Target Details
| UniProt AC | P49760 |
|---|---|
| Gene Symbol | CLK2 |
| Protein Name | Dual specificity protein kinase CLK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 806
- Clinical molecules 29
- Avg pChEMBL 6.95
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PMWVYONICYRLNY
|
10.0 | Kd | 4 | — | |
IUWWRSQCDUQDEZ
|
9.6 | IC50 | 8 | — | |
IUWWRSQCDUQDEZ
|
9.6 | IC50 | 9 | — | |
QDITZBLZQQZVEE
|
9.4 | Kd | 19 | — | |
BPNUQXPIQBZCMR
|
9.3 | Kd | 83 | Yes | |
HEVBCYZPXGZFGS
|
9.2 | IC50 | 11 | — | |
NWMPVMMGSHXANZ
|
9.1 | Ki | 58 | — | |
YDPWZFPXWFTXNT
|
9.1 | IC50 | 2 | — | |
KYOPCGIPHGGWMV
|
9.1 | Kd | 7 | — | |
KHVQTEBOVFILCQ
|
9.0 | IC50 | 10 | — | |
QXFBTYPBHYOEMX
|
9.0 | IC50 | 9 | — | |
QTHCAAFKVUWAFI
|
9.0 | IC50 | 23 | — | |
UZRAEHXTBCQLPV
|
9.0 | IC50 | 5 | — | |
VEZMWMSMHXKTFY
|
8.8 | IC50 | 4 | — | |
MCYPGAGHAANYON
|
8.8 | IC50 | 3 | — | |
KRNUKEYMMFBVIP
|
8.8 | IC50 | 5 | — | |
PNQOONYTDXMPLQ
|
8.8 | IC50 | 5 | — | |
YMYOREROCXXANC
|
8.7 | IC50 | 4 | — | |
BQWWOBKMDWACGC
|
8.7 | IC50 | 8 | — | |
BUDHVVXPBGMAPV
|
8.7 | IC50 | 11 | — | |
BULHRWBHKAVJMT
|
8.7 | IC50 | 8 | — | |
BWNQBFHVFFZHMR
|
8.7 | IC50 | 10 | — | |
YEZMGVBTPDYRPO
|
8.7 | IC50 | 8 | — | |
GWFMLYGNGYNZGY
|
8.7 | IC50 | 2 | — | |
HVEXJKQESNIDLM
|
8.7 | Kd | 10 | — | |
YGZQMRHVQUGUPG
|
8.7 | IC50 | 2 | — | |
JQBMRWMXRCFFOP
|
8.6 | IC50 | 2 | — | |
RJPWVZWPESKSOM
|
8.6 | IC50 | 3 | — | |
CCGBGSFDXIBQHC
|
8.6 | IC50 | 3 | — | |
BNBGXFKXNXXHEZ
|
8.6 | IC50 | 2 | — | |
OEZBNMVDJLSIKU
|
8.6 | IC50 | 5 | — | |
VVKCXCCJTOATLV
|
8.6 | IC50 | 2 | — | |
LHQWPYOYDRVMFI
|
8.6 | Ki | 21 | — | |
BBCSUMURJUYILA
|
8.5 | IC50 | 10 | — | |
QMUKOEKTUBVPFU
|
8.5 | IC50 | 12 | — | |
SLKHMZQUNIHINK
|
8.5 | IC50 | 10 | — | |
BGYVWFZMYBWCNY
|
8.5 | Ki | 30 | — | |
YWTBGJGMTBHQTM
|
8.5 | Ki | 65 | — | |
WNMOTZHMKYYWSU
|
8.5 | IC50 | 3 | — | |
DUZMKFLMNMTYDM
|
8.5 | IC50 | 4 | — | |
IEEIUNGYFLCIKQ
|
8.5 | IC50 | 3 | — | |
MNWOBOAJPYEQBE
|
8.4 | IC50 | 2 | — | |
ACSYKUPGCXYRRO
|
8.4 | Ki | 26 | — | |
KHGPYYFCIAISBU
|
8.4 | Ki | 31 | — | |
MUOKSQABCJCOPU
|
8.4 | IC50 | 36 | — | |
ROPFCXUWNMYMSW
|
8.4 | IC50 | 10 | — | |
SKKBUBMBPCJYKW
|
8.4 | IC50 | 9 | — | |
XFWUTMHVDGPWLH
|
8.4 | Ki | 75 | — | |
FUHFNJSGFRFDJZ
|
8.4 | IC50 | 2 | — | |
NJLSVJABWRFGRL
|
8.3 | IC50 | 2 | — |