Target Details
| UniProt AC | P49759 |
|---|---|
| Gene Symbol | CLK1 |
| Protein Name | Dual specificity protein kinase CLK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 576
- Clinical molecules 18
- Avg pChEMBL 7.27
KEGG Pathways (1)
Active Molecules (576)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ADJWQFUAOONPHD
|
6.7 | IC50 | 8 | — | |
AMHZZMGEDQCWKL
|
6.7 | IC50 | 4 | — | |
CYVGSDYVNUNREA
|
6.7 | IC50 | 5 | — | |
QKNWFPRGYBXQMF
|
6.7 | IC50 | 2 | — | |
ZHTZVZJNJGCSJO
|
6.7 | IC50 | 7 | — | |
HWDFAHKJNADKKP
|
6.7 | IC50 | 5 | — | |
RUQXGVGYNKIGJD
|
6.7 | IC50 | 4 | — | |
DNTVXDZWVOVLOD
|
6.7 | IC50 | 5 | — | |
MHPMAOLCNNEBOA
|
6.7 | IC50 | 6 | — | |
YRFAWSIUIFNVQA
|
6.7 | IC50 | 4 | — | |
DSQFWMPIQBMOJL
|
6.7 | IC50 | 5 | — | |
PKQJCYXKRNGUKQ
|
6.7 | IC50 | 6 | — | |
YDGTUAFFLKCKEE
|
6.7 | IC50 | 3 | — | |
GFUQINLLDUOCSK
|
6.7 | IC50 | 3 | — | |
SLKJEEPATPIULR
|
6.7 | IC50 | 2 | — | |
HOLVNBCAYHKGJL
|
6.6 | IC50 | 5 | — | |
MHURZKJMJCNXDR
|
6.6 | IC50 | 5 | — | |
NJETXHOGHMMTEB
|
6.6 | IC50 | 4 | — | |
AQDWDWAYVBQMAM
|
6.6 | IC50 | 7 | — | |
FVXILEFBMIKZCO
|
6.6 | IC50 | 3 | — | |
RVSPPVBZRQFLQY
|
6.6 | IC50 | 6 | — | |
FWLMVFUGMHIOAA
|
6.6 | IC50 | 26 | — | |
USSKXRGFNVFHFF
|
6.6 | IC50 | 7 | — | |
QJVXFDORJYYPAW
|
6.6 | IC50 | 4 | — | |
PHEXTCXTBBPBOL
|
6.6 | IC50 | 2 | — | |
FUSZCAJFRIHBLV
|
6.6 | IC50 | 4 | — | |
QFWQVHZBLABPSP
|
6.6 | IC50 | 3 | — | |
AHJRHEGDXFFMBM
|
6.6 | Kd | 28 | — | |
CUXJJQQRHNRQEY
|
6.6 | IC50 | 4 | — | |
HFYNRAVQEUKOFF
|
6.6 | IC50 | 3 | — | |
KIUXCHKRJQPHFK
|
6.6 | IC50 | 4 | — | |
LFSFZGXABLTIEJ
|
6.6 | IC50 | 3 | — | |
WYVDFOFDVCFARJ
|
6.6 | IC50 | 6 | — | |
ZYDSDRZMIWGATN
|
6.6 | IC50 | 3 | — | |
CQVPRKIEJBHBLO
|
6.5 | IC50 | 2 | — | |
CWJLAVRXVFHDSJ
|
6.5 | IC50 | 13 | — | |
GGYHYBCBNXKDBY
|
6.5 | IC50 | 3 | — | |
XRLNWNALNXYYBG
|
6.5 | IC50 | 2 | — | |
CJWBPPWAPHJBEQ
|
6.5 | IC50 | 6 | — | |
JBGYKRAZYDNCNV
|
6.5 | Kd | 6 | — | |
WLKJMISWXHORCR
|
6.5 | IC50 | 11 | — | |
XDVWHWQSQJFRPP
|
6.5 | IC50 | 4 | — | |
LASLZTNNTZVYMJ
|
6.5 | IC50 | 4 | — | |
NRHKUKQUEJSGMG
|
6.5 | IC50 | 3 | — | |
BMGQWWVMWDBQGC
|
6.5 | Kd | 147 | Yes | |
YGVLUDLFNRZMNT
|
6.5 | IC50 | 8 | — | |
BFZIDBAEKWSVSX
|
6.5 | IC50 | 5 | — | |
CTNPALGJUAXMMC
|
6.4 | Kd | 151 | — | |
MZDKLVOWGIOKTN
|
6.4 | Kd | 80 | — | |
HMDPCTZKMDHQTP
|
6.4 | IC50 | 5 | — |