Target Details
| UniProt AC | P49759 |
|---|---|
| Gene Symbol | CLK1 |
| Protein Name | Dual specificity protein kinase CLK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 576
- Clinical molecules 18
- Avg pChEMBL 7.27
KEGG Pathways (1)
Active Molecules (576)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UTBSBSOBZHXMHI
|
6.4 | IC50 | 3 | — | |
CBTNARFZVOPLBO
|
6.4 | IC50 | 5 | — | |
IWKDQQIVXBSVBE
|
6.4 | IC50 | 3 | — | |
JMVDIGHUQAXWIE
|
6.4 | IC50 | 10 | — | |
OWCUQTMFJUAAHV
|
6.4 | IC50 | 3 | — | |
JPJBCKSRGYPABG
|
6.4 | IC50 | 3 | — | |
OUSFTKFNBAZUKL
|
6.4 | Kd | 58 | Yes | |
QKJVKBQUUQVOCF
|
6.4 | IC50 | 4 | — | |
ABDPBSXQLBJPTL
|
6.4 | IC50 | 6 | — | |
DORZPJWJOBMQKC
|
6.4 | IC50 | 9 | — | |
TWKWEBMGDALHPN
|
6.4 | IC50 | 9 | — | |
TZFBRBFUNGMUNQ
|
6.4 | IC50 | 3 | — | |
JOZUGIHTSIWTIK
|
6.3 | IC50 | 4 | — | |
AOAMCMGMDKVPBS
|
6.3 | IC50 | 2 | — | |
GIUDIYZVSXHPDJ
|
6.3 | IC50 | 2 | — | |
CWWKTGHWIFDKSB
|
6.3 | IC50 | 6 | — | |
JLUXIHDOQQZMIZ
|
6.3 | IC50 | 4 | — | |
JDUBGYFRJFOXQC
|
6.3 | Kd | 13 | — | |
KQGHLDMPONJRNE
|
6.3 | IC50 | 3 | — | |
NDCWSHMFDBDIQV
|
6.3 | IC50 | 3 | — | |
FQBRQRVXPUQKLG
|
6.3 | IC50 | 10 | — | |
IXTKPNOXAVTBCW
|
6.3 | IC50 | 4 | — | |
NHAUZBMUXRGRCV
|
6.3 | IC50 | 3 | — | |
AXRCEOKUDYDWLF
|
6.3 | Kd | 31 | — | |
HDAJDNHIBCDLQF
|
6.3 | IC50 | 14 | — | |
ZHMXXVNQAFCXKK
|
6.3 | IC50 | 15 | — | |
KXMLNXWIFJZEJN
|
6.3 | IC50 | 3 | — | |
QNMZWFNNJMGJPU
|
6.3 | IC50 | 2 | — | |
ZJVGZWWTWGRGFK
|
6.3 | IC50 | 4 | — | |
CXQHYVUVSFXTMY
|
6.3 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.3 | Kd | 149 | — | |
JMCSSDLJENEFRD
|
6.2 | IC50 | 2 | — | |
GQBQUBULFDQKBM
|
6.2 | IC50 | 4 | — | |
TUOLABPPWINYRW
|
6.2 | IC50 | 4 | — | |
NWQZSQAVEPZDBP
|
6.2 | IC50 | 5 | — | |
UBPYILGKFZZVDX
|
6.2 | Kd | 130 | Yes | |
XKLPRHHLSQBUIC
|
6.2 | IC50 | 3 | — | |
DSISPBFCWKLZEA
|
6.2 | IC50 | 3 | — | |
SEERTRJTWMFXIC
|
6.2 | IC50 | 2 | — | |
UXXQOJXBIDBUAC
|
6.2 | Kd | 21 | Yes | |
DDJAQBRJAZWAAX
|
6.2 | IC50 | 4 | — | |
HUFOZJXAKZVRNJ
|
6.2 | Kd | 10 | — | |
PKEDBIGNILOTHW
|
6.2 | IC50 | 5 | — | |
ZNOLRTPMNMPLHY
|
6.2 | Kd | 6 | — | |
KDKUVYLMPJIGKA
|
6.2 | Kd | 91 | Yes | |
CIUGVTHIGIBJMT
|
6.2 | IC50 | 5 | — | |
PIMQWRZWLQKKBJ
|
6.2 | Kd | 36 | — | |
BEFUFKXGAMLMTP
|
6.1 | IC50 | 2 | — | |
OYONTEXKYJZFHA
|
6.1 | Kd | 69 | Yes | |
JKUDSDIXIGYMFG
|
6.1 | IC50 | 4 | — |