Target Details
| UniProt AC | P49760 |
|---|---|
| Gene Symbol | CLK2 |
| Protein Name | Dual specificity protein kinase CLK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 806
- Clinical molecules 29
- Avg pChEMBL 6.95
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UDOOJICAHXLHPL
|
6.5 | IC50 | 2 | — | |
UYTQWUKVIAOCJI
|
6.5 | IC50 | 2 | — | |
XTJRKTBELWGSDN
|
6.5 | IC50 | 8 | — | |
ZHELCWGHFGQNAY
|
6.5 | IC50 | 2 | — | |
ADJWQFUAOONPHD
|
6.5 | Kd | 8 | — | |
AHJRHEGDXFFMBM
|
6.5 | Ki | 28 | — | |
AOBLBPWPSKBHSI
|
6.5 | Ki | 55 | — | |
CTJAMSGCMYAVCZ
|
6.5 | Ki | 14 | — | |
GCSZJMUFYOAHFY
|
6.5 | IC50 | 8 | — | |
HEUSUIRCBWROMH
|
6.5 | Ki | 64 | — | |
KPVCGFZWGAYXMV
|
6.5 | Ki | 7 | — | |
MMMPFWNSQKXKDX
|
6.5 | Ki | 14 | — | |
NXSJMRCTGYTSTK
|
6.5 | Kd | 200 | — | |
RWEHAHIEUDLKGT
|
6.5 | Ki | 33 | — | |
WWRVEMKSOIGGCS
|
6.5 | IC50 | 5 | — | |
XCHWBXBDZRJVDP
|
6.5 | Ki | 51 | — | |
YNUMBZPWLHDVEX
|
6.5 | Ki | 6 | — | |
ZWVZORIKUNOTCS
|
6.5 | Ki | 69 | — | |
GBVJYBSBYUKDMI
|
6.5 | IC50 | 2 | — | |
JOQWRLVZVPMTGG
|
6.5 | IC50 | 2 | — | |
VQXFVWAFGKCRFO
|
6.5 | IC50 | 2 | — | |
YJMYXQDIARLBTI
|
6.5 | IC50 | 2 | — | |
TZGUAAJXHPFHGU
|
6.5 | IC50 | 2 | — | |
CTMIHQOVGICMNG
|
6.5 | IC50 | 2 | — | |
GIQDYWGEMOCDSN
|
6.5 | IC50 | 5 | — | |
LDYVHYUGOBDUMZ
|
6.5 | IC50 | 6 | — | |
MJXIIYIGVBRQNO
|
6.5 | IC50 | 4 | — | |
OYICKRPKZVEBNG
|
6.5 | IC50 | 2 | — | |
RPAZCKZIZMEAIN
|
6.5 | IC50 | 2 | — | |
YVGAYXYYCJPQMU
|
6.5 | IC50 | 2 | — | |
ICVZNFCMFZXHJG
|
6.4 | IC50 | 2 | — | |
PEVDNKUCOHNRTA
|
6.4 | IC50 | 2 | — | |
PGPHHJBZEGSUNE
|
6.4 | Kd | 17 | — | |
RSXNAOYYABIBBH
|
6.4 | IC50 | 2 | — | |
YCFRZMCRPHNZOC
|
6.4 | IC50 | 7 | — | |
YCFRZMCRPHNZOC
|
6.4 | IC50 | 6 | — | |
CHQYAWLKOUOTQO
|
6.4 | IC50 | 7 | — | |
JMVDIGHUQAXWIE
|
6.4 | IC50 | 10 | — | |
KXXOSVXRQOSRGY
|
6.4 | IC50 | 2 | — | |
LELRIWOVACJYND
|
6.4 | Kd | 5 | — | |
OEVQTWCGWDOIFZ
|
6.4 | IC50 | 6 | — | |
OGPJOAYIAOEJAM
|
6.4 | IC50 | 8 | — | |
QCTKFZKNAAEORA
|
6.4 | IC50 | 2 | — | |
RUQXGVGYNKIGJD
|
6.4 | IC50 | 7 | — | |
IJFKKIMDRSZOOW
|
6.4 | IC50 | 6 | — | |
VNRLVGZOAVIXDU
|
6.4 | IC50 | 4 | — | |
ACOQCSBMVFAWQV
|
6.4 | IC50 | 8 | — | |
CQBXPNGRORFMAH
|
6.4 | IC50 | 2 | — | |
DBKQWGCVGCVPIP
|
6.4 | Ki | 21 | — | |
DQPYZHUAILXFJI
|
6.4 | Ki | 27 | — |