Target Details
| UniProt AC | P49759 |
|---|---|
| Gene Symbol | CLK1 |
| Protein Name | Dual specificity protein kinase CLK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 576
- Clinical molecules 18
- Avg pChEMBL 7.27
KEGG Pathways (1)
Active Molecules (576)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RAQBQAXSLHDSKW
|
7.8 | IC50 | 8 | — | |
RVYFLJXKEYHVBR
|
7.8 | IC50 | 5 | — | |
UKWWUFBDIVBOBD
|
7.8 | IC50 | 5 | — | |
UZKITQOBTXEXSY
|
7.8 | IC50 | 2 | — | |
WFOMWAYINPJPDX
|
7.8 | IC50 | 9 | — | |
YAXGFAAKCUOWNM
|
7.8 | IC50 | 9 | — | |
HEONRZCTDBNSAL
|
7.7 | IC50 | 2 | — | |
IDUYBYPYFGSSPE
|
7.7 | IC50 | 2 | — | |
NMUDZNRXZXDYEQ
|
7.7 | IC50 | 9 | — | |
XQQYRDDJENLAME
|
7.7 | IC50 | 8 | — | |
GUXARCGBVPDGMI
|
7.7 | IC50 | 3 | — | |
QTHCAAFKVUWAFI
|
7.7 | IC50 | 23 | — | |
BGVLELSCIHASRV
|
7.7 | Kd | 12 | — | |
CBTNARFZVOPLBO
|
7.7 | IC50 | 8 | — | |
PMDAVRLCSZSLRH
|
7.7 | IC50 | 13 | — | |
PUGXENIKUPHCAF
|
7.7 | IC50 | 3 | — | |
XTJRKTBELWGSDN
|
7.7 | IC50 | 8 | — | |
ZYFRJAWGLQYBTJ
|
7.7 | IC50 | 5 | — | |
KKIQOEOELHJGQJ
|
7.7 | IC50 | 2 | — | |
BGVLELSCIHASRV
|
7.7 | IC50 | 12 | — | |
CXJCGSPAPOTTSF
|
7.7 | IC50 | 3 | — | |
GCUNCFYJKLSBKK
|
7.7 | IC50 | 5 | — | |
HAPIHWIYVZOFQR
|
7.7 | IC50 | 4 | — | |
KVKWXEDCCDYLBI
|
7.7 | IC50 | 3 | — | |
MGEGGAFJSKMJJD
|
7.7 | IC50 | 5 | — | |
MXEZQEFCKXVMFN
|
7.7 | IC50 | 5 | — | |
OEVQTWCGWDOIFZ
|
7.7 | IC50 | 7 | — | |
UMWJBFSPIYCGRG
|
7.7 | IC50 | 7 | — | |
VJSOYRZFTRFBFM
|
7.7 | IC50 | 5 | — | |
XQSZOOXIJIGDLV
|
7.7 | IC50 | 2 | — | |
GXCOUFPTCZUTEE
|
7.7 | IC50 | 10 | — | |
HQAFQRVIFUNAKT
|
7.7 | IC50 | 3 | — | |
HZTYDQRUAWIZRE
|
7.7 | Kd | 40 | Yes | |
MVRRAWJPZXNFMK
|
7.7 | IC50 | 6 | — | |
NNPWUWSWEGWPMQ
|
7.7 | IC50 | 8 | — | |
QCHDHJOEPUQALZ
|
7.7 | IC50 | 9 | — | |
VEZMWMSMHXKTFY
|
7.7 | IC50 | 4 | — | |
YGEWBHASCYHHKW
|
7.7 | IC50 | 2 | — | |
ZYDSDRZMIWGATN
|
7.7 | IC50 | 3 | — | |
GRHRWVRWLAIBGN
|
7.7 | IC50 | 5 | — | |
UZWDCWONPYILKI
|
7.7 | IC50 | 47 | — | |
LVSVYVPFNYRNOF
|
7.7 | IC50 | 8 | — | |
PBJIOVQCYBRCRK
|
7.7 | IC50 | 5 | — | |
RUQXGVGYNKIGJD
|
7.7 | IC50 | 9 | — | |
WINHZLLDWRZWRT
|
7.7 | Kd | 201 | Yes | |
AILRADAXUVEEIR
|
7.6 | IC50 | 75 | — | |
BBCSUMURJUYILA
|
7.6 | IC50 | 9 | — | |
FRPGBGWSLAGPND
|
7.6 | IC50 | 7 | — | |
QSGKPYRFWJINEH
|
7.6 | IC50 | 12 | — | |
UVJQEKJPAVSBTA
|
7.6 | IC50 | 8 | — |