Target Details
| UniProt AC | P49354 |
|---|---|
| Gene Symbol | FNTA |
| Protein Name | Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01239 (PPTA) |
Summary
- Multi-target molecules 1,421
- Clinical molecules 1125
- Avg pChEMBL 7.75
KEGG Pathways (1)
Active Molecules (1,421)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BAHABGBETCGAQD
|
8.7 | IC50 | 2 | — | |
DJZAMXRHXDPZOJ
|
8.7 | IC50 | 2 | — | |
FPGQOPQFYFPTBS
|
8.7 | pIC50 | 2 | Yes | |
IDVLFUHLBYSGQS
|
8.7 | pIC50 | 3 | Yes | |
KPLVUGOBZAXWSW
|
8.7 | pIC50 | 2 | Yes | |
MILFHOSIWZCDMY
|
8.7 | pIC50 | 2 | Yes | |
QTWCLYHBMVRTFX
|
8.7 | pIC50 | 2 | Yes | |
RKNQPYFCXGJISA
|
8.7 | pIC50 | 2 | Yes | |
YUXOGMIOPNYIQR
|
8.7 | pIC50 | 2 | Yes | |
CIFGPLIJBYKXOG
|
8.7 | pIC50 | 2 | Yes | |
DHMTURDWPRKSOA
|
8.7 | pIC50 | 4 | Yes | |
FJEFQPVMMYHHJX
|
8.7 | pIC50 | 2 | Yes | |
JINSQACWIAVMPU
|
8.7 | IC50 | 2 | — | |
RDRLCMALXVPSHH
|
8.7 | pIC50 | 2 | Yes | |
RPSVZMJVPOGOLG
|
8.7 | pIC50 | 3 | Yes | |
BTSOBCOKYPXYPA
|
8.7 | pIC50 | 2 | Yes | |
JNUGFGAVPBYSHF
|
8.7 | pIC50 | 5 | Yes | |
JQBMSMWRNHYILW
|
8.7 | pIC50 | 3 | Yes | |
NKHVWSYSXNBDDJ
|
8.7 | IC50 | 2 | — | |
NSDUAWRPFPUQFV
|
8.7 | Kd | 2 | — | |
UUNGZSLCFUPOGA
|
8.7 | pIC50 | 3 | Yes | |
VWFJDQUYCIWHTN
|
8.7 | Kd | 4 | — | |
ZMLABZGKVVLXFI
|
8.7 | pIC50 | 2 | Yes | |
BMKLSRFMQGRZMC
|
8.7 | pIC50 | 2 | Yes | |
CWDMNHRPPUTQRX
|
8.7 | pIC50 | 2 | Yes | |
FUMOSLFZEUUPBJ
|
8.7 | pIC50 | 3 | Yes | |
IFMBONPPUMOMTJ
|
8.7 | pIC50 | 2 | Yes | |
LHVRPFUHPLSLAX
|
8.7 | pIC50 | 2 | Yes | |
OJMDOBBZTGRJTI
|
8.7 | pIC50 | 2 | Yes | |
PMTPGTRNSODWEN
|
8.7 | pIC50 | 2 | Yes | |
QDYHAAJQNSIFDZ
|
8.7 | pIC50 | 2 | Yes | |
YUFXAWQITMCWMO
|
8.7 | pIC50 | 3 | Yes | |
HCAOKPQDIXSPIN
|
8.7 | pIC50 | 2 | Yes | |
KXPIURLUHSBSHE
|
8.7 | pIC50 | 2 | Yes | |
LNGVYELZGYGYAE
|
8.7 | pIC50 | 2 | Yes | |
SMMNYIDTWGBSRQ
|
8.7 | pIC50 | 2 | Yes | |
VCUKCTLNWUDZBP
|
8.7 | pIC50 | 2 | Yes | |
AFXXVFSLJYLSOC
|
8.6 | pIC50 | 3 | Yes | |
HRHHNNZCUHMMDC
|
8.6 | pIC50 | 2 | Yes | |
LHMOVHABFVYLCF
|
8.6 | pIC50 | 2 | Yes | |
OCDYJHKSCLBYLE
|
8.6 | IC50 | 2 | — | |
OFEALQXVDCUNBG
|
8.6 | pIC50 | 3 | Yes | |
UKCWQHOIIOCHPE
|
8.6 | pIC50 | 2 | Yes | |
CEKADIOTDWYKGE
|
8.6 | pIC50 | 2 | Yes | |
MVPXMHNFAQUXRM
|
8.6 | pIC50 | 3 | Yes | |
WASCAVIAFHINFK
|
8.6 | pIC50 | 3 | Yes | |
XIVVAPJAZVPZQR
|
8.6 | pIC50 | 2 | Yes | |
XOFBXIHLMNJMOE
|
8.6 | pIC50 | 3 | Yes | |
YQYGDEQYTHPZGX
|
8.6 | pIC50 | 2 | Yes | |
ZFBLLHIHVGCQFY
|
8.6 | pIC50 | 2 | Yes |