Target Details
| UniProt AC | P49759 |
|---|---|
| Gene Symbol | CLK1 |
| Protein Name | Dual specificity protein kinase CLK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 576
- Clinical molecules 18
- Avg pChEMBL 7.27
KEGG Pathways (1)
Active Molecules (576)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FGBSSPMQGRUJPS
|
7.5 | IC50 | 10 | — | |
DBFPRZJVPTXHSY
|
7.4 | IC50 | 2 | — | |
RLTCEYSNDOXWKS
|
7.4 | IC50 | 7 | — | |
MFLKPCAUPXBTPC
|
7.4 | IC50 | 5 | — | |
OWDVXJJCVWTPPW
|
7.4 | IC50 | 8 | — | |
QFBOPHGXTBOQRN
|
7.4 | IC50 | 7 | — | |
AKTCVLPOZVXXJU
|
7.4 | IC50 | 4 | — | |
JPJBCKSRGYPABG
|
7.4 | IC50 | 7 | — | |
YGVKOSRPXIWQPQ
|
7.4 | IC50 | 4 | — | |
JXQZHHAAJMQJKU
|
7.4 | IC50 | 6 | — | |
PRCDPUXQFRMFMC
|
7.4 | IC50 | 2 | — | |
QKCAXXVNZDAJAD
|
7.4 | IC50 | 5 | — | |
CEFPPDKMUCDGCU
|
7.4 | IC50 | 3 | — | |
QNWARURWFRZNNO
|
7.4 | IC50 | 7 | — | |
YIEXHVPVWYOPCC
|
7.4 | IC50 | 3 | — | |
GJYVLTPTDBQQCY
|
7.4 | IC50 | 7 | — | |
MQJVDVMWBFSFHI
|
7.4 | IC50 | 5 | — | |
UHOPJKMQVDXYAV
|
7.4 | IC50 | 8 | — | |
NJLSVJABWRFGRL
|
7.4 | IC50 | 2 | — | |
YVQOYBIBWBAHKH
|
7.4 | Kd | 12 | — | |
ZUADZDBGZDSSAB
|
7.4 | IC50 | 5 | — | |
VWCSZVWZRTZNCH
|
7.4 | Kd | 8 | — | |
XTJRKTBELWGSDN
|
7.4 | IC50 | 8 | — | |
DGSCWEKDRWDCOB
|
7.4 | IC50 | 5 | — | |
GCSZJMUFYOAHFY
|
7.4 | IC50 | 8 | — | |
RUQXGVGYNKIGJD
|
7.4 | IC50 | 6 | — | |
WROAXSSJZFFCSV
|
7.4 | IC50 | 2 | — | |
YSBCFQVEEKUZSU
|
7.4 | IC50 | 7 | — | |
MIRUXNAUNULTKO
|
7.3 | IC50 | 2 | — | |
MJXIIYIGVBRQNO
|
7.3 | IC50 | 4 | — | |
WPPYPSPZKNAEEZ
|
7.3 | IC50 | 2 | — | |
XUAFNTGABGAVRC
|
7.3 | IC50 | 2 | — | |
ACOQCSBMVFAWQV
|
7.3 | IC50 | 8 | — | |
SMVHCOBBHAPLPU
|
7.3 | IC50 | 3 | — | |
URXJBXVGNBGIJA
|
7.3 | IC50 | 9 | — | |
VQAZMVUNBILJGW
|
7.3 | IC50 | 5 | — | |
DJVYXMINSBMUHH
|
7.3 | IC50 | 8 | — | |
DJVYXMINSBMUHH
|
7.3 | IC50 | 8 | — | |
GQIHUCLIFWOITE
|
7.3 | IC50 | 4 | — | |
QUAHGPDRFLAKAC
|
7.3 | IC50 | 2 | — | |
VGWCJGBQHCMHNJ
|
7.3 | IC50 | 8 | — | |
MXRBAJVBWGVZJI
|
7.3 | IC50 | 4 | — | |
OGXQCQYWBIOFNU
|
7.3 | IC50 | 3 | — | |
PAHHKMMVQJCPJI
|
7.3 | IC50 | 8 | — | |
XDJCLCLBSGGNKS
|
7.3 | IC50 | 21 | — | |
BZUXWEBTNNKFBN
|
7.3 | IC50 | 3 | — | |
CRVHQVJVMWGKAV
|
7.3 | IC50 | 3 | — | |
RUQXGVGYNKIGJD
|
7.3 | IC50 | 7 | — | |
XTJRKTBELWGSDN
|
7.3 | IC50 | 6 | — | |
YKFHBMIPXGSMRS
|
7.3 | IC50 | 7 | — |