Target Details
| UniProt AC | P49760 |
|---|---|
| Gene Symbol | CLK2 |
| Protein Name | Dual specificity protein kinase CLK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 806
- Clinical molecules 29
- Avg pChEMBL 6.95
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LHNIIDJUOCFXAP
|
6.2 | Kd | 20 | Yes | |
PWHUGOZQQCNCHC
|
6.2 | IC50 | 2 | — | |
AQLWSCZCZJWUMZ
|
6.2 | IC50 | 6 | — | |
CHEAAIPINNRRKM
|
6.2 | IC50 | 2 | — | |
GYIWPHYGXVVJQR
|
6.2 | IC50 | 2 | — | |
MHURZKJMJCNXDR
|
6.2 | IC50 | 5 | — | |
SMVHCOBBHAPLPU
|
6.2 | IC50 | 3 | — | |
YKFHBMIPXGSMRS
|
6.2 | IC50 | 7 | — | |
YORVMWUGDVGXOQ
|
6.2 | IC50 | 8 | — | |
BKIAHCJPMJSHSQ
|
6.2 | IC50 | 6 | — | |
DGVVZCKWBRQGCX
|
6.2 | Ki | 2 | — | |
FLHJZUQGFPJXRD
|
6.2 | Ki | 12 | — | |
GHMRUNOHAHJNNA
|
6.2 | Ki | 29 | — | |
ISEDKXOMRIKZPK
|
6.2 | Ki | 13 | — | |
JAMDNXUAYUHJLJ
|
6.2 | Ki | 40 | — | |
KOHNRDPXFDZZJF
|
6.2 | Ki | 31 | — | |
NLNMWQUTXDGLJU
|
6.2 | IC50 | 5 | — | |
NSDIHUXUFJHXRA
|
6.2 | Ki | 11 | — | |
OHZYECRAEHSCIB
|
6.2 | IC50 | 2 | — | |
QEWSTOOMTBAUAG
|
6.2 | Ki | 17 | — | |
QNUKRWAIZMBVCU
|
6.2 | Ki | 46 | — | |
RYYNGWLOYLRZLK
|
6.2 | Ki | 104 | — | |
UWDBNTXEKYRMSG
|
6.2 | Ki | 26 | — | |
UWQBVYXTLXNIOO
|
6.2 | Ki | 10 | — | |
UZERBHWLKRWETL
|
6.2 | IC50 | 2 | — | |
XBDWKVLCDCUNHH
|
6.2 | Ki | 18 | — | |
XEYUDLCFZLNWLI
|
6.2 | IC50 | 2 | — | |
YGUMGYOBTNGZKS
|
6.2 | Ki | 12 | — | |
YMIJUBCSOKSFRU
|
6.2 | Ki | 87 | — | |
ZDPGLLQANLROFM
|
6.2 | Ki | 17 | — | |
CWWKTGHWIFDKSB
|
6.2 | IC50 | 6 | — | |
QKCAXXVNZDAJAD
|
6.2 | IC50 | 5 | — | |
USSKXRGFNVFHFF
|
6.2 | IC50 | 7 | — | |
XTJRKTBELWGSDN
|
6.2 | IC50 | 6 | — | |
BWUOLNXJAQPJKF
|
6.2 | IC50 | 7 | — | |
YCEAZZWLNZYSCL
|
6.2 | IC50 | 5 | — | |
COUZVMMRGYONAQ
|
6.2 | IC50 | 7 | — | |
QFBOPHGXTBOQRN
|
6.2 | Kd | 7 | — | |
YFJHJYHTHWHQSE
|
6.2 | IC50 | 2 | — | |
ZHTZVZJNJGCSJO
|
6.2 | IC50 | 7 | — | |
AMHZZMGEDQCWKL
|
6.2 | IC50 | 4 | — | |
BTIHMVBBUGXLCJ
|
6.2 | Kd | 21 | Yes | |
FFESRGFMLQEDRD
|
6.2 | IC50 | 5 | — | |
GQCAWHLYBCYTDM
|
6.2 | IC50 | 2 | — | |
GYXOBURXCQKQPD
|
6.2 | IC50 | 2 | — | |
PBJIOVQCYBRCRK
|
6.2 | IC50 | 5 | — | |
WVUNYSQLFKLYNI
|
6.2 | Kd | 46 | Yes | |
XDTNBUUASJMQJU
|
6.2 | IC50 | 2 | — | |
JONPTLGCLPUHKH
|
6.2 | Kd | 8 | — | |
COYCDCAUDJBGOV
|
6.1 | IC50 | 6 | — |