Target Details
| UniProt AC | P49759 |
|---|---|
| Gene Symbol | CLK1 |
| Protein Name | Dual specificity protein kinase CLK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 576
- Clinical molecules 18
- Avg pChEMBL 7.27
KEGG Pathways (1)
Active Molecules (576)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AOLMNCAPVYTEHC
|
6.9 | IC50 | 6 | — | |
LDNVJIDFNXGSGT
|
6.9 | IC50 | 6 | — | |
GPXCDUCDIFDAGL
|
6.9 | IC50 | 3 | — | |
WBQNJPBYOGNEQC
|
6.9 | IC50 | 5 | — | |
VBPYLWZBNRFLEM
|
6.9 | IC50 | 4 | — | |
IEEIUNGYFLCIKQ
|
6.9 | IC50 | 3 | — | |
WQYUNADCLFWKGN
|
6.9 | IC50 | 5 | — | |
BGVLELSCIHASRV
|
6.9 | Kd | 11 | — | |
KCTCLVINURCCIL
|
6.9 | IC50 | 6 | — | |
NKZBIBZXOHFILQ
|
6.9 | IC50 | 3 | — | |
OSVUGUHRKMMBSE
|
6.9 | Kd | 170 | — | |
XOBINHQHMGZFDI
|
6.9 | IC50 | 5 | — | |
ABRIIMZXUFHPCH
|
6.9 | IC50 | 5 | — | |
BYMPGMQLSBLSIU
|
6.9 | IC50 | 5 | — | |
MQSQPFAQNYDQLL
|
6.9 | IC50 | 5 | — | |
RJPWVZWPESKSOM
|
6.9 | IC50 | 3 | — | |
JGJABYQWCCWLPP
|
6.9 | IC50 | 4 | — | |
COYCDCAUDJBGOV
|
6.9 | IC50 | 6 | — | |
HRPVUZOOJOMDCC
|
6.9 | IC50 | 2 | — | |
HWXVIOGONBBTBY
|
6.9 | Kd | 27 | — | |
FANUXQYVRUHAAH
|
6.8 | IC50 | 6 | — | |
UJIAQDJKSXQLIT
|
6.8 | Kd | 38 | — | |
CSNGPDJYNPSXNA
|
6.8 | IC50 | 5 | — | |
CVDZJUNTQGTGHF
|
6.8 | IC50 | 4 | — | |
FVIUKIZPDJZQKD
|
6.8 | IC50 | 5 | — | |
VDJFUWZMISVQGO
|
6.8 | IC50 | 4 | — | |
UTBSBSOBZHXMHI
|
6.8 | IC50 | 15 | Yes | |
NGOGFTYYXHNFQH
|
6.8 | Kd | 15 | — | |
UFGCTWUIESUHQP
|
6.8 | IC50 | 7 | — | |
TYCNIAHUXCRTIA
|
6.8 | IC50 | 2 | — | |
MXIKVRCYCKFUND
|
6.8 | IC50 | 6 | — | |
BWNXEFDIXGZHPQ
|
6.8 | IC50 | 4 | — | |
BWUOLNXJAQPJKF
|
6.8 | IC50 | 7 | — | |
COUZVMMRGYONAQ
|
6.8 | IC50 | 7 | — | |
LKROTCXRJRCMTD
|
6.8 | IC50 | 4 | — | |
MLMUOABLNWGSQB
|
6.8 | IC50 | 3 | — | |
NKDOPEFRNJXAOV
|
6.8 | IC50 | 6 | — | |
OSWHZHVVVZAPRN
|
6.8 | IC50 | 6 | — | |
ZYVXTMKTGDARKR
|
6.8 | IC50 | 6 | — | |
BAUOZGQJLRLMNO
|
6.8 | IC50 | 4 | — | |
KGRWKIHBWPXUHQ
|
6.8 | IC50 | 5 | — | |
DKKAPUBGRWMMGK
|
6.7 | IC50 | 5 | — | |
OAUMCWJJYNUCIM
|
6.7 | IC50 | 5 | — | |
FFESRGFMLQEDRD
|
6.7 | IC50 | 5 | — | |
RDXUXJLQXOFAJG
|
6.7 | IC50 | 4 | — | |
HTMYPIWEXZOFDM
|
6.7 | IC50 | 4 | — | |
KOEWWBBSRQMABA
|
6.7 | IC50 | 3 | — | |
OHNZJKJYATYGCV
|
6.7 | IC50 | 5 | — | |
PWBGPHVFGDQYNG
|
6.7 | IC50 | 3 | — | |
VOXHNNQHNDOGSK
|
6.7 | IC50 | 4 | — |