Target Details
| UniProt AC | P49354 |
|---|---|
| Gene Symbol | FNTA |
| Protein Name | Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01239 (PPTA) |
Summary
- Multi-target molecules 1,421
- Clinical molecules 1125
- Avg pChEMBL 7.75
KEGG Pathways (1)
Active Molecules (1,421)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AIFZYTDMYQYJMV
|
8.6 | pIC50 | 2 | Yes | |
BAHABGBETCGAQD
|
8.6 | IC50 | 2 | — | |
DLGBJQBKHJRAGN
|
8.6 | IC50 | 2 | — | |
GRYJAJAKPOELII
|
8.6 | IC50 | 2 | — | |
NEOIEGUWAIIVDV
|
8.6 | pIC50 | 2 | Yes | |
NJUJMRKMMSIRJG
|
8.6 | pIC50 | 2 | Yes | |
USAPKSGHDXEZDU
|
8.6 | pIC50 | 2 | Yes | |
XERHITVNXGBWSR
|
8.6 | pIC50 | 2 | Yes | |
BYAJXJYFHAJINJ
|
8.6 | pIC50 | 3 | Yes | |
BZEILLJNWWUORJ
|
8.6 | pIC50 | 2 | Yes | |
CZURMACSQFAGFQ
|
8.6 | pIC50 | 2 | Yes | |
KJOXPCYQYCFTOG
|
8.6 | pIC50 | 2 | Yes | |
PTTLMXCKVOMVSG
|
8.6 | pIC50 | 2 | Yes | |
VWNBOOIWICWEPL
|
8.6 | IC50 | 3 | — | |
DHUULRFMFRMVOC
|
8.6 | pIC50 | 2 | Yes | |
DVKDXGDRDHMPRP
|
8.6 | pIC50 | 2 | Yes | |
IJUOKQKEBKCTSC
|
8.6 | pIC50 | 2 | Yes | |
IVPSGCFSOHVCMQ
|
8.6 | pIC50 | 2 | Yes | |
NYEPLLLECMESPU
|
8.6 | IC50 | 2 | — | |
PCMGNEFMPPLRII
|
8.6 | pIC50 | 2 | Yes | |
SWMJHZDPPZYMMV
|
8.6 | pIC50 | 2 | Yes | |
XIVVAPJAZVPZQR
|
8.6 | pIC50 | 2 | Yes | |
IFXSQDDDAIKBNZ
|
8.5 | pIC50 | 2 | Yes | |
KMNYYAJYASNHCC
|
8.5 | pIC50 | 3 | Yes | |
WKAGYWLHSJYLDM
|
8.5 | pIC50 | 2 | Yes | |
WOTDIFKPTDYJBL
|
8.5 | IC50 | 2 | — | |
GKTZPBPAMFCBNI
|
8.5 | pIC50 | 2 | Yes | |
GPHWYYSELXGMGI
|
8.5 | pIC50 | 2 | Yes | |
HLZAMOBHOGVCHD
|
8.5 | pIC50 | 2 | Yes | |
JHSZMWDOIIIMSL
|
8.5 | pIC50 | 2 | Yes | |
JZRFTYGHLKQOLR
|
8.5 | pIC50 | 2 | Yes | |
KMMDHGFUBJRYRM
|
8.5 | pIC50 | 2 | Yes | |
SACRSUCIYWDREQ
|
8.5 | pIC50 | 2 | Yes | |
SFPGSGWLJOJIDY
|
8.5 | pIC50 | 2 | Yes | |
UUXJPDYOJAJQGO
|
8.5 | IC50 | 4 | — | |
LKXBYRYJOKCGTP
|
8.5 | pIC50 | 2 | Yes | |
SSJTVXWXKSIJDO
|
8.5 | pIC50 | 2 | Yes | |
VABJTMPBSQEKRT
|
8.5 | pIC50 | 2 | Yes | |
XCKIUXVZLPDAPE
|
8.5 | pIC50 | 2 | Yes | |
FISVBHHSQNPBPG
|
8.5 | pIC50 | 3 | Yes | |
BRIVIXLMMUIBJY
|
8.5 | IC50 | 2 | — | |
HUDSUDXSXHERGK
|
8.5 | IC50 | 2 | — | |
HUDSUDXSXHERGK
|
8.5 | IC50 | 2 | — | |
JRYNPHOWGSLDME
|
8.5 | IC50 | 2 | — | |
AWZZZEMGYQBBLL
|
8.5 | pIC50 | 2 | Yes | |
OGHMZBMHULTCAH
|
8.5 | pIC50 | 2 | Yes | |
OQOGBHWUNRAOOD
|
8.5 | IC50 | 2 | — | |
RWNAKQQQDZHREQ
|
8.5 | IC50 | 2 | — | |
RZBRPHGLFWWUEG
|
8.5 | pIC50 | 3 | Yes | |
TXMWWHNPHYEWNP
|
8.5 | pIC50 | 3 | Yes |