Ki | 47 | Yes | |
NWAUBAGBGOPJLF
|
6.0 | Ki | 51 | Yes | |
OHPRWVPOPFGLJG
|
6.0 | Ki | 19 | — | |
OWDRQHVEJIYVOI
|
6.0 | Ki | 47 | — | |
PHWHNHYZZNJPLB
|
6.0 | Ki | 16 | — | |
PQNWNVWJXPSZFR
|
6.0 | Ki | 21 | — | |
WONUEZVTDVQBDC
|
6.0 | Ki | 7 | — | |
WQYUNADCLFWKGN
|
6.0 | IC50 | 5 | — | |
XBNSDTLFWKORGH
|
6.0 | Ki | 10 | — |