Target Details
| UniProt AC | P49760 |
|---|---|
| Gene Symbol | CLK2 |
| Protein Name | Dual specificity protein kinase CLK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 806
- Clinical molecules 29
- Avg pChEMBL 6.95
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HOLVNBCAYHKGJL
|
6.3 | IC50 | 5 | — | |
NQBZANYXIXJZEH
|
6.3 | IC50 | 2 | — | |
YQLKBWUOUBOKRE
|
6.3 | IC50 | 3 | — | |
ZCLCMLMHEMDXAK
|
6.3 | IC50 | 2 | — | |
BQYDGSNDLAZAEW
|
6.3 | Ki | 13 | — | |
BTIHMVBBUGXLCJ
|
6.3 | Ki | 7 | Yes | |
FAIHBCXQSBIRIL
|
6.3 | Ki | 22 | — | |
GJOXRIYWDHESDF
|
6.3 | Ki | 27 | — | |
GUMBHNMWKMFKRT
|
6.3 | Ki | 23 | — | |
JGKVEXCUPFIDIE
|
6.3 | Ki | 5 | — | |
JOIUJUJSHIHBDT
|
6.3 | Ki | 18 | — | |
KIUHBHFVVQQALF
|
6.3 | Ki | 9 | — | |
LXVBELDBJGYFEM
|
6.3 | Ki | 20 | — | |
NPHKXSDZIKFIRU
|
6.3 | Ki | 5 | — | |
PAIFYAZSILXLBO
|
6.3 | Ki | 26 | — | |
QONPPIZSNSSCSK
|
6.3 | Ki | 45 | Yes | |
SPYHMOFSJGTUNP
|
6.3 | Ki | 9 | — | |
UTBSBSOBZHXMHI
|
6.3 | IC50 | 4 | — | |
UYJNQQDJUOUFQJ
|
6.3 | Ki | 68 | — | |
VOAZYSSSBBQYMU
|
6.3 | Ki | 4 | — | |
WYLVFMBGPRCDQF
|
6.3 | Ki | 14 | — | |
XQVVPGYIWAGRNI
|
6.3 | Ki | 19 | — | |
XTRYJNHCUFWVJN
|
6.3 | IC50 | 2 | — | |
BYOFCPSWTJCYNJ
|
6.3 | IC50 | 2 | — | |
CIEDQRFRRJHOSA
|
6.3 | IC50 | 6 | — | |
NGWGFXYGZQEEQC
|
6.3 | IC50 | 2 | — | |
QTRZNDLLYHSJSH
|
6.3 | IC50 | 7 | — | |
SPXYVKFVIYDTRR
|
6.3 | IC50 | 2 | — | |
VANUWFIFOADNQT
|
6.3 | IC50 | 2 | — | |
VGWCJGBQHCMHNJ
|
6.3 | IC50 | 8 | — | |
VQAZMVUNBILJGW
|
6.3 | IC50 | 5 | — | |
XBOHQXULVSSBPU
|
6.3 | IC50 | 2 | — | |
XXIXFZAUCITSCM
|
6.3 | IC50 | 7 | — | |
XZCWNSGWBUAUOO
|
6.3 | IC50 | 3 | — | |
DOXJZOCIJLRFLH
|
6.3 | IC50 | 2 | — | |
LDNVJIDFNXGSGT
|
6.3 | IC50 | 6 | — | |
YGVLUDLFNRZMNT
|
6.3 | IC50 | 8 | — | |
KVCPSOPLIQVJAJ
|
6.3 | IC50 | 2 | — | |
KEXVDKQNGWPBHW
|
6.3 | IC50 | 2 | — | |
BXPGHMIGIJEWJO
|
6.2 | IC50 | 2 | — | |
OVPVHNVPZGYWDN
|
6.2 | IC50 | 2 | — | |
YVLMVVBOFKFZII
|
6.2 | IC50 | 2 | — | |
ZLDBGXKKPKKVSH
|
6.2 | IC50 | 2 | — | |
BKBQCPCLHUADAX
|
6.2 | IC50 | 2 | — | |
BUDGLAJKNWCXIM
|
6.2 | IC50 | 4 | — | |
OSWHZHVVVZAPRN
|
6.2 | IC50 | 6 | — | |
PAEFKCSDRFLRMD
|
6.2 | IC50 | 5 | — | |
RDXUXJLQXOFAJG
|
6.2 | IC50 | 4 | — | |
ATUUNJCZCOMUKD
|
6.2 | IC50 | 7 | — | |
KEJZNRXUODJMCY
|
6.2 | IC50 | 2 | — |