Target Details
| UniProt AC | P49759 |
|---|---|
| Gene Symbol | CLK1 |
| Protein Name | Dual specificity protein kinase CLK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 576
- Clinical molecules 18
- Avg pChEMBL 7.27
KEGG Pathways (1)
Active Molecules (576)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FTZBKRUJACNIDE
|
7.3 | IC50 | 2 | — | |
OEVQTWCGWDOIFZ
|
7.3 | IC50 | 6 | — | |
UBUJLBVNZCRWPX
|
7.3 | IC50 | 7 | — | |
JNTIINGGIOJIMW
|
7.2 | IC50 | 4 | — | |
PGPHHJBZEGSUNE
|
7.2 | IC50 | 21 | — | |
TVUWQDLBEOZVOU
|
7.2 | IC50 | 41 | — | |
VTDMTVMKVZXVSP
|
7.2 | IC50 | 4 | — | |
ZYDSDRZMIWGATN
|
7.2 | IC50 | 3 | — | |
YVSLJAICTSVCDB
|
7.2 | IC50 | 6 | — | |
MCYPGAGHAANYON
|
7.2 | IC50 | 3 | — | |
YEFYCSKFDBXSSK
|
7.2 | IC50 | 7 | — | |
YMYOREROCXXANC
|
7.2 | IC50 | 4 | — | |
JUQUOEZMUSCAFN
|
7.2 | IC50 | 3 | — | |
AQLWSCZCZJWUMZ
|
7.2 | IC50 | 6 | — | |
CHQYAWLKOUOTQO
|
7.2 | IC50 | 5 | — | |
ACOQCSBMVFAWQV
|
7.2 | IC50 | 6 | — | |
BEILWJKGWBDPRG
|
7.2 | IC50 | 7 | — | |
CHQYAWLKOUOTQO
|
7.2 | IC50 | 7 | — | |
IEDDDZFQZKDRBJ
|
7.2 | IC50 | 9 | — | |
JCBQCDPNTUDHRX
|
7.2 | IC50 | 2 | — | |
VHKRTWNLRWRPSB
|
7.2 | IC50 | 2 | — | |
YORVMWUGDVGXOQ
|
7.2 | IC50 | 8 | — | |
YYLKKYCXAOBSRM
|
7.2 | Kd | 191 | — | |
DLDXMINZRQNSDI
|
7.2 | IC50 | 3 | — | |
IRBWROIEALHOPH
|
7.2 | IC50 | 7 | — | |
JFIBFRPEOMMHJL
|
7.2 | IC50 | 2 | — | |
JRNJNYBQQYBCLE
|
7.2 | Kd | 40 | Yes | |
NKRFEKCLNDSTNO
|
7.2 | IC50 | 2 | — | |
NLNMWQUTXDGLJU
|
7.2 | IC50 | 5 | — | |
JQSJAVBMIMDUFO
|
7.2 | IC50 | 4 | — | |
MFLKPCAUPXBTPC
|
7.2 | IC50 | 6 | — | |
OTHYGYNOCOBONC
|
7.2 | IC50 | 4 | — | |
UQRGNUXIYRRBER
|
7.2 | IC50 | 6 | — | |
IFLBFWBMAWIBBZ
|
7.2 | Kd | 7 | — | |
LELRIWOVACJYND
|
7.2 | IC50 | 5 | — | |
OTKZKCGOQJKFMT
|
7.2 | IC50 | 4 | — | |
SQWZFLMPDUSYGV
|
7.2 | IC50 | 11 | — | |
VNRLVGZOAVIXDU
|
7.2 | IC50 | 4 | — | |
FKRHOHUJMCOWDZ
|
7.2 | IC50 | 5 | — | |
GPXCDUCDIFDAGL
|
7.2 | IC50 | 3 | — | |
QCLXNOBXQUWUEW
|
7.2 | IC50 | 9 | — | |
RJTQBPCQZQSZFF
|
7.2 | Kd | 9 | — | |
SQWZFLMPDUSYGV
|
7.2 | IC50 | 8 | — | |
ZBKFRVXDYILXFJ
|
7.2 | IC50 | 6 | — | |
BXNJHAXVSOCGBA
|
7.1 | IC50 | 14 | — | |
PGPHHJBZEGSUNE
|
7.1 | IC50 | 17 | — | |
QLSWEZZOYCDEGC
|
7.1 | IC50 | 5 | — | |
JPJBCKSRGYPABG
|
7.1 | IC50 | 3 | — | |
WWRVEMKSOIGGCS
|
7.1 | IC50 | 5 | — | |
CKKUHARWBUXFAW
|
7.1 | IC50 | 5 | — |