Target Details
| UniProt AC | P49759 |
|---|---|
| Gene Symbol | CLK1 |
| Protein Name | Dual specificity protein kinase CLK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 576
- Clinical molecules 18
- Avg pChEMBL 7.27
KEGG Pathways (1)
Active Molecules (576)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MWKSRKSEWLRPBL
|
9.7 | Kd | 1075 | — | |
IEFFSHLHNYVSEF
|
9.2 | IC50 | 8 | — | |
PBVAHEBIEXXNNA
|
9.0 | IC50 | 4 | — | |
BNBGXFKXNXXHEZ
|
9.0 | IC50 | 2 | — | |
GWFMLYGNGYNZGY
|
9.0 | IC50 | 2 | — | |
VVKCXCCJTOATLV
|
9.0 | IC50 | 2 | — | |
BPNUQXPIQBZCMR
|
8.8 | Kd | 83 | Yes | |
JEIKSQPRRWEWBN
|
8.8 | IC50 | 4 | — | |
MNVPCONHWCXDES
|
8.8 | IC50 | 9 | — | |
BHKVSOQUPYXVRZ
|
8.7 | IC50 | 6 | — | |
FFJGYBJUQCZAAY
|
8.7 | IC50 | 5 | — | |
XLSYZSRXVVCHLS
|
8.7 | Kd | 48 | — | |
AAYFHKFUAWLHMY
|
8.4 | IC50 | 5 | — | |
CIICGXXZCWRFQE
|
8.4 | IC50 | 7 | — | |
JFDRONLMXPRQPP
|
8.4 | IC50 | 9 | — | |
PMWVYONICYRLNY
|
8.3 | Kd | 4 | — | |
ASLGQVPNOSGBQR
|
8.3 | IC50 | 10 | — | |
YEZMGVBTPDYRPO
|
8.3 | IC50 | 8 | — | |
YJKPCYDSZXIODK
|
8.3 | IC50 | 8 | — | |
YORVMWUGDVGXOQ
|
8.3 | IC50 | 8 | — | |
FSBMCTDYWXIBLM
|
8.3 | IC50 | 22 | — | |
BBCSUMURJUYILA
|
8.2 | IC50 | 10 | — | |
CGPYAXSYKQBYKJ
|
8.2 | IC50 | 12 | — | |
IJELDUSMVKXTCW
|
8.2 | IC50 | 2 | — | |
OYDWEMSWMQKSLK
|
8.2 | IC50 | 8 | — | |
QMUKOEKTUBVPFU
|
8.2 | IC50 | 12 | — | |
USYASDQVUTWEQM
|
8.2 | IC50 | 9 | — | |
HHUOQHKKRABAQB
|
8.2 | IC50 | 5 | — | |
DPDVVGCNUWGGRS
|
8.2 | IC50 | 10 | — | |
DXVSNYWBRDTHFF
|
8.2 | IC50 | 10 | — | |
FIVWKNZKXNNFCW
|
8.2 | IC50 | 8 | — | |
QIYXLIZWXGGKOO
|
8.2 | IC50 | 10 | — | |
QXFBTYPBHYOEMX
|
8.2 | IC50 | 9 | — | |
RJYLSCSDDDQEPD
|
8.2 | IC50 | 10 | — | |
SBZWDKFEGYDKIU
|
8.2 | IC50 | 2 | — | |
YSODDCRKIDDXKM
|
8.2 | IC50 | 9 | — | |
KYOPCGIPHGGWMV
|
8.1 | IC50 | 7 | — | |
BQWWOBKMDWACGC
|
8.1 | IC50 | 8 | — | |
BUDHVVXPBGMAPV
|
8.1 | IC50 | 11 | — | |
BWNQBFHVFFZHMR
|
8.1 | IC50 | 10 | — | |
HEAGNKNMQVIVMM
|
8.1 | IC50 | 8 | — | |
JTYIDARLAQQHPP
|
8.1 | IC50 | 4 | — | |
RMQRHTAARSAOHF
|
8.1 | IC50 | 5 | — | |
QHTJZFWEQYRYQE
|
8.1 | IC50 | 9 | — | |
YRFOQHHFWYWAST
|
8.1 | IC50 | 22 | — | |
XZXHXSATPCNXJR
|
8.1 | Kd | 165 | Yes | |
ARIOBGGRZJITQX
|
8.1 | IC50 | 24 | — | |
ATVTUVKVZSYFBE
|
8.1 | IC50 | 7 | — | |
CHQYAWLKOUOTQO
|
8.1 | IC50 | 20 | — | |
FIVWKNZKXNNFCW
|
8.1 | IC50 | 9 | — |