Target Details
| UniProt AC | P49682 |
|---|---|
| Gene Symbol | CXCR3 |
| Protein Name | C-X-C chemokine receptor type 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 246
- Clinical molecules 0
- Avg pChEMBL 6.96
KEGG Pathways (3)
Active Molecules (246)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VWSXKWXISJLOQM
|
8.9 | IC50 | 6 | — | |
YVQHSLWAWYYPCD
|
8.7 | IC50 | 2 | — | |
VSHOBSIPZJJYRP
|
8.6 | IC50 | 2 | — | |
AXOCJQGAWLLMQP
|
8.4 | IC50 | 2 | — | |
FDZFVXKCJKOSRC
|
8.3 | IC50 | 2 | — | |
IENZWNOPOBXYDA
|
8.2 | Ki | 4 | — | |
WQTKNBPCJKRYPA
|
8.1 | IC50 | 2 | — | |
NYCIVVXGRDGDMY
|
8.0 | IC50 | 2 | — | |
QFFORRJHQQNWMP
|
8.0 | IC50 | 2 | — | |
TWFPYTXAUJBOEA
|
7.9 | IC50 | 2 | — | |
CCZJAXJXLVRTOE
|
7.7 | IC50 | 2 | — | |
VZXZFKXYJZNBEH
|
7.7 | IC50 | 2 | — | |
PMHSHQROYXKTQD
|
7.7 | IC50 | 2 | — | |
YJQHILPRMXWVIB
|
7.7 | IC50 | 2 | — | |
JKXDGMZWBPPROG
|
7.6 | IC50 | 2 | — | |
TUPOCPGYUUCHPM
|
7.6 | IC50 | 2 | — | |
YTTXMLVAKAHNID
|
7.6 | IC50 | 2 | — | |
KUMMJDVNAVFTPY
|
7.6 | IC50 | 2 | — | |
LEHFCHSREMRJMI
|
7.6 | IC50 | 2 | — | |
VTAGICUPFBJLSU
|
7.5 | IC50 | 2 | — | |
DWUJCNUMUUIVJW
|
7.5 | IC50 | 2 | — | |
NTFKMMZGMLEXET
|
7.5 | IC50 | 2 | — | |
UBFQUEJRKRXITC
|
7.5 | IC50 | 2 | — | |
BDLBVAVQJIHSTG
|
7.5 | IC50 | 2 | — | |
XCIQQRKISAZMHB
|
7.5 | IC50 | 2 | — | |
ZLWWAAACJPQOFS
|
7.5 | IC50 | 2 | — | |
ZLWWAAACJPQOFS
|
7.5 | IC50 | 2 | — | |
MRFUPQLMYRTEEA
|
7.5 | IC50 | 2 | — | |
AYNOFJPXPRZEFF
|
7.5 | IC50 | 2 | — | |
CJOQSGGCLIAOJR
|
7.5 | IC50 | 2 | — | |
ZNWFCQZFDRTLLU
|
7.5 | IC50 | 2 | — | |
CIDBZTRWEVTAGN
|
7.4 | IC50 | 2 | — | |
TYNAETKGNMEPLS
|
7.4 | IC50 | 2 | — | |
MZQYPJCDZAIFRC
|
7.4 | IC50 | 2 | — | |
QFOOZQUUYROMBF
|
7.4 | IC50 | 2 | — | |
RYJPJPFFPGHUEX
|
7.4 | IC50 | 2 | — | |
ZEXUFBYOIYYCJZ
|
7.4 | IC50 | 2 | — | |
BPZDYOBYHIQUAE
|
7.4 | IC50 | 2 | — | |
VKICYGOKMFVXSW
|
7.4 | IC50 | 2 | — | |
CZAZMOQKGAJBRY
|
7.4 | IC50 | 2 | — | |
ZYFUWRCUDWMSHP
|
7.4 | IC50 | 2 | — | |
YTTXMLVAKAHNID
|
7.4 | IC50 | 2 | — | |
FTCPWMLMDAMQKY
|
7.3 | IC50 | 2 | — | |
WYHMARFYRUASMT
|
7.3 | IC50 | 2 | — | |
FZBDZRSLVNCEML
|
7.3 | IC50 | 2 | — | |
JDXLPTGJYJLRPC
|
7.3 | IC50 | 2 | — | |
OAHYZWIOGSMNLF
|
7.3 | IC50 | 2 | — | |
QIPWTYSOANVUKJ
|
7.3 | IC50 | 4 | — | |
ZZYORQSGFMFKLW
|
7.3 | IC50 | 2 | — | |
POSRUELBUNHWTK
|
7.3 | IC50 | 2 | — |