Target Details
| UniProt AC | P49760 |
|---|---|
| Gene Symbol | CLK2 |
| Protein Name | Dual specificity protein kinase CLK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 806
- Clinical molecules 29
- Avg pChEMBL 6.95
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QVYXLOYBJBMXNP
|
6.7 | IC50 | 7 | — | |
IFLBFWBMAWIBBZ
|
6.7 | Kd | 7 | — | |
OEVQTWCGWDOIFZ
|
6.7 | IC50 | 7 | — | |
WQYUNADCLFWKGN
|
6.7 | IC50 | 7 | — | |
GGHCFHXCBYOKTF
|
6.6 | IC50 | 2 | — | |
JQSJAVBMIMDUFO
|
6.6 | IC50 | 4 | — | |
JXQZHHAAJMQJKU
|
6.6 | IC50 | 6 | — | |
OJAHYTKDTIYGRY
|
6.6 | IC50 | 2 | — | |
XHBVYDAKJHETMP
|
6.6 | IC50 | 24 | Yes | |
AILRADAXUVEEIR
|
6.6 | IC50 | 75 | — | |
ZYPJRFNOUPSZFL
|
6.6 | IC50 | 3 | — | |
YGVTUORKHNWPJC
|
6.6 | IC50 | 2 | — | |
BQWACEUCYSZDBQ
|
6.6 | Ki | 5 | — | |
DKXHSOUZPMHNIZ
|
6.6 | Ki | 51 | Yes | |
DNTVXDZWVOVLOD
|
6.6 | IC50 | 5 | — | |
HDEZJSLYUKYKAZ
|
6.6 | Ki | 6 | — | |
HEONRZCTDBNSAL
|
6.6 | IC50 | 2 | — | |
KAICHBSRWFIESE
|
6.6 | Ki | 14 | — | |
KCKXYZOBGBJZEG
|
6.6 | Ki | 36 | — | |
NGDNKYRUKIPCLK
|
6.6 | Ki | 12 | — | |
OWRXHGAFWZFFCW
|
6.6 | Ki | 113 | — | |
PUYIXDDMOUMMRR
|
6.6 | Ki | 27 | — | |
QATMNAAQTUISJK
|
6.6 | Ki | 13 | — | |
QNLMLEYLZSGBHP
|
6.6 | Ki | 8 | — | |
SYLTYCLPHHSEIJ
|
6.6 | Ki | 27 | — | |
UXUQVXDYXKMCGA
|
6.6 | Ki | 21 | — | |
VBIYDORVDCFKHM
|
6.6 | Ki | 13 | — | |
XSRHBCYNCKAFKS
|
6.6 | Ki | 45 | — | |
YGEWBHASCYHHKW
|
6.6 | IC50 | 2 | — | |
YRVHWCZERXVDLL
|
6.6 | Ki | 6 | — | |
NTDKLKYQUXISQG
|
6.6 | IC50 | 2 | — | |
OAUMCWJJYNUCIM
|
6.6 | IC50 | 5 | — | |
UPSNQHGCEYRORJ
|
6.6 | IC50 | 2 | — | |
ANKYADWZYKSCAJ
|
6.6 | IC50 | 7 | — | |
BCNGHEQNBDRXPI
|
6.6 | IC50 | 2 | — | |
XOBINHQHMGZFDI
|
6.6 | IC50 | 5 | — | |
GVAGYBSZWYSWEQ
|
6.6 | IC50 | 2 | — | |
MXKUOZKGRRIYDM
|
6.5 | IC50 | 2 | — | |
QCHDHJOEPUQALZ
|
6.5 | IC50 | 9 | — | |
QIYSFZUFUMZRFH
|
6.5 | IC50 | 2 | — | |
DKFCBLGIHHZPIR
|
6.5 | IC50 | 2 | — | |
DORZPJWJOBMQKC
|
6.5 | IC50 | 9 | — | |
KDKUVYLMPJIGKA
|
6.5 | Kd | 91 | Yes | |
PPZINUUIYSVIGC
|
6.5 | IC50 | 6 | — | |
KPKJNCKJNAZTGG
|
6.5 | IC50 | 2 | — | |
DGSCWEKDRWDCOB
|
6.5 | IC50 | 5 | — | |
KRIUNPBAQZGFQA
|
6.5 | Kd | 76 | — | |
LMLCQJNTDFFXBL
|
6.5 | IC50 | 2 | — | |
OHNZJKJYATYGCV
|
6.5 | IC50 | 5 | — | |
OKCYRFPVWRGQBV
|
6.5 | IC50 | 5 | — |