Target Details
| UniProt AC | P49682 |
|---|---|
| Gene Symbol | CXCR3 |
| Protein Name | C-X-C chemokine receptor type 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 246
- Clinical molecules 0
- Avg pChEMBL 6.96
KEGG Pathways (3)
Active Molecules (246)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FBQNMCMALXRQBR
|
7.1 | IC50 | 2 | — | |
MLOXODPCDBYBBP
|
7.1 | IC50 | 2 | — | |
VKUYJARRAIUUAD
|
7.1 | IC50 | 2 | — | |
YPGDFCIRWJTBDH
|
7.1 | IC50 | 2 | — | |
MNAQBXUONFDHPQ
|
7.1 | IC50 | 2 | — | |
YYSJSPQLIYPDAB
|
7.1 | IC50 | 2 | — | |
OXWRKQLUEVNIIN
|
7.1 | IC50 | 2 | — | |
TYNAETKGNMEPLS
|
7.1 | IC50 | 2 | — | |
CNXUJVGPBOPVAK
|
7.0 | IC50 | 2 | — | |
JXPUMVOZGFZTNE
|
7.0 | IC50 | 2 | — | |
VAVQXDOAGHWXRV
|
7.0 | IC50 | 2 | — | |
DGPHJNJINCRCKW
|
7.0 | IC50 | 5 | — | |
WTAHTUGESFTJSD
|
7.0 | IC50 | 2 | — | |
ZNFCDOWCJQHQST
|
7.0 | IC50 | 2 | — | |
MRYPFKGCZCOPFK
|
7.0 | IC50 | 2 | — | |
ONYUJTYQWWNCAY
|
7.0 | IC50 | 2 | — | |
ODLBTEFRHPAFAN
|
7.0 | IC50 | 2 | — | |
XMLDXJBAIQBCIA
|
7.0 | IC50 | 2 | — | |
QVDKRFQCOBHRLE
|
7.0 | IC50 | 2 | — | |
KVDXKCFLJUBKBA
|
7.0 | IC50 | 2 | — | |
YTTXMLVAKAHNID
|
7.0 | IC50 | 2 | — | |
JCAGFVJEYSJWFI
|
7.0 | IC50 | 2 | — | |
MZMYJUORJONGQJ
|
7.0 | Ki | 2 | — | |
WSZQIXJQKLWWTJ
|
7.0 | IC50 | 2 | — | |
IGWQHTIRDXXITB
|
6.9 | IC50 | 2 | — | |
MXLASYWTQOBDEQ
|
6.9 | IC50 | 2 | — | |
AJOMCHZZJNMEHT
|
6.9 | IC50 | 2 | — | |
BYNZSRRNMOCSHJ
|
6.9 | IC50 | 2 | — | |
NRQLXULGRSHBGH
|
6.9 | IC50 | 2 | — | |
PAMZWJYOPJIVKJ
|
6.9 | IC50 | 2 | — | |
HBIBUYOXTLVSCE
|
6.9 | IC50 | 2 | — | |
NPRWPPHHOHQWNK
|
6.9 | IC50 | 2 | — | |
ZBBGEASLVSVRMD
|
6.9 | IC50 | 2 | — | |
ZBQUTHQUWHAFCU
|
6.9 | IC50 | 2 | — | |
BRFOKOHQJVNCED
|
6.9 | IC50 | 2 | — | |
IKSIQQMWYSWFTD
|
6.9 | IC50 | 2 | — | |
SEQWDPKCVCIRLJ
|
6.9 | IC50 | 2 | — | |
FZTNOFZANLDOCJ
|
6.9 | IC50 | 2 | — | |
NVDMYRPSMBTQKR
|
6.9 | IC50 | 2 | — | |
OGIBJXAXIVNBKC
|
6.9 | IC50 | 2 | — | |
QFFORRJHQQNWMP
|
6.9 | IC50 | 2 | — | |
RBIAPJNHXRJYQZ
|
6.9 | IC50 | 2 | — | |
VZEBVARQHHPPMI
|
6.9 | IC50 | 2 | — | |
XHVZGAFAZKPJHQ
|
6.9 | IC50 | 2 | — | |
DAFKTUHZZXUBLN
|
6.8 | IC50 | 2 | — | |
VGODIKINXLVGDI
|
6.8 | IC50 | 2 | — | |
HRBJRJICAXJECH
|
6.8 | IC50 | 2 | — | |
MWIXMEAIQGTQEO
|
6.8 | IC50 | 2 | — | |
NTFKMMZGMLEXET
|
6.8 | IC50 | 2 | — | |
WJBFXDYRKBQOKC
|
6.8 | IC50 | 2 | — |