Target Details
| UniProt AC | P49760 |
|---|---|
| Gene Symbol | CLK2 |
| Protein Name | Dual specificity protein kinase CLK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 806
- Clinical molecules 29
- Avg pChEMBL 6.95
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GSXRCPJTNIGKSZ
|
6.4 | Ki | 43 | — | |
HBMHNAPZOMEESB
|
6.4 | IC50 | 2 | — | |
HHSVICUMCOBRPT
|
6.4 | Ki | 33 | — | |
JJGSOVIZOMZMCS
|
6.4 | Ki | 35 | — | |
LRLDYTTWQIFWBD
|
6.4 | Ki | 25 | — | |
NXNQLECPAXXYTR
|
6.4 | Ki | 29 | — | |
OADRBDVURCEKRP
|
6.4 | Ki | 44 | — | |
OSVUGUHRKMMBSE
|
6.4 | Kd | 170 | — | |
QYGMZFLXMWJYRJ
|
6.4 | Ki | 14 | — | |
RRAMBEGOYIJQHY
|
6.4 | Ki | 11 | — | |
SUULIUKTZNKMMB
|
6.4 | Ki | 10 | — | |
UFGCTWUIESUHQP
|
6.4 | IC50 | 7 | — | |
URXJBXVGNBGIJA
|
6.4 | IC50 | 9 | — | |
WUWDLXZGHZSWQZ
|
6.4 | Ki | 41 | — | |
XZWVOUQIYLZUCJ
|
6.4 | Ki | 23 | — | |
YKJSWMAVAKRUAN
|
6.4 | Ki | 19 | — | |
ZVWRFVCNQOECJS
|
6.4 | Ki | 71 | — | |
ACOQCSBMVFAWQV
|
6.4 | IC50 | 6 | — | |
CKKUHARWBUXFAW
|
6.4 | IC50 | 5 | — | |
LGCHSPYDLIKTIC
|
6.4 | IC50 | 6 | — | |
MFWFIUOCHGFKKK
|
6.4 | IC50 | 2 | — | |
OYONTEXKYJZFHA
|
6.4 | Kd | 69 | Yes | |
SRKWBNXTMZQFGN
|
6.4 | IC50 | 2 | — | |
XDJCLCLBSGGNKS
|
6.4 | IC50 | 21 | — | |
KGRWKIHBWPXUHQ
|
6.4 | IC50 | 5 | — | |
RFOWEVIHKPOKTL
|
6.4 | IC50 | 4 | — | |
ZCBUQCWBWNUWSU
|
6.4 | Kd | 59 | — | |
AXRCEOKUDYDWLF
|
6.4 | Kd | 31 | — | |
DKKAPUBGRWMMGK
|
6.4 | IC50 | 5 | — | |
RUQXGVGYNKIGJD
|
6.4 | IC50 | 6 | — | |
VPCMAPSJWQZILZ
|
6.4 | IC50 | 2 | — | |
QFKKWZVCSJUTOA
|
6.4 | IC50 | 2 | — | |
AMBKAVGTUWUVBS
|
6.3 | IC50 | 8 | — | |
KBEZZFIQPRMPRG
|
6.3 | IC50 | 5 | — | |
KCTCLVINURCCIL
|
6.3 | IC50 | 6 | — | |
MEGVZXPQKGWUAG
|
6.3 | IC50 | 2 | — | |
NZIRTWSQGCVBRE
|
6.3 | IC50 | 2 | — | |
CKDCFGNOHLPEKW
|
6.3 | IC50 | 2 | — | |
HFNKQEVNSGCOJV
|
6.3 | Kd | 65 | — | |
PGPHHJBZEGSUNE
|
6.3 | IC50 | 21 | — | |
QLSWEZZOYCDEGC
|
6.3 | IC50 | 5 | — | |
URXJBXVGNBGIJA
|
6.3 | IC50 | 5 | — | |
XMKRZXOTGFXMPH
|
6.3 | Kd | 5 | — | |
XQVVPGYIWAGRNI
|
6.3 | Kd | 34 | — | |
BEILWJKGWBDPRG
|
6.3 | IC50 | 7 | — | |
RDHCLVFMADHPEQ
|
6.3 | IC50 | 2 | — | |
CUENLDJTQKFFPA
|
6.3 | IC50 | 2 | — | |
MFLKPCAUPXBTPC
|
6.3 | IC50 | 6 | — | |
CAFIVVHIKSBSPE
|
6.3 | IC50 | 2 | — | |
FFIUILKFHSTZEP
|
6.3 | IC50 | 2 | — |