Target Details
| UniProt AC | P49759 |
|---|---|
| Gene Symbol | CLK1 |
| Protein Name | Dual specificity protein kinase CLK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 576
- Clinical molecules 18
- Avg pChEMBL 7.27
KEGG Pathways (1)
Active Molecules (576)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CYUDBMRFRZUOTH
|
6.1 | IC50 | 5 | — | |
SWPXADMCNLNAGW
|
6.1 | IC50 | 10 | — | |
XUZMWHLSFXCVMG
|
6.1 | Kd | 24 | — | |
KRJRCFXYZBUBRL
|
6.1 | IC50 | 2 | — | |
JIPWXCWXQYQCQS
|
6.1 | IC50 | 4 | — | |
VURLRACCOCGFDB
|
6.1 | IC50 | 6 | — | |
UAKPWAFLNKBBFC
|
6.1 | IC50 | 2 | — | |
UTBSBSOBZHXMHI
|
6.1 | IC50 | 4 | — | |
GUBJNPWVIUFSTR
|
6.0 | Kd | 103 | — | |
MCUJGJCMGRDTIE
|
6.0 | IC50 | 2 | — | |
QASZHVBKEAXRMM
|
6.0 | IC50 | 3 | — | |
RWUAJNWQCLQAAA
|
6.0 | IC50 | 4 | — | |
MFAQYJIYDMLAIM
|
6.0 | Kd | 130 | Yes | |
ZCBUQCWBWNUWSU
|
6.0 | Kd | 59 | — | |
LGQKIASGYQMERJ
|
6.0 | IC50 | 3 | — | |
VWMJHAFYPMOMGF
|
6.0 | Kd | 15 | — | |
XQVVPGYIWAGRNI
|
6.0 | Kd | 34 | — | |
CGBKQGQXEFGPDM
|
6.0 | IC50 | 6 | — | |
FJICMLZOGOVQRG
|
6.0 | IC50 | 4 | — | |
OOLXXVMFVSTNLJ
|
6.0 | IC50 | 4 | — | |
YCEAZZWLNZYSCL
|
6.0 | IC50 | 5 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
OVPNQJVDAFNBDN
|
6.0 | Kd | 44 | Yes | |
WVUNYSQLFKLYNI
|
6.0 | Kd | 46 | Yes |