Target Details
| UniProt AC | P49759 |
|---|---|
| Gene Symbol | CLK1 |
| Protein Name | Dual specificity protein kinase CLK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 576
- Clinical molecules 18
- Avg pChEMBL 7.27
KEGG Pathways (1)
Active Molecules (576)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FWVIJMBZQGDXNQ
|
7.1 | IC50 | 2 | — | |
OKCYRFPVWRGQBV
|
7.1 | IC50 | 5 | — | |
XNWRZAZVQKFHKW
|
7.1 | IC50 | 2 | — | |
YDTHCIZMSQZYMR
|
7.1 | IC50 | 7 | — | |
JPJBCKSRGYPABG
|
7.1 | IC50 | 3 | — | |
ZIKVYDDNZDVYHF
|
7.1 | IC50 | 2 | — | |
AMBKAVGTUWUVBS
|
7.1 | IC50 | 8 | — | |
CCGBGSFDXIBQHC
|
7.1 | IC50 | 3 | — | |
FUHFNJSGFRFDJZ
|
7.1 | IC50 | 2 | — | |
LDYVHYUGOBDUMZ
|
7.1 | IC50 | 6 | — | |
MPXAWSABMVLIBU
|
7.1 | IC50 | 6 | — | |
RFOWEVIHKPOKTL
|
7.1 | IC50 | 4 | — | |
FRPUHWUHZZNNOB
|
7.1 | IC50 | 5 | — | |
HGMCNIGKEVZHFM
|
7.1 | IC50 | 8 | — | |
LFAHWMOZPVCJAY
|
7.1 | Kd | 8 | — | |
ONVZMCUWBPPGDN
|
7.1 | IC50 | 4 | — | |
RWAVDFHFFDMSHX
|
7.1 | IC50 | 4 | — | |
YGZQMRHVQUGUPG
|
7.1 | IC50 | 2 | — | |
XZCWNSGWBUAUOO
|
7.1 | IC50 | 3 | — | |
AYCPARAPKDAOEN
|
7.0 | Kd | 73 | — | |
BKIAHCJPMJSHSQ
|
7.0 | IC50 | 6 | — | |
FMWMKOOUBGJSJD
|
7.0 | IC50 | 4 | — | |
IXRCZLGBPPMVSP
|
7.0 | Kd | 9 | — | |
MNTINTDTQABOKE
|
7.0 | IC50 | 4 | — | |
SJXZXKOJVKYIJT
|
7.0 | IC50 | 2 | — | |
URXJBXVGNBGIJA
|
7.0 | IC50 | 5 | — | |
BUDGLAJKNWCXIM
|
7.0 | IC50 | 4 | — | |
LRPOHOOPSDHHPW
|
7.0 | IC50 | 5 | — | |
QTRZNDLLYHSJSH
|
7.0 | IC50 | 7 | — | |
MJQUKUIDCUNAAB
|
7.0 | IC50 | 4 | — | |
NXSJMRCTGYTSTK
|
7.0 | Kd | 200 | — | |
ZFOMCSNUEHMROO
|
7.0 | IC50 | 7 | — | |
CKEWXVJUPNKAPF
|
7.0 | IC50 | 3 | — | |
UZUFLDRZLTUMAC
|
7.0 | IC50 | 3 | — | |
WNMOTZHMKYYWSU
|
7.0 | IC50 | 3 | — | |
AYTIPFHOSNFHGV
|
7.0 | IC50 | 5 | — | |
BOSSBLQXHFNQIF
|
7.0 | IC50 | 3 | — | |
CIEDQRFRRJHOSA
|
7.0 | IC50 | 6 | — | |
DUZMKFLMNMTYDM
|
7.0 | IC50 | 4 | — | |
GQVSWGAIIWEDCW
|
7.0 | IC50 | 2 | — | |
PKEDBIGNILOTHW
|
7.0 | IC50 | 3 | — | |
PRJNNPMIUGYOST
|
7.0 | IC50 | 14 | — | |
VCCCOYOXNKTQFO
|
7.0 | IC50 | 9 | — | |
GIQDYWGEMOCDSN
|
7.0 | IC50 | 5 | — | |
UMYSGMXAOXMMGG
|
7.0 | IC50 | 7 | — | |
DVZORWAPBGBTCT
|
7.0 | IC50 | 4 | — | |
QWHFOOHDGGEJAI
|
7.0 | IC50 | 3 | — | |
KRPDWHZTPZNLAZ
|
7.0 | IC50 | 5 | — | |
ODPGGGTTYSGTGO
|
7.0 | Kd | 153 | — | |
DPIAIAIQEINUNP
|
7.0 | IC50 | 4 | — |