Target Details
| UniProt AC | P49759 |
|---|---|
| Gene Symbol | CLK1 |
| Protein Name | Dual specificity protein kinase CLK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 576
- Clinical molecules 18
- Avg pChEMBL 7.27
KEGG Pathways (1)
Active Molecules (576)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IJFKKIMDRSZOOW
|
8.1 | IC50 | 9 | — | |
JBWDTSLHUJHODF
|
8.1 | IC50 | 9 | — | |
NBTJWRPKGNQBJS
|
8.1 | IC50 | 8 | — | |
SJYQOVMGZOATNK
|
8.1 | IC50 | 9 | — | |
SLKHMZQUNIHINK
|
8.1 | IC50 | 10 | — | |
HEVBCYZPXGZFGS
|
8.0 | IC50 | 11 | — | |
ZDJFIKFQLKJRBA
|
8.0 | IC50 | 4 | — | |
SDRAETFVRBBLOB
|
8.0 | IC50 | 5 | — | |
UIARLYUEJFELEN
|
8.0 | Kd | 289 | Yes | |
YQLKBWUOUBOKRE
|
8.0 | IC50 | 3 | — | |
CEWIXDGUKGVYDQ
|
8.0 | IC50 | 7 | — | |
DXVSNYWBRDTHFF
|
8.0 | IC50 | 9 | — | |
JBWDTSLHUJHODF
|
8.0 | IC50 | 9 | — | |
KHVQTEBOVFILCQ
|
8.0 | IC50 | 10 | — | |
KOZFSFOOLUUIGY
|
8.0 | Kd | 88 | Yes | |
QTRZNDLLYHSJSH
|
8.0 | IC50 | 9 | — | |
RILDWXOQLWEXDG
|
8.0 | IC50 | 6 | — | |
SKKBUBMBPCJYKW
|
8.0 | IC50 | 9 | — | |
MUOKSQABCJCOPU
|
8.0 | IC50 | 36 | — | |
BULHRWBHKAVJMT
|
8.0 | IC50 | 8 | — | |
DCJOTKUJWJFCSP
|
8.0 | IC50 | 9 | — | |
DKZYXHCYPUVGAF
|
8.0 | Kd | 112 | — | |
JEPGNFQKCRZPHJ
|
8.0 | IC50 | 3 | — | |
KCTCLVINURCCIL
|
8.0 | IC50 | 7 | — | |
LXDHFJUOCGKVAV
|
8.0 | IC50 | 5 | — | |
PPALZSWDMRGSQV
|
8.0 | IC50 | 5 | — | |
ROPFCXUWNMYMSW
|
8.0 | IC50 | 10 | — | |
RYBNARZBIXTFJS
|
8.0 | IC50 | 9 | — | |
RYBNARZBIXTFJS
|
8.0 | IC50 | 9 | — | |
VCTLOEWZYIGVBO
|
8.0 | IC50 | 12 | — | |
WFOMWAYINPJPDX
|
8.0 | IC50 | 9 | — | |
XYFHSCKRPLMJIO
|
8.0 | IC50 | 3 | — | |
CGRDYMCBGXJNLR
|
7.9 | IC50 | 9 | — | |
AOGIFFVMTGMFBP
|
7.9 | IC50 | 8 | — | |
GEJSQZULGDKBQV
|
7.9 | IC50 | 8 | — | |
QQWUGDVOUVUTOY
|
7.9 | Kd | 231 | Yes | |
WREJZZXSNOJGIW
|
7.9 | IC50 | 8 | — | |
FLWYCOJREJRWLJ
|
7.9 | IC50 | 3 | — | |
HJEKFRDOAYXXRU
|
7.9 | IC50 | 8 | — | |
BDMXFIMYKGLQAL
|
7.9 | IC50 | 9 | — | |
HMUYSTSHIXJVRO
|
7.9 | IC50 | 5 | — | |
MQRHLOPPMRFMKM
|
7.9 | IC50 | 9 | — | |
QDNBLKZVYODRLC
|
7.9 | IC50 | 5 | — | |
RYWACTNAXCMTTN
|
7.9 | IC50 | 9 | — | |
WREJZZXSNOJGIW
|
7.9 | IC50 | 9 | — | |
YHZQZEGQCKWCLP
|
7.9 | IC50 | 9 | — | |
CXJCGSPAPOTTSF
|
7.9 | IC50 | 6 | — | |
UZIATSFXNVOVFE
|
7.9 | IC50 | 9 | — | |
KBEZZFIQPRMPRG
|
7.8 | IC50 | 5 | — | |
MEZZCEDCBNWCRR
|
7.8 | IC50 | 7 | — |